Peringatan Keamanan

The most common adverse reactions to Anthrasil observed in >5% of healthy volunteers in clinical trials were headache, infusion site pain and swelling, nausea, and back pain.

Anthrax immune globulin human

DB09057

biotech approved

Deskripsi

Anthrax immune globulin is a human antibody given with antibiotics for the treatment of anthrax. It is derived from the plasma of humans immunized with BioThrax (adsorbed anthrax vaccine), which is then further purified. Available as the product Anthrasil (FDA), the result is a solution for slow IV infusion containing polyclonal antibodies that bind the protective antigen (PA) component of Bacillus anthracis lethal and edema toxins. This binding of antibody to PA prevents PA-mediated cellular entry of toxic factors. It is administered in combination with appropriate antibiotic therapy as the immunoglobulin itself is not known to have direct antibacterial activity against anthrax bacteria, which otherwise may continue to grow and produce anthrax toxins.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 24.3 days
Volume Distribusi 5714.8 mL
Klirens (Clearance) 174.2 mL/day

Absorpsi

Peak levels were reached immediately after infusion and then declined over the duration of study (84 days). Mean activity remained above the lower limit of quantitation (5 milliunits per mL) over the entire 84-day post-dose period for the three doses studied. Cmax was found to be 83.0 mU/mL while Tmax was found to be 0.116 days.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

601 Data
Diethylstilbestrol Diethylstilbestrol may increase the thrombogenic activities of Anthrax immune globulin human.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Anthrax immune globulin human.
Conjugated estrogens Conjugated estrogens may increase the thrombogenic activities of Anthrax immune globulin human.
Estrone Estrone may increase the thrombogenic activities of Anthrax immune globulin human.
Estradiol Estradiol may increase the thrombogenic activities of Anthrax immune globulin human.
Dienestrol Dienestrol may increase the thrombogenic activities of Anthrax immune globulin human.
Ethinylestradiol Ethinylestradiol may increase the thrombogenic activities of Anthrax immune globulin human.
Mestranol Mestranol may increase the thrombogenic activities of Anthrax immune globulin human.
Estriol Estriol may increase the thrombogenic activities of Anthrax immune globulin human.
Estrone sulfate Estrone sulfate may increase the thrombogenic activities of Anthrax immune globulin human.
Quinestrol Quinestrol may increase the thrombogenic activities of Anthrax immune globulin human.
Hexestrol Hexestrol may increase the thrombogenic activities of Anthrax immune globulin human.
Tibolone Tibolone may increase the thrombogenic activities of Anthrax immune globulin human.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Anthrax immune globulin human.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Anthrax immune globulin human.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Anthrax immune globulin human.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Anthrax immune globulin human.
Zeranol Zeranol may increase the thrombogenic activities of Anthrax immune globulin human.
Equol Equol may increase the thrombogenic activities of Anthrax immune globulin human.
Promestriene Promestriene may increase the thrombogenic activities of Anthrax immune globulin human.
Methallenestril Methallenestril may increase the thrombogenic activities of Anthrax immune globulin human.
Epimestrol Epimestrol may increase the thrombogenic activities of Anthrax immune globulin human.
Moxestrol Moxestrol may increase the thrombogenic activities of Anthrax immune globulin human.
Estradiol acetate Estradiol acetate may increase the thrombogenic activities of Anthrax immune globulin human.
Estradiol benzoate Estradiol benzoate may increase the thrombogenic activities of Anthrax immune globulin human.
Estradiol cypionate Estradiol cypionate may increase the thrombogenic activities of Anthrax immune globulin human.
Estradiol valerate Estradiol valerate may increase the thrombogenic activities of Anthrax immune globulin human.
Biochanin A Biochanin A may increase the thrombogenic activities of Anthrax immune globulin human.
Formononetin Formononetin may increase the thrombogenic activities of Anthrax immune globulin human.
Estetrol Estetrol may increase the thrombogenic activities of Anthrax immune globulin human.
Etanercept The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Etanercept.
Peginterferon alfa-2a The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Peginterferon alfa-2a.
Interferon alfa-n1 The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Interferon alfa-n1.
Interferon alfa-n3 The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Interferon alfa-n3.
Peginterferon alfa-2b The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Peginterferon alfa-2b.
Anakinra The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Anakinra.
Interferon gamma-1b The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Interferon gamma-1b.
Interferon alfa-2a The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Interferon alfa-2a.
Aldesleukin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Aldesleukin.
Adalimumab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Adalimumab.
Gemtuzumab ozogamicin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Gemtuzumab ozogamicin.
Pegaspargase The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Pegaspargase.
Infliximab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Infliximab.
Interferon beta-1b The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Interferon beta-1b.
Interferon alfacon-1 The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Interferon alfacon-1.
Trastuzumab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Trastuzumab.
Rituximab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Rituximab.
Basiliximab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Basiliximab.
Muromonab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Muromonab.
Ibritumomab tiuxetan The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Ibritumomab tiuxetan.
Tositumomab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Tositumomab.
Alemtuzumab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Alemtuzumab.
Cyclosporine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Cyclosporine.
Alefacept The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Alefacept.
Efalizumab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Efalizumab.
Antithymocyte immunoglobulin (rabbit) The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Antithymocyte immunoglobulin (rabbit).
Interferon alfa-2b The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Interferon alfa-2b.
Natalizumab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Natalizumab.
Daclizumab The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Daclizumab.
Phenylalanine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Phenylalanine.
Bortezomib The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Bortezomib.
Cladribine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Cladribine.
Carmustine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Carmustine.
Amsacrine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Amsacrine.
Bleomycin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Bleomycin.
Chlorambucil The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Chlorambucil.
Raltitrexed The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Raltitrexed.
Mitomycin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Mitomycin.
Bexarotene The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Bexarotene.
Vindesine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Vindesine.
Floxuridine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Floxuridine.
Indomethacin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Indomethacin.
Tioguanine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Tioguanine.
Vinorelbine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Vinorelbine.
Dexrazoxane The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Dexrazoxane.
Sorafenib The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Sorafenib.
Streptozocin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Streptozocin.
Trifluridine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Trifluridine.
Gemcitabine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Gemcitabine.
Teniposide The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Teniposide.
Epirubicin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Epirubicin.
Chloramphenicol The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Chloramphenicol.
Lenalidomide The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Lenalidomide.
Altretamine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Altretamine.
Zidovudine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Zidovudine.
Cisplatin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Cisplatin.
Oxaliplatin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Oxaliplatin.
Cyclophosphamide The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Cyclophosphamide.
Vincristine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Vincristine.
Fluorouracil The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Fluorouracil.
Propylthiouracil The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Propylthiouracil.
Pentostatin The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Pentostatin.
Methotrexate The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Methotrexate.
Carbamazepine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Carbamazepine.
Vinblastine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Vinblastine.
Linezolid The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Linezolid.
Imatinib The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Imatinib.
Clofarabine The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Clofarabine.
Pemetrexed The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Pemetrexed.
Mycophenolate mofetil The therapeutic efficacy of Anthrax immune globulin human can be decreased when used in combination with Mycophenolate mofetil.

Target Protein

Protective antigen pagA

Referensi & Sumber

Artikel (PubMed)
  • PMID: 23979731
    Mytle N, Hopkins RJ, Malkevich NV, Basu S, Meister GT, Sanford DC, Comer JE, Van Zandt KE, Al-Ibrahim M, Kramer WG, Howard C, Daczkowski N, Chakrabarti AC, Ionin B, Nabors GS, Skiadopoulos MH: Evaluation of intravenous anthrax immune globulin for treatment of inhalation anthrax. Antimicrob Agents Chemother. 2013 Nov;57(11):5684-92. doi: 10.1128/AAC.00458-13. Epub 2013 Aug 26.

Contoh Produk & Brand

Produk: 2 • International brands: 0
Produk
  • Anthrasil
    Liquid • 60 [iU]/35mL • Intravenous • US • Approved
  • Anthrasil
    Solution • 60 unit / vial • Intravenous • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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