Befunolol

DB09013

small molecule experimental

Deskripsi

Befunolol is a beta blocker introduced in 1983 by Kakenyaku Kakko. It is currently in experimental status, and is being tested for the management of open angle glaucoma.

Struktur Molekul 2D

Berat 291.347
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

24 Data
Methimazole The excretion of Befunolol can be decreased when combined with Methimazole.
Escitalopram The serum concentration of Befunolol can be increased when it is combined with Escitalopram.
Dronedarone The metabolism of Befunolol can be decreased when combined with Dronedarone.
Lasmiditan Lasmiditan may increase the bradycardic activities of Befunolol.
Givosiran The serum concentration of Befunolol can be increased when it is combined with Givosiran.
Verapamil The risk or severity of adverse effects can be increased when Verapamil is combined with Befunolol.
Ranolazine The serum concentration of Befunolol can be increased when it is combined with Ranolazine.
Formoterol Befunolol may increase the sympathomimetic activities of Formoterol.
Haloperidol The serum concentration of Befunolol can be increased when it is combined with Haloperidol.
Fluoxetine The serum concentration of Befunolol can be increased when it is combined with Fluoxetine.
Octreotide The serum concentration of the active metabolites of Octreotide can be increased when Octreotide is used in combination with Befunolol.
Ponesimod The risk or severity of bradycardia can be increased when Ponesimod is combined with Befunolol.
Estetrol The risk or severity of hyperkalemia can be increased when Befunolol is combined with Estetrol.
Fexinidazole The risk or severity of adverse effects can be increased when Befunolol is combined with Fexinidazole.
Viloxazine The metabolism of Befunolol can be decreased when combined with Viloxazine.
Imatinib The serum concentration of Befunolol can be increased when it is combined with Imatinib.
Clozapine The serum concentration of Befunolol can be increased when it is combined with Clozapine.
Clobazam The serum concentration of Befunolol can be increased when it is combined with Clobazam.
Vilanterol The therapeutic efficacy of Vilanterol can be decreased when used in combination with Befunolol.
Fedratinib The serum concentration of Befunolol can be increased when it is combined with Fedratinib.
Spironolactone The risk or severity of hyperkalemia can be increased when Befunolol is combined with Spironolactone.
Desvenlafaxine The serum concentration of Befunolol can be increased when it is combined with Desvenlafaxine.
Etrasimod The risk or severity of bradycardia can be increased when Etrasimod is combined with Befunolol.
Lacosamide The risk or severity of ventricular arrhythmias, bradycardia, and heart block can be increased when Befunolol is combined with Lacosamide.

Target Protein

Beta-1 adrenergic receptor ADRB1
Beta-2 adrenergic receptor ADRB2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 12480285
    Reichl S, Muller-Goymann CC: The use of a porcine organotypic cornea construct for permeation studies from formulations containing befunolol hydrochloride. Int J Pharm. 2003 Jan 2;250(1):191-201.

Contoh Produk & Brand

Produk: 0 • International brands: 3
International Brands
  • Bentos — Kakenyaku Kakko
  • Bentox
  • Glauconex

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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