Peringatan Keamanan

Dimetacrine may induce severe cardiac toxicity in overdose. This property is unique among the tricyclic antidepressants.

Dimetacrine

DB08996

small molecule experimental withdrawn

Deskripsi

Dimetacrine is also known as dimethacrine or acripamine. It is marketed under the names Istonil, Istonyl, Linostil, and Miroistonil. Dimetacrine is a tricyclic antidepressant (TCA) with imipramine-like effects used in Europe for the treatment of depression. Dimetacrine is no longer used in Japan.

Struktur Molekul 2D

Berat 294.4338
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Approximately 10 hours.[A7566]
Volume Distribusi The highest concentrations of dimetacrine were found at 1 hour after administration but at 3 hours in brain, heart, lung, liver, spleen, kidney, skeletal muscle and adipose tissue of testes.[A7566]
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Approximately 70% of the doses were excreted in urine and feces within 2 days after treatment.A7566

Interaksi Obat

1759 Data
Valsartan Dimetacrine may decrease the antihypertensive activities of Valsartan.
Ramipril Dimetacrine may decrease the antihypertensive activities of Ramipril.
Esmolol Dimetacrine may decrease the antihypertensive activities of Esmolol.
Betaxolol Dimetacrine may decrease the antihypertensive activities of Betaxolol.
Remikiren Dimetacrine may decrease the antihypertensive activities of Remikiren.
Guanadrel Dimetacrine may decrease the antihypertensive activities of Guanadrel.
Olmesartan Dimetacrine may decrease the antihypertensive activities of Olmesartan.
Atenolol Dimetacrine may decrease the antihypertensive activities of Atenolol.
Diltiazem Dimetacrine may decrease the antihypertensive activities of Diltiazem.
Minoxidil Dimetacrine may decrease the antihypertensive activities of Minoxidil.
Treprostinil Dimetacrine may decrease the antihypertensive activities of Treprostinil.
Amlodipine Dimetacrine may decrease the antihypertensive activities of Amlodipine.
Nimodipine Dimetacrine may decrease the antihypertensive activities of Nimodipine.
Prazosin Dimetacrine may decrease the antihypertensive activities of Prazosin.
Trandolapril Dimetacrine may decrease the antihypertensive activities of Trandolapril.
Lercanidipine Dimetacrine may decrease the antihypertensive activities of Lercanidipine.
Benazepril Dimetacrine may decrease the antihypertensive activities of Benazepril.
Bosentan Dimetacrine may decrease the antihypertensive activities of Bosentan.
Enalapril Dimetacrine may decrease the antihypertensive activities of Enalapril.
Doxazosin Dimetacrine may decrease the antihypertensive activities of Doxazosin.
Candoxatril Dimetacrine may decrease the antihypertensive activities of Candoxatril.
Losartan Dimetacrine may decrease the antihypertensive activities of Losartan.
Moexipril Dimetacrine may decrease the antihypertensive activities of Moexipril.
Nitroglycerin Dimetacrine may decrease the antihypertensive activities of Nitroglycerin.
Cryptenamine Dimetacrine may decrease the antihypertensive activities of Cryptenamine.
Candesartan cilexetil Dimetacrine may decrease the antihypertensive activities of Candesartan cilexetil.
Eprosartan Dimetacrine may decrease the antihypertensive activities of Eprosartan.
Quinapril Dimetacrine may decrease the antihypertensive activities of Quinapril.
Telmisartan Dimetacrine may decrease the antihypertensive activities of Telmisartan.
Felodipine Dimetacrine may decrease the antihypertensive activities of Felodipine.
Irbesartan Dimetacrine may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Dimetacrine may decrease the antihypertensive activities of Nitrendipine.
Deserpidine Dimetacrine may decrease the antihypertensive activities of Deserpidine.
Carvedilol Dimetacrine may decrease the antihypertensive activities of Carvedilol.
Bretylium Dimetacrine may decrease the antihypertensive activities of Bretylium.
Terazosin Dimetacrine may decrease the antihypertensive activities of Terazosin.
Acebutolol Dimetacrine may decrease the antihypertensive activities of Acebutolol.
Captopril Dimetacrine may decrease the antihypertensive activities of Captopril.
Bepridil Dimetacrine may decrease the antihypertensive activities of Bepridil.
Bevantolol Dimetacrine may decrease the antihypertensive activities of Bevantolol.
Practolol Dimetacrine may decrease the antihypertensive activities of Practolol.
Cilazapril Dimetacrine may decrease the antihypertensive activities of Cilazapril.
Saprisartan Dimetacrine may decrease the antihypertensive activities of Saprisartan.
Spirapril Dimetacrine may decrease the antihypertensive activities of Spirapril.
Mibefradil Dimetacrine may decrease the antihypertensive activities of Mibefradil.
Dexpropranolol Dimetacrine may decrease the antihypertensive activities of Dexpropranolol.
Debrisoquine Dimetacrine may decrease the antihypertensive activities of Debrisoquine.
Sitaxentan Dimetacrine may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Dimetacrine may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Dimetacrine may decrease the antihypertensive activities of Diethylnorspermine.
Nilvadipine Dimetacrine may decrease the antihypertensive activities of Nilvadipine.
Pinacidil Dimetacrine may decrease the antihypertensive activities of Pinacidil.
Bupranolol Dimetacrine may decrease the antihypertensive activities of Bupranolol.
Temocapril Dimetacrine may decrease the antihypertensive activities of Temocapril.
Riociguat Dimetacrine may decrease the antihypertensive activities of Riociguat.
Indenolol Dimetacrine may decrease the antihypertensive activities of Indenolol.
Aliskiren Dimetacrine may decrease the antihypertensive activities of Aliskiren.
Trimazosin Dimetacrine may decrease the antihypertensive activities of Trimazosin.
Lacidipine Dimetacrine may decrease the antihypertensive activities of Lacidipine.
Manidipine Dimetacrine may decrease the antihypertensive activities of Manidipine.
Niguldipine Dimetacrine may decrease the antihypertensive activities of Niguldipine.
Rauwolfia serpentina root Dimetacrine may decrease the antihypertensive activities of Rauwolfia serpentina root.
Selexipag Dimetacrine may decrease the antihypertensive activities of Selexipag.
Angiotensin 1-7 Dimetacrine may decrease the antihypertensive activities of Angiotensin 1-7.
Talinolol Dimetacrine may decrease the antihypertensive activities of Talinolol.
Imidapril Dimetacrine may decrease the antihypertensive activities of Imidapril.
BQ-123 Dimetacrine may decrease the antihypertensive activities of BQ-123.
Landiolol Dimetacrine may decrease the antihypertensive activities of Landiolol.
Dihydralazine Dimetacrine may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Dimetacrine may decrease the antihypertensive activities of Zofenopril.
Guanoxan Dimetacrine may decrease the antihypertensive activities of Guanoxan.
Delapril Dimetacrine may decrease the antihypertensive activities of Delapril.
Vincamine Dimetacrine may decrease the antihypertensive activities of Vincamine.
Linsidomine Dimetacrine may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Dimetacrine may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Dimetacrine may decrease the antihypertensive activities of Tolonidine.
Endralazine Dimetacrine may decrease the antihypertensive activities of Endralazine.
Esatenolol Dimetacrine may decrease the antihypertensive activities of Esatenolol.
Cadralazine Dimetacrine may decrease the antihypertensive activities of Cadralazine.
Cloranolol Dimetacrine may decrease the antihypertensive activities of Cloranolol.
Bietaserpine Dimetacrine may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Dimetacrine may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Dimetacrine may decrease the antihypertensive activities of Methoserpidine.
Epanolol Dimetacrine may decrease the antihypertensive activities of Epanolol.
Guanoclor Dimetacrine may decrease the antihypertensive activities of Guanoclor.
Candesartan Dimetacrine may decrease the antihypertensive activities of Candesartan.
Dexniguldipine Dimetacrine may decrease the antihypertensive activities of Dexniguldipine.
Tocopherylquinone Dimetacrine may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Dimetacrine may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Dimetacrine may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Dimetacrine may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Dimetacrine may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Dimetacrine may decrease the antihypertensive activities of Quinaprilat.
Metoprolol Dimetacrine may decrease the antihypertensive activities of Metoprolol.
Isradipine Dimetacrine may decrease the antihypertensive activities of Isradipine.
Nitroprusside Dimetacrine may decrease the antihypertensive activities of Nitroprusside.
Timolol Dimetacrine may decrease the antihypertensive activities of Timolol.
Nisoldipine Dimetacrine may decrease the antihypertensive activities of Nisoldipine.
Fosinopril Dimetacrine may decrease the antihypertensive activities of Fosinopril.
Propranolol Dimetacrine may decrease the antihypertensive activities of Propranolol.

Target Protein

Acetylcholinesterase ACHE

Referensi & Sumber

Synthesis reference: GB933875(http://worldwide.espacenet.com/publicationDetails/biblio?CC=GB&NR=933875&KC=&FT=E&locale=en_EP)
Artikel (PubMed)
  • PMID: 5312397
    Ishitani R, Saito E, Kitagawa H: The pharmacological studies on dimetacrine. I. Studies on the absorption, distribution and excretion of H3-labeled dimetacrine in the rat. Jpn J Pharmacol. 1970 Sep;20(3):432-8.

Contoh Produk & Brand

Produk: 0 • International brands: 0
Belum ada data produk/brand untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field produk/brand.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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