Peringatan Keamanan

The most frequently reported adverse reactions were rash, pain in extremity, pruritus, and somnolence.

Raxibacumab

DB08902

biotech approved

Deskripsi

Raxibacumab is a human IgG1? monoclonal antibody that binds the protective antigen (PA) component of B. anthracis toxin. Raxibacumab has a molecular weight of approximately 146 kilodaltons. Raxibacumab is produced by recombinant DNA technology in a murine cell expression system. FDA approved on December 14, 2012.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Mean terminal elimination half-lives of raxibacumab are as follows: IM dose = 15-19 days; IV dose = 16-19 days
Volume Distribusi Steady state volume of distribution exceeded plasma volume. This suggests that there is some distribution into the tissues.
Klirens (Clearance) Clearance values were much smaller than the glomerular filtration rate indicating that there is virtually no renal clearance of raxibacumab.

Absorpsi

Raxibacumab does not cross the blood-brain-barrier. When a single IV dose of 40 mg/kg was administered to healthy, male and female human subjects, the pharmacokinetic parameters are as follows: Cmax = 1020.3 ± 140.6 mcg/mL; AUCinf = 15845.8 ± 4333.5 mcg·day/mL. Bioavailability is also dependent on site of injection. When administered to the vastus lateralis, the bioavailability is 71-85%. When administered to the gluteus maximus, the bioavailability is 50-54%.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

373 Data
Diethylstilbestrol Diethylstilbestrol may increase the thrombogenic activities of Raxibacumab.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Raxibacumab.
Conjugated estrogens Conjugated estrogens may increase the thrombogenic activities of Raxibacumab.
Estrone Estrone may increase the thrombogenic activities of Raxibacumab.
Estradiol Estradiol may increase the thrombogenic activities of Raxibacumab.
Dienestrol Dienestrol may increase the thrombogenic activities of Raxibacumab.
Ethinylestradiol Ethinylestradiol may increase the thrombogenic activities of Raxibacumab.
Mestranol Mestranol may increase the thrombogenic activities of Raxibacumab.
Estriol Estriol may increase the thrombogenic activities of Raxibacumab.
Estrone sulfate Estrone sulfate may increase the thrombogenic activities of Raxibacumab.
Quinestrol Quinestrol may increase the thrombogenic activities of Raxibacumab.
Hexestrol Hexestrol may increase the thrombogenic activities of Raxibacumab.
Tibolone Tibolone may increase the thrombogenic activities of Raxibacumab.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Raxibacumab.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Raxibacumab.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Raxibacumab.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Raxibacumab.
Zeranol Zeranol may increase the thrombogenic activities of Raxibacumab.
Equol Equol may increase the thrombogenic activities of Raxibacumab.
Promestriene Promestriene may increase the thrombogenic activities of Raxibacumab.
Methallenestril Methallenestril may increase the thrombogenic activities of Raxibacumab.
Epimestrol Epimestrol may increase the thrombogenic activities of Raxibacumab.
Moxestrol Moxestrol may increase the thrombogenic activities of Raxibacumab.
Estradiol acetate Estradiol acetate may increase the thrombogenic activities of Raxibacumab.
Estradiol benzoate Estradiol benzoate may increase the thrombogenic activities of Raxibacumab.
Estradiol cypionate Estradiol cypionate may increase the thrombogenic activities of Raxibacumab.
Estradiol valerate Estradiol valerate may increase the thrombogenic activities of Raxibacumab.
Biochanin A Biochanin A may increase the thrombogenic activities of Raxibacumab.
Formononetin Formononetin may increase the thrombogenic activities of Raxibacumab.
Estetrol Estetrol may increase the thrombogenic activities of Raxibacumab.
Cetuximab The risk or severity of adverse effects can be increased when Cetuximab is combined with Raxibacumab.
Human immunoglobulin G The risk or severity of adverse effects can be increased when Human immunoglobulin G is combined with Raxibacumab.
Omalizumab The risk or severity of adverse effects can be increased when Omalizumab is combined with Raxibacumab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Raxibacumab.
Abciximab The risk or severity of adverse effects can be increased when Abciximab is combined with Raxibacumab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Raxibacumab.
Indium In-111 satumomab pendetide The risk or severity of adverse effects can be increased when Indium In-111 satumomab pendetide is combined with Raxibacumab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Raxibacumab.
Trastuzumab The risk or severity of adverse effects can be increased when Trastuzumab is combined with Raxibacumab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Raxibacumab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Raxibacumab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Raxibacumab.
Digoxin Immune Fab (Ovine) The risk or severity of adverse effects can be increased when Digoxin Immune Fab (Ovine) is combined with Raxibacumab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Raxibacumab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Raxibacumab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Raxibacumab.
Capromab pendetide The risk or severity of adverse effects can be increased when Capromab pendetide is combined with Raxibacumab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Raxibacumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Raxibacumab.
Natalizumab The risk or severity of adverse effects can be increased when Natalizumab is combined with Raxibacumab.
Palivizumab The risk or severity of adverse effects can be increased when Palivizumab is combined with Raxibacumab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Raxibacumab.
Bevacizumab The risk or severity of adverse effects can be increased when Bevacizumab is combined with Raxibacumab.
Technetium Tc-99m arcitumomab The risk or severity of adverse effects can be increased when Technetium Tc-99m arcitumomab is combined with Raxibacumab.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Raxibacumab.
Panitumumab The risk or severity of adverse effects can be increased when Panitumumab is combined with Raxibacumab.
Ranibizumab The risk or severity of adverse effects can be increased when Ranibizumab is combined with Raxibacumab.
Galiximab The risk or severity of adverse effects can be increased when Galiximab is combined with Raxibacumab.
Pexelizumab The risk or severity of adverse effects can be increased when Pexelizumab is combined with Raxibacumab.
Afelimomab The risk or severity of adverse effects can be increased when Afelimomab is combined with Raxibacumab.
Epratuzumab The risk or severity of adverse effects can be increased when Epratuzumab is combined with Raxibacumab.
Bectumomab The risk or severity of adverse effects can be increased when Bectumomab is combined with Raxibacumab.
Oregovomab The risk or severity of adverse effects can be increased when Oregovomab is combined with Raxibacumab.
IGN311 The risk or severity of adverse effects can be increased when IGN311 is combined with Raxibacumab.
Adecatumumab The risk or severity of adverse effects can be increased when Adecatumumab is combined with Raxibacumab.
Labetuzumab The risk or severity of adverse effects can be increased when Labetuzumab is combined with Raxibacumab.
Matuzumab The risk or severity of adverse effects can be increased when Matuzumab is combined with Raxibacumab.
Fontolizumab The risk or severity of adverse effects can be increased when Fontolizumab is combined with Raxibacumab.
Bavituximab The risk or severity of adverse effects can be increased when Bavituximab is combined with Raxibacumab.
CR002 The risk or severity of adverse effects can be increased when CR002 is combined with Raxibacumab.
Rozrolimupab The risk or severity of adverse effects can be increased when Rozrolimupab is combined with Raxibacumab.
Girentuximab The risk or severity of adverse effects can be increased when Girentuximab is combined with Raxibacumab.
Obiltoxaximab The risk or severity of adverse effects can be increased when Obiltoxaximab is combined with Raxibacumab.
XTL-001 The risk or severity of adverse effects can be increased when XTL-001 is combined with Raxibacumab.
NAV 1800 The risk or severity of adverse effects can be increased when NAV 1800 is combined with Raxibacumab.
Briakinumab The risk or severity of adverse effects can be increased when Briakinumab is combined with Raxibacumab.
Otelixizumab The risk or severity of adverse effects can be increased when Otelixizumab is combined with Raxibacumab.
AMG 108 The risk or severity of adverse effects can be increased when AMG 108 is combined with Raxibacumab.
Iratumumab The risk or severity of adverse effects can be increased when Iratumumab is combined with Raxibacumab.
Enokizumab The risk or severity of adverse effects can be increased when Enokizumab is combined with Raxibacumab.
Ramucirumab The risk or severity of adverse effects can be increased when Ramucirumab is combined with Raxibacumab.
Farletuzumab The risk or severity of adverse effects can be increased when Farletuzumab is combined with Raxibacumab.
Veltuzumab The risk or severity of adverse effects can be increased when Veltuzumab is combined with Raxibacumab.
Ustekinumab The risk or severity of adverse effects can be increased when Ustekinumab is combined with Raxibacumab.
Trastuzumab emtansine The risk or severity of adverse effects can be increased when Trastuzumab emtansine is combined with Raxibacumab.
PRO-542 The risk or severity of adverse effects can be increased when PRO-542 is combined with Raxibacumab.
TNX-901 The risk or severity of adverse effects can be increased when TNX-901 is combined with Raxibacumab.
Inotuzumab ozogamicin The risk or severity of adverse effects can be increased when Inotuzumab ozogamicin is combined with Raxibacumab.
RI 624 The risk or severity of adverse effects can be increased when RI 624 is combined with Raxibacumab.
Stamulumab The risk or severity of adverse effects can be increased when MYO-029 is combined with Raxibacumab.
CT-011 The risk or severity of adverse effects can be increased when CT-011 is combined with Raxibacumab.
Leronlimab The risk or severity of adverse effects can be increased when Leronlimab is combined with Raxibacumab.
Glembatumumab vedotin The risk or severity of adverse effects can be increased when Glembatumumab vedotin is combined with Raxibacumab.
Olaratumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Raxibacumab.
IPH 2101 The risk or severity of adverse effects can be increased when IPH 2101 is combined with Raxibacumab.
TB-402 The risk or severity of adverse effects can be increased when TB-402 is combined with Raxibacumab.
Caplacizumab The risk or severity of adverse effects can be increased when Caplacizumab is combined with Raxibacumab.
IMC-1C11 The risk or severity of adverse effects can be increased when IMC-1C11 is combined with Raxibacumab.
Eldelumab The risk or severity of adverse effects can be increased when Eldelumab is combined with Raxibacumab.
Lumiliximab The risk or severity of adverse effects can be increased when Lumiliximab is combined with Raxibacumab.

Target Protein

Protective antigen pagA

Referensi & Sumber

Artikel (PubMed)
  • PMID: 20068396
    Mazumdar S: Raxibacumab. MAbs. 2009 Nov-Dec;1(6):531-8. Epub 2009 Nov 29.

Contoh Produk & Brand

Produk: 5 • International brands: 1
Produk
  • Raxibacumab
    Injection • 50 mg/1mL • Intravenous • US • Approved
  • Raxibacumab
    Injection • 50 mg/1mL • Intravenous • US • Approved
  • Raxibacumab
    Injection • 50 mg/1mL • Intravenous • US • Approved
  • Raxibacumab
    Injection • 50 mg/1mL • Intravenous • US • Approved
  • Raxibacumab
    Injection • 50 mg/1mL • Intravenous • US • Approved
International Brands
  • Abthrax — Human Genome Sciences Inc.

Sekuens Gen/Protein (FASTA)

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