Peringatan Keamanan

Icosapent ethyl is generally well tolerated and adverse effects are unrelated to treatment.

Icosapent ethyl

DB08887

small molecule approved investigational nutraceutical

Deskripsi

Icosapent ethyl or ethyl eicosapentaenoic acid is a synthetic derivative of the omega-3 fatty acid eicosapentaenoic acid (EPA). It is used as an adjunct therapy for severe hypertriglyceridemia (TG levels > 500 mg/dL) and to reduce the risk of cardiovascular events in certain patients with elevated triglycerides. FDA approved on July 26, 2012.

Struktur Molekul 2D

Berat 330.5042
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The half life of EPA is 89 hours.
Volume Distribusi Steady state volume of distribution of active EPA is 88 L
Klirens (Clearance) Total plasma clearance, EPA = 684 mL/hr

Absorpsi

Icosapent ethyl is de-esterfied, converted into active EPA, and then absorbed in the small intestine. It reaches peak plasma concentration in 5 hours post-oral administration. Very little (<1%) is left circulating in the plasma as EPA incorporates into phospholipids, TG's, and cholesteryl esters.

Metabolisme

Once converted into active EPA, it is hepatically metabolized into acetyl Coenzyme A via beta-oxidation.

Rute Eliminasi

Icosapent ethyl is not renally excreted

Interaksi Makanan

1 Data
  • 1. Take with food.

Interaksi Obat

416 Data
Apixaban The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Apixaban.
Dasatinib Dasatinib may increase the anticoagulant activities of Icosapent ethyl.
Ursodeoxycholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Ursodeoxycholic acid.
Glycochenodeoxycholic Acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Glycochenodeoxycholic Acid.
Cholic Acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Cholic Acid.
Glycocholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Glycocholic acid.
Deoxycholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Deoxycholic acid.
Taurocholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Taurocholic acid.
Obeticholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Obeticholic acid.
Chenodeoxycholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Chenodeoxycholic acid.
Taurochenodeoxycholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Taurochenodeoxycholic acid.
Tauroursodeoxycholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Tauroursodeoxycholic acid.
Bamet-UD2 The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Bamet-UD2.
Dehydrocholic acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Dehydrocholic acid.
Hyodeoxycholic Acid The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Hyodeoxycholic Acid.
Glucosamine Glucosamine may increase the antiplatelet activities of Icosapent ethyl.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Ibritumomab tiuxetan.
Obinutuzumab The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the antiplatelet activities of Icosapent ethyl.
Rivaroxaban Icosapent ethyl may increase the anticoagulant activities of Rivaroxaban.
Tipranavir Tipranavir may increase the antiplatelet activities of Icosapent ethyl.
Urokinase Icosapent ethyl may increase the anticoagulant activities of Urokinase.
Ibrutinib Icosapent ethyl may increase the antiplatelet activities of Ibrutinib.
Pentosan polysulfate The risk or severity of adverse effects can be increased when Pentosan polysulfate is combined with Icosapent ethyl.
Limaprost Limaprost may increase the antiplatelet activities of Icosapent ethyl.
Omega-3 fatty acids Omega-3 fatty acids may increase the antiplatelet activities of Icosapent ethyl.
Tositumomab The risk or severity of adverse effects can be increased when Icosapent ethyl is combined with Tositumomab.
Lepirudin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Lepirudin.
Bivalirudin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Bivalirudin.
Alteplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Alteplase.
Reteplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Reteplase.
Anistreplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Anistreplase.
Tenecteplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Tenecteplase.
Abciximab The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Abciximab.
Drotrecogin alfa The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Drotrecogin alfa.
Streptokinase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Streptokinase.
Dicoumarol The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Dicoumarol.
Argatroban The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Argatroban.
Ardeparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Ardeparin.
Phenindione The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Phenindione.
Fondaparinux The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Fondaparinux.
Warfarin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Warfarin.
Phenprocoumon The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Phenprocoumon.
Dipyridamole The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Dipyridamole.
Heparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Heparin.
Enoxaparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Enoxaparin.
Epoprostenol The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Epoprostenol.
Acenocoumarol The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Coumarin.
Ximelagatran The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Ximelagatran.
Desmoteplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Desmoteplase.
Defibrotide The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Defibrotide.
Ancrod The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Ancrod.
Beraprost The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Beraprost.
Prasugrel The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Prasugrel.
Sulodexide The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Sulodexide.
Semuloparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Semuloparin.
Idraparinux The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Idraparinux.
Cangrelor The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Cangrelor.
Astaxanthin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Astaxanthin.
Otamixaban The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Otamixaban.
Amediplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Amediplase.
Danaparoid The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Danaparoid.
Dalteparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Dalteparin.
Tinzaparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Tinzaparin.
(R)-warfarin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Ethyl biscoumacetate.
Nadroparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Nadroparin.
Triflusal The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Triflusal.
Ticagrelor The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Ticagrelor.
Ditazole The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Ditazole.
Vorapaxar The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Vorapaxar.
Edoxaban The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Edoxaban.
Sodium citrate The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Sodium citrate.
Dextran The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Dextran.
Bemiparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Bemiparin.
Parnaparin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Parnaparin.
Desirudin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Desirudin.
Antithrombin Alfa The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Antithrombin Alfa.
Protein C The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Protein C.
Antithrombin III human The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Antithrombin III human.
Letaxaban The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Letaxaban.
Darexaban The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Darexaban.
Betrixaban The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Betrixaban.
Nafamostat The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Nafamostat.
Monteplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Monteplase.
Gabexate The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Gabexate.
Fluindione The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Fluindione.
Protein S human The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Protein S human.
Brinase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Brinase.
Clorindione The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Clorindione.
Diphenadione The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Diphenadione.
Tioclomarol The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Tioclomarol.
Melagatran The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Melagatran.
Saruplase The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Saruplase.
(S)-Warfarin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with (S)-Warfarin.
Tocopherylquinone The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Tocopherylquinone.
Dabigatran The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Dabigatran.
Troxerutin The risk or severity of bleeding can be increased when Icosapent ethyl is combined with Troxerutin.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 23701295
    Ballantyne CM, Braeckman RA, Soni PN: Icosapent ethyl for the treatment of hypertriglyceridemia. Expert Opin Pharmacother. 2013 Jul;14(10):1409-16. doi: 10.1517/14656566.2013.798645. Epub 2013 May 24.

Contoh Produk & Brand

Produk: 36 • International brands: 1
Produk
  • Calcium PNV
    Tablet, coated • - • Oral • US
  • Icosapent
    Capsule • 1000 mg/1 • Oral • US • Generic • Approved
  • Icosapent
    Capsule • 1000 mg/1 • Oral • US • Generic • Approved
  • Icosapent
    Capsule • 1000 mg/1 • Oral • US • Generic • Approved
  • Icosapent Ethyl
    Capsule • 1 g/1 • Oral • US • Generic • Approved
  • Icosapent Ethyl
    Capsule • 1 g/1 • Oral • US • Generic • Approved
  • Icosapent Ethyl
    Capsule • 1 g/1 • Oral • US • Generic • Approved
  • Icosapent Ethyl
    Capsule, liquid filled • 500 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 36 produk.
International Brands
  • Epadel

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