Uric acid

DB08844

small molecule investigational

Deskripsi

Uric acid is the last product of purine metabolism in humans. The formation of uric acid is through the enzyme xanthine oxidase, which oxidizes oxypurines. Normally a small amount of uric acid is present in the body, but when there is an excess amount in the blood, called hyperuricemia, this can lead to gout and formation of kidney stones. As a therapeutic agent, it is known that uric acid is increased in response to oxidative stress, and as such, uric acid acts as an antioxidant. At present (August 2013), there is no approved formulation or indication for uric acid. In one country, Spain, uric acid is an investigational drug in a phase 3 trial studying its effects as an adjunct to alteplase in acute ischemic stroke.

Struktur Molekul 2D

Berat 168.1103
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

In higher primates and humans, the enzyme, uricase, is absent, and thus uric acid is not further metabolized and is excreted. In all other mammals, uric acid is metabolized by uricase to allantoin, which is then excreted.

Rute Eliminasi

Uric acid is eliminated by the kidneys.

Interaksi Obat

370 Data
Regadenoson Uric acid may decrease effectiveness of Regadenoson as a diagnostic agent.
Adalimumab The serum concentration of Uric acid can be decreased when it is combined with Adalimumab.
Adenosine The therapeutic efficacy of Adenosine can be decreased when used in combination with Uric acid.
Allopurinol The serum concentration of Uric acid can be increased when it is combined with Allopurinol.
Carbamazepine The serum concentration of Uric acid can be decreased when it is combined with Carbamazepine.
Cimetidine The metabolism of Uric acid can be decreased when combined with Cimetidine.
Disulfiram The serum concentration of Uric acid can be increased when it is combined with Disulfiram.
Febuxostat The serum concentration of the active metabolites of Uric acid can be increased when Uric acid is used in combination with Febuxostat.
Fluvoxamine The metabolism of Uric acid can be decreased when combined with Fluvoxamine.
Formoterol The risk or severity of hypokalemia can be increased when Uric acid is combined with Formoterol.
Indacaterol The risk or severity of adverse effects can be increased when Uric acid is combined with Indacaterol.
Isoniazid The serum concentration of Uric acid can be increased when it is combined with Isoniazid.
Lithium citrate The serum concentration of Lithium citrate can be decreased when it is combined with Uric acid.
Lithium carbonate The serum concentration of Lithium carbonate can be decreased when it is combined with Uric acid.
Lithium hydroxide The serum concentration of Lithium hydroxide can be decreased when it is combined with Uric acid.
Mexiletine The metabolism of Uric acid can be decreased when combined with Mexiletine.
Olodaterol Uric acid may increase the hyperkalemic activities of Olodaterol.
Pancuronium The therapeutic efficacy of Pancuronium can be decreased when used in combination with Uric acid.
Pentoxifylline The serum concentration of Uric acid can be increased when it is combined with Pentoxifylline.
Phenytoin The serum concentration of Uric acid can be decreased when it is combined with Phenytoin.
Fosphenytoin The serum concentration of Uric acid can be decreased when it is combined with Fosphenytoin.
Propafenone The serum concentration of Uric acid can be increased when it is combined with Propafenone.
Quinine The serum concentration of Uric acid can be increased when it is combined with Quinine.
Quinidine The serum concentration of Uric acid can be increased when it is combined with Quinidine.
Riociguat Uric acid may increase the hypotensive activities of Riociguat.
Thiabendazole The metabolism of Uric acid can be decreased when combined with Thiabendazole.
Ticlopidine The metabolism of Uric acid can be decreased when combined with Ticlopidine.
Zafirlukast The serum concentration of Zafirlukast can be decreased when it is combined with Uric acid.
Probenecid The serum concentration of Uric acid can be increased when it is combined with Probenecid.
Isoprenaline The serum concentration of Uric acid can be decreased when it is combined with Isoprenaline.
Amphetamine The risk or severity of adverse effects can be increased when Amphetamine is combined with Uric acid.
Phentermine The risk or severity of adverse effects can be increased when Phentermine is combined with Uric acid.
Midodrine The risk or severity of adverse effects can be increased when Midodrine is combined with Uric acid.
Norepinephrine The risk or severity of adverse effects can be increased when Norepinephrine is combined with Uric acid.
Phenylephrine The risk or severity of adverse effects can be increased when Phenylephrine is combined with Uric acid.
Phenylpropanolamine The risk or severity of adverse effects can be increased when Phenylpropanolamine is combined with Uric acid.
Labetalol The risk or severity of adverse effects can be increased when Labetalol is combined with Uric acid.
Metaraminol The risk or severity of adverse effects can be increased when Metaraminol is combined with Uric acid.
Epinephrine The risk or severity of adverse effects can be increased when Epinephrine is combined with Uric acid.
Methoxamine The risk or severity of adverse effects can be increased when Methoxamine is combined with Uric acid.
Orciprenaline The risk or severity of adverse effects can be increased when Orciprenaline is combined with Uric acid.
Phenmetrazine The risk or severity of adverse effects can be increased when Phenmetrazine is combined with Uric acid.
Dobutamine The risk or severity of adverse effects can be increased when Dobutamine is combined with Uric acid.
Pseudoephedrine The risk or severity of adverse effects can be increased when Pseudoephedrine is combined with Uric acid.
Benzphetamine The risk or severity of adverse effects can be increased when Benzphetamine is combined with Uric acid.
Ritodrine The risk or severity of adverse effects can be increased when Ritodrine is combined with Uric acid.
Terbutaline The risk or severity of adverse effects can be increased when Terbutaline is combined with Uric acid.
Oxymetazoline The risk or severity of adverse effects can be increased when Oxymetazoline is combined with Uric acid.
Diethylpropion The risk or severity of adverse effects can be increased when Diethylpropion is combined with Uric acid.
Dopamine The risk or severity of adverse effects can be increased when Dopamine is combined with Uric acid.
Acebutolol The risk or severity of adverse effects can be increased when Acebutolol is combined with Uric acid.
Lisdexamfetamine The risk or severity of adverse effects can be increased when Lisdexamfetamine is combined with Uric acid.
Fenoterol The risk or severity of adverse effects can be increased when Fenoterol is combined with Uric acid.
Ephedrine The risk or severity of adverse effects can be increased when Ephedrine is combined with Uric acid.
Mephentermine The risk or severity of adverse effects can be increased when Mephentermine is combined with Uric acid.
Procaterol The risk or severity of adverse effects can be increased when Procaterol is combined with Uric acid.
Clenbuterol The risk or severity of adverse effects can be increased when Clenbuterol is combined with Uric acid.
MMDA The risk or severity of adverse effects can be increased when MMDA is combined with Uric acid.
Midomafetamine The risk or severity of adverse effects can be increased when Midomafetamine is combined with Uric acid.
2,5-Dimethoxy-4-ethylamphetamine The risk or severity of adverse effects can be increased when 2,5-Dimethoxy-4-ethylamphetamine is combined with Uric acid.
4-Bromo-2,5-dimethoxyamphetamine The risk or severity of adverse effects can be increased when 4-Bromo-2,5-dimethoxyamphetamine is combined with Uric acid.
Tenamfetamine The risk or severity of adverse effects can be increased when Tenamfetamine is combined with Uric acid.
Chlorphentermine The risk or severity of adverse effects can be increased when Chlorphentermine is combined with Uric acid.
Methylenedioxyethamphetamine The risk or severity of adverse effects can be increased when Methylenedioxyethamphetamine is combined with Uric acid.
Dextroamphetamine The risk or severity of adverse effects can be increased when Dextroamphetamine is combined with Uric acid.
Metamfetamine The risk or severity of adverse effects can be increased when Metamfetamine is combined with Uric acid.
Celiprolol The risk or severity of adverse effects can be increased when Celiprolol is combined with Uric acid.
Nylidrin The risk or severity of adverse effects can be increased when Nylidrin is combined with Uric acid.
Tetryzoline The risk or severity of adverse effects can be increased when Tetryzoline is combined with Uric acid.
Tyramine The risk or severity of adverse effects can be increased when Tyramine is combined with Uric acid.
Isoxsuprine The risk or severity of adverse effects can be increased when Isoxsuprine is combined with Uric acid.
Etilefrine The risk or severity of adverse effects can be increased when Etilefrine is combined with Uric acid.
Synephrine The risk or severity of adverse effects can be increased when Synephrine is combined with Uric acid.
Hydroxyamphetamine The risk or severity of adverse effects can be increased when Hydroxyamphetamine is combined with Uric acid.
Iofetamine I-123 The risk or severity of adverse effects can be increased when Iofetamine I-123 is combined with Uric acid.
Racepinephrine The risk or severity of adverse effects can be increased when Racepinephrine is combined with Uric acid.
Ritobegron The risk or severity of adverse effects can be increased when Ritobegron is combined with Uric acid.
Bucindolol The risk or severity of adverse effects can be increased when Bucindolol is combined with Uric acid.
Tramazoline The risk or severity of adverse effects can be increased when Tramazoline is combined with Uric acid.
Mephedrone The risk or severity of adverse effects can be increased when Mephedrone is combined with Uric acid.
Fenozolone The risk or severity of adverse effects can be increased when Fenozolone is combined with Uric acid.
Methoxyphenamine The risk or severity of adverse effects can be increased when Methoxyphenamine is combined with Uric acid.
Tretoquinol The risk or severity of adverse effects can be increased when Tretoquinol is combined with Uric acid.
Gepefrine The risk or severity of adverse effects can be increased when Gepefrine is combined with Uric acid.
Epanolol The risk or severity of adverse effects can be increased when Epanolol is combined with Uric acid.
Prenalterol The risk or severity of adverse effects can be increased when Prenalterol is combined with Uric acid.
Mefenorex The risk or severity of adverse effects can be increased when Mefenorex is combined with Uric acid.
2,5-Dimethoxy-4-ethylthioamphetamine The risk or severity of adverse effects can be increased when 2,5-Dimethoxy-4-ethylthioamphetamine is combined with Uric acid.
Esmolol The risk or severity of adverse effects can be increased when Esmolol is combined with Uric acid.
Betaxolol The risk or severity of adverse effects can be increased when Betaxolol is combined with Uric acid.
Metoprolol The risk or severity of adverse effects can be increased when Metoprolol is combined with Uric acid.
Atenolol The risk or severity of adverse effects can be increased when Atenolol is combined with Uric acid.
Timolol The risk or severity of adverse effects can be increased when Timolol is combined with Uric acid.
Sotalol The risk or severity of adverse effects can be increased when Sotalol is combined with Uric acid.
Propranolol The risk or severity of adverse effects can be increased when Propranolol is combined with Uric acid.
Bisoprolol The risk or severity of adverse effects can be increased when Bisoprolol is combined with Uric acid.
Alprenolol The risk or severity of adverse effects can be increased when Alprenolol is combined with Uric acid.
Pindolol The risk or severity of adverse effects can be increased when Pindolol is combined with Uric acid.
Carvedilol The risk or severity of adverse effects can be increased when Carvedilol is combined with Uric acid.
Bevantolol The risk or severity of adverse effects can be increased when Bevantolol is combined with Uric acid.

Target Protein

Glycogen phosphorylase, liver form PYGL

Referensi & Sumber

Synthesis reference: Brenner-Holzach, O.; Leuthardt, F. Uric acid formation from glucose carbon in Drosophila melanogaster. Preliminary report. Helvetica Chimica Acta (1963), 46(4), 1426-8.
Artikel (PubMed)
  • PMID: 14962621
    Chamorro A, Planas AM, Muner DS, Deulofeu R: Uric acid administration for neuroprotection in patients with acute brain ischemia. Med Hypotheses. 2004;62(2):173-6.
  • PMID: 16596120
    Romanos E, Planas AM, Amaro S, Chamorro A: Uric acid reduces brain damage and improves the benefits of rt-PA in a rat model of thromboembolic stroke. J Cereb Blood Flow Metab. 2007 Jan;27(1):14-20. Epub 2006 Apr 5.
  • PMID: 17525395
    Amaro S, Soy D, Obach V, Cervera A, Planas AM, Chamorro A: A pilot study of dual treatment with recombinant tissue plasminogen activator and uric acid in acute ischemic stroke. Stroke. 2007 Jul;38(7):2173-5. Epub 2007 May 24.
  • PMID: 9229228
    Maxwell SR, Thomason H, Sandler D, Leguen C, Baxter MA, Thorpe GH, Jones AF, Barnett AH: Antioxidant status in patients with uncomplicated insulin-dependent and non-insulin-dependent diabetes mellitus. Eur J Clin Invest. 1997 Jun;27(6):484-90.

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Sekuens Gen/Protein (FASTA)

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