Peringatan Keamanan

Agranulocytosis and neutropenia may occur, which can lead to fatal infections. Hepatoxicity is also possible. Most common side effects that lead to discontinuation of therapy were the gastrointestinal adverse effects (diarrhea, ulcer, nausea, gastrointestinal disturbances)

Deferiprone

DB08826

small molecule approved

Deskripsi

Deferiprone is an oral iron chelator used as a second line agent in thalassemia syndromes when iron overload from blood transfusions occurs. Thalassemias are a type of hereditary anaemia due a defect in the production of hemoglobin. As a result, erythropoiesis, the production of new red blood cells, is impaired. FDA approved on October 14, 2011.

Struktur Molekul 2D

Berat 139.1519
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The half-life is 1.9 hours.
Volume Distribusi In healthy patients, the volume of distribution is 1L/kg, and in thalassemia patients, the volume of distribution is 1.6L/kg.
Klirens (Clearance) -

Absorpsi

Deferiprone is absorbed in the upper gastrointestinal tract. Absorption is rapid with maximum plasma concentrations occurring after 1 hour in the fasted state and after 2 hours in the fed state.

Metabolisme

Deferiprone is mainly metabolized by UGT1A6 to the 3-O-glucuronide metabolite. This metabolite cannot chelate iron.

Rute Eliminasi

Within 5-6 hours of administration, more than 90% of deferiprone is eliminated from the plasma. 75 to 90% of deferiprone is excreted in the urine as the metabolite.

Interaksi Makanan

1 Data
  • 1. Take with or without food. Food does not affect absorption.

Interaksi Obat

804 Data
Calcium acetate The serum concentration of Deferiprone can be decreased when it is combined with Calcium acetate.
Calcium glucoheptonate The serum concentration of Deferiprone can be decreased when it is combined with Calcium glucoheptonate.
Calcium chloride The serum concentration of Deferiprone can be decreased when it is combined with Calcium chloride.
Calcium The serum concentration of Deferiprone can be decreased when it is combined with Calcium.
Calcium carbonate The serum concentration of Deferiprone can be decreased when it is combined with Calcium carbonate.
Calcium citrate The serum concentration of Deferiprone can be decreased when it is combined with Calcium citrate.
Calcium gluconate The serum concentration of Deferiprone can be decreased when it is combined with Calcium gluconate.
Calcium Phosphate The serum concentration of Deferiprone can be decreased when it is combined with Calcium Phosphate.
Calcium lactate The serum concentration of Deferiprone can be decreased when it is combined with Calcium lactate.
Calcium lactate gluconate The serum concentration of Deferiprone can be decreased when it is combined with Calcium lactate gluconate.
Calcium pangamate The serum concentration of Deferiprone can be decreased when it is combined with Calcium pangamate.
Calcium polycarbophil The serum concentration of Deferiprone can be decreased when it is combined with Calcium polycarbophil.
Troglitazone The serum concentration of Deferiprone can be increased when it is combined with Troglitazone.
Phenytoin The serum concentration of Deferiprone can be increased when it is combined with Phenytoin.
Fosphenytoin The serum concentration of Deferiprone can be increased when it is combined with Fosphenytoin.
Eltrombopag The serum concentration of Deferiprone can be increased when it is combined with Eltrombopag.
Magnesium sulfate Magnesium sulfate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium oxide Magnesium oxide can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium salicylate Magnesium salicylate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magaldrate Magaldrate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium hydroxide Magnesium hydroxide can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium trisilicate Magnesium trisilicate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium chloride Magnesium chloride can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium carbonate Magnesium carbonate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Talc Talc can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium citrate Magnesium citrate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium silicate Magnesium silicate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Hydrotalcite Hydrotalcite can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium aspartate Magnesium aspartate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium peroxide Magnesium peroxide can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium gluconate Magnesium gluconate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium orotate Magnesium orotate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium Magnesium can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium levulinate Magnesium levulinate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium lactate Magnesium lactate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc Zinc can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc trihydroxide Zinc trihydroxide can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc Substituted Heme C Zinc Substituted Heme C can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Polaprezinc Polaprezinc can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc oxide Zinc oxide can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc sulfate Zinc sulfate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc citrate Zinc citrate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc picolinate Zinc picolinate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc gluconate Zinc gluconate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Acetylcysteine zinc Acetylcysteine zinc can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc ascorbate Zinc ascorbate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc acetate Zinc acetate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc glycinate Zinc glycinate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc chloride Zinc chloride can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc sulfate, unspecified form Zinc sulfate, unspecified form can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zinc cation Zinc cation can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Selenium Selenium can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Magnesium cation Magnesium cation can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferrous ascorbate Ferrous ascorbate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Aluminum cation Aluminum cation can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nitroprusside The serum concentration of Deferiprone can be decreased when it is combined with Nitroprusside.
Iron Dextran The serum concentration of Deferiprone can be decreased when it is combined with Iron Dextran.
Iron The serum concentration of Deferiprone can be decreased when it is combined with Iron.
Ferumoxytol The serum concentration of Deferiprone can be decreased when it is combined with Ferumoxytol.
Prussian blue The serum concentration of Deferiprone can be decreased when it is combined with Prussian blue.
Ferric carboxymaltose The serum concentration of Deferiprone can be decreased when it is combined with Ferric carboxymaltose.
Iron sucrose The serum concentration of Deferiprone can be decreased when it is combined with Iron sucrose.
Ferric pyrophosphate The serum concentration of Deferiprone can be decreased when it is combined with Ferric pyrophosphate.
Ferric ammonium citrate The serum concentration of Deferiprone can be decreased when it is combined with Ferric ammonium citrate.
Ferumoxsil The serum concentration of Deferiprone can be decreased when it is combined with Ferumoxsil.
Ferumoxides The serum concentration of Deferiprone can be decreased when it is combined with Ferumoxides.
Ferric sulfate The serum concentration of Deferiprone can be decreased when it is combined with Ferric sulfate.
Ferrous bisglycinate The serum concentration of Deferiprone can be decreased when it is combined with Ferrous bisglycinate.
Gleptoferron The serum concentration of Deferiprone can be decreased when it is combined with Gleptoferron.
Ferric oxide The serum concentration of Deferiprone can be decreased when it is combined with Ferric oxide.
Perflubutane The serum concentration of Deferiprone can be decreased when it is combined with Perflubutane.
Ferrous sulfate anhydrous Ferrous sulfate anhydrous can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sodium feredetate The serum concentration of Deferiprone can be decreased when it is combined with Sodium feredetate.
Ferric hydroxide The serum concentration of Deferiprone can be decreased when it is combined with Ferric hydroxide.
Ferrous chloride The serum concentration of Deferiprone can be decreased when it is combined with Ferrous chloride.
Ferric cation Ferric cation can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferrous gluconate Ferrous gluconate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferrous succinate The serum concentration of Deferiprone can be decreased when it is combined with Ferrous succinate.
Ferrous fumarate The serum concentration of Deferiprone can be decreased when it is combined with Ferrous fumarate.
Tetraferric tricitrate decahydrate The serum concentration of Deferiprone can be decreased when it is combined with Tetraferric tricitrate decahydrate.
Ferric oxyhydroxide The serum concentration of Deferiprone can be decreased when it is combined with Ferric oxyhydroxide.
Ferric maltol The serum concentration of Deferiprone can be decreased when it is combined with Ferric maltol.
Iron isomaltoside 1000 The serum concentration of Deferiprone can be decreased when it is combined with Iron isomaltoside 1000.
Iron polymaltose The serum concentration of Deferiprone can be decreased when it is combined with Iron polymaltose.
Technetium Tc-99m oxidronate Deferiprone may decrease effectiveness of Technetium Tc-99m oxidronate as a diagnostic agent.
Cyclosporine Cyclosporine may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Icosapent Icosapent may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Cefotiam Cefotiam may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Mesalazine Mesalazine may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Cefmenoxime Cefmenoxime may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Cefmetazole Cefmetazole may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Pamidronic acid Pamidronic acid may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Tenofovir disoproxil Tenofovir disoproxil may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Indomethacin Indomethacin may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Cidofovir Cidofovir may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Cefpiramide Cefpiramide may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Ceftazidime Ceftazidime may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Loracarbef Loracarbef may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Cefalotin Cefalotin may decrease the excretion rate of Deferiprone which could result in a higher serum level.
Nabumetone Nabumetone may decrease the excretion rate of Deferiprone which could result in a higher serum level.

Target Protein

Iron

Referensi & Sumber

Artikel (PubMed)
  • PMID: 17636775
    Roberts DJ, Brunskill SJ, Doree C, Williams S, Howard J, Hyde CJ: Oral deferiprone for iron chelation in people with thalassaemia. Cochrane Database Syst Rev. 2007 Jul 18;(3):CD004839.
  • PMID: 15737892
    Victor Hoffbrand A: Deferiprone therapy for transfusional iron overload. Best Pract Res Clin Haematol. 2005 Jun;18(2):299-317.

Contoh Produk & Brand

Produk: 23 • International brands: 0
Produk
  • Deferiprone
    Tablet • 500 mg/1 • Oral • US • Generic • Approved
  • Deferiprone
    Tablet, coated • 500 mg/1 • Oral • US • Generic • Approved
  • Deferiprone
    Tablet, coated • 1000 mg/1 • Oral • US • Generic • Approved
  • Deferiprone
    Tablet • 1000 mg/1 • Oral • US • Generic • Approved
  • Deferiprone Lipomed
    Tablet, film coated • 500 mg • Oral • EU • Approved
  • Ferriprox
    Tablet, film coated • 500 mg • Oral • EU • Approved
  • Ferriprox
    Solution • 100 mg/ml • Oral • EU • Approved
  • Ferriprox
    Solution • 100 mg/ml • Oral • EU • Approved
Menampilkan 8 dari 23 produk.

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