Peringatan Keamanan

As with other antihistaminic drugs, overdosage can produce the following symptoms: CNS depression accompanied by drowsiness (especially in adults), CNS stimulation and antimuscarinic effects (especially in children) including the following: excitation, ataxia, hallucinations, tonic or clonic spasms, mydriasis, dryness of the mouth, redness of the face, urine retention, fever and tachycardia. Blood hypotension is also possible. In its terminal phase, coma can be aggravated by cardiorespiratory colapse and death. There has been no report of a fatal outcome of Dimethindene overdosage.

Dimetindene

DB08801

small molecule approved investigational

Deskripsi

Dimetindene (Fenistil) is an antihistamine/anticholinergic used orally and locally as an antipruritic.

Struktur Molekul 2D

Berat 292.418
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

524 Data
Aclidinium The risk or severity of adverse effects can be increased when Dimetindene is combined with Aclidinium.
Mianserin Mianserin may increase the anticholinergic activities of Dimetindene.
Mirabegron The risk or severity of urinary retention can be increased when Dimetindene is combined with Mirabegron.
Potassium chloride The risk or severity of gastrointestinal ulceration can be increased when Dimetindene is combined with Potassium chloride.
Pramlintide The risk or severity of reduced gastrointestinal motility can be increased when Pramlintide is combined with Dimetindene.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Dimetindene.
Tiotropium The risk or severity of adverse effects can be increased when Dimetindene is combined with Tiotropium.
Topiramate The risk or severity of hyperthermia and oligohydrosis can be increased when Dimetindene is combined with Topiramate.
Umeclidinium The risk or severity of adverse effects can be increased when Dimetindene is combined with Umeclidinium.
Benzylpenicilloyl polylysine Dimetindene may decrease effectiveness of Benzylpenicilloyl polylysine as a diagnostic agent.
Betahistine The therapeutic efficacy of Betahistine can be decreased when used in combination with Dimetindene.
Hyaluronidase (ovine) The therapeutic efficacy of Hyaluronidase (ovine) can be decreased when used in combination with Dimetindene.
Hyaluronidase (human recombinant) The therapeutic efficacy of Hyaluronidase (human recombinant) can be decreased when used in combination with Dimetindene.
Hyaluronidase The therapeutic efficacy of Hyaluronidase can be decreased when used in combination with Dimetindene.
Glycopyrronium The risk or severity of adverse effects can be increased when Dimetindene is combined with Glycopyrronium.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Dimetindene is combined with Botulinum toxin type A.
Glucagon Dimetindene may increase the gastrointestinal motility reducing activities of Glucagon.
Sulpiride Dimetindene may increase the anticholinergic activities of Sulpiride.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Dimetindene is combined with Botulinum toxin type B.
Eluxadoline The risk or severity of constipation can be increased when Dimetindene is combined with Eluxadoline.
Ramosetron The risk or severity of constipation can be increased when Dimetindene is combined with Ramosetron.
Amphetamine Amphetamine may decrease the sedative activities of Dimetindene.
Phentermine Phentermine may decrease the sedative activities of Dimetindene.
Pseudoephedrine Pseudoephedrine may decrease the sedative activities of Dimetindene.
Benzphetamine Benzphetamine may decrease the sedative activities of Dimetindene.
Diethylpropion Diethylpropion may decrease the sedative activities of Dimetindene.
Lisdexamfetamine Lisdexamfetamine may decrease the sedative activities of Dimetindene.
Mephentermine Mephentermine may decrease the sedative activities of Dimetindene.
MMDA MMDA may decrease the sedative activities of Dimetindene.
Midomafetamine Midomafetamine may decrease the sedative activities of Dimetindene.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the sedative activities of Dimetindene.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the sedative activities of Dimetindene.
Tenamfetamine Tenamfetamine may decrease the sedative activities of Dimetindene.
Chlorphentermine Chlorphentermine may decrease the sedative activities of Dimetindene.
Methylenedioxyethamphetamine Methylenedioxyethamphetamine may decrease the sedative activities of Dimetindene.
Dextroamphetamine Dextroamphetamine may decrease the sedative activities of Dimetindene.
Metamfetamine Metamfetamine may decrease the sedative activities of Dimetindene.
Iofetamine I-123 Iofetamine I-123 may decrease the sedative activities of Dimetindene.
Ritobegron Ritobegron may decrease the sedative activities of Dimetindene.
Mephedrone Mephedrone may decrease the sedative activities of Dimetindene.
Methoxyphenamine Methoxyphenamine may decrease the sedative activities of Dimetindene.
Gepefrine Gepefrine may decrease the sedative activities of Dimetindene.
2,5-Dimethoxy-4-ethylthioamphetamine 2,5-Dimethoxy-4-ethylthioamphetamine may decrease the sedative activities of Dimetindene.
Phendimetrazine Phendimetrazine may decrease the sedative activities of Dimetindene.
Naltrexone The risk or severity of adverse effects can be increased when Dimetindene is combined with Naltrexone.
Bezitramide The risk or severity of adverse effects can be increased when Dimetindene is combined with Bezitramide.
Tramadol The risk or severity of adverse effects can be increased when Dimetindene is combined with Tramadol.
Morphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Morphine.
Codeine The risk or severity of adverse effects can be increased when Dimetindene is combined with Codeine.
Hydromorphone The risk or severity of adverse effects can be increased when Dimetindene is combined with Hydromorphone.
Methadone The risk or severity of adverse effects can be increased when Dimetindene is combined with Methadone.
Meperidine The risk or severity of adverse effects can be increased when Dimetindene is combined with Meperidine.
Oxycodone The risk or severity of adverse effects can be increased when Dimetindene is combined with Oxycodone.
Butorphanol The risk or severity of adverse effects can be increased when Dimetindene is combined with Butorphanol.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Dimetindene is combined with Dextropropoxyphene.
Pentazocine The risk or severity of adverse effects can be increased when Dimetindene is combined with Pentazocine.
Sufentanil The risk or severity of adverse effects can be increased when Dimetindene is combined with Sufentanil.
Alfentanil The risk or severity of adverse effects can be increased when Dimetindene is combined with Alfentanil.
Fentanyl The risk or severity of adverse effects can be increased when Dimetindene is combined with Fentanyl.
Nalbuphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Nalbuphine.
Levorphanol The risk or severity of adverse effects can be increased when Dimetindene is combined with Levorphanol.
Remifentanil The risk or severity of adverse effects can be increased when Dimetindene is combined with Remifentanil.
Buprenorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Buprenorphine.
Hydrocodone The risk or severity of adverse effects can be increased when Dimetindene is combined with Hydrocodone.
Diphenoxylate The risk or severity of adverse effects can be increased when Dimetindene is combined with Diphenoxylate.
Oxymorphone The risk or severity of adverse effects can be increased when Dimetindene is combined with Oxymorphone.
Dezocine The risk or severity of adverse effects can be increased when Dimetindene is combined with Dezocine.
Levacetylmethadol The risk or severity of adverse effects can be increased when Dimetindene is combined with Levacetylmethadol.
Methadyl acetate The risk or severity of adverse effects can be increased when Dimetindene is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Dihydroetorphine.
Diamorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Diamorphine.
Ethylmorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Ethylmorphine.
Etorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Etorphine.
Dextromoramide The risk or severity of adverse effects can be increased when Dimetindene is combined with Dextromoramide.
Desomorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Desomorphine.
Carfentanil The risk or severity of adverse effects can be increased when Dimetindene is combined with Carfentanil.
Dihydrocodeine The risk or severity of adverse effects can be increased when Dimetindene is combined with Dihydrocodeine.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Dimetindene is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Dihydromorphine.
Tapentadol The risk or severity of urinary retention and constipation can be increased when Dimetindene is combined with Tapentadol.
Ketobemidone The risk or severity of adverse effects can be increased when Dimetindene is combined with Ketobemidone.
DPDPE The risk or severity of adverse effects can be increased when Dimetindene is combined with DPDPE.
Lofentanil The risk or severity of adverse effects can be increased when Dimetindene is combined with Lofentanil.
Opium The risk or severity of adverse effects can be increased when Dimetindene is combined with Opium.
Normethadone The risk or severity of adverse effects can be increased when Dimetindene is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Dimetindene is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Dimetindene is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Dimetindene is combined with Nicomorphine.
Meptazinol The risk or severity of adverse effects can be increased when Dimetindene is combined with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Dimetindene is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Dimetindene is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Dimetindene is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Dimetindene is combined with Carfentanil, C-11.
Benzhydrocodone The risk or severity of adverse effects can be increased when Dimetindene is combined with Benzhydrocodone.
Naloxegol The risk or severity of adverse effects can be increased when Dimetindene is combined with Naloxegol.
Trospium The risk or severity of adverse effects can be increased when Trospium is combined with Dimetindene.
Oxyphenonium The risk or severity of adverse effects can be increased when Oxyphenonium is combined with Dimetindene.
Benzatropine The risk or severity of adverse effects can be increased when Benzatropine is combined with Dimetindene.
Disopyramide The risk or severity of adverse effects can be increased when Disopyramide is combined with Dimetindene.
Metixene The risk or severity of adverse effects can be increased when Metixene is combined with Dimetindene.

Target Protein

Histamine H1 receptor HRH1
Muscarinic acetylcholine receptor M2 CHRM2

Referensi & Sumber

Synthesis reference: Huebner, C.F.; U S . Patent 2,970,149; January 31, 1961; assigned to Ciba Pharmaceutical Products, Inc.
Artikel (PubMed)
  • PMID: 10069503
    Lambrecht G, Gross J, Mutschler E: Neuronal soma-dendritic and prejunctional M1-M4 receptors in gastrointestinal and genitourinary smooth muscle. Life Sci. 1999;64(6-7):403-10.

Contoh Produk & Brand

Produk: 0 • International brands: 3
International Brands
  • Fenistil — Novartis
  • Foristal — Novartis
  • Vibrocil — Novartis

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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