Tranilast

DB07615

small molecule investigational

Deskripsi

Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. In 1982, it was approved in Japan and South Korea for the management of bronchial asthma. Indications for keloid and hypertrophic scar were added in 1993. It has been used for the treatment of allergic disorders such as asthma, allergic rhinitis and atopic dermatitis.

Struktur Molekul 2D

Berat 327.3313
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1211 Data
Apixaban The risk or severity of adverse effects can be increased when Tranilast is combined with Apixaban.
Dasatinib Dasatinib may increase the anticoagulant activities of Tranilast.
Ursodeoxycholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Ursodeoxycholic acid.
Glycochenodeoxycholic Acid The risk or severity of adverse effects can be increased when Tranilast is combined with Glycochenodeoxycholic Acid.
Cholic Acid The risk or severity of adverse effects can be increased when Tranilast is combined with Cholic Acid.
Glycocholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Glycocholic acid.
Deoxycholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Deoxycholic acid.
Taurocholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Taurocholic acid.
Obeticholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Obeticholic acid.
Chenodeoxycholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Chenodeoxycholic acid.
Taurochenodeoxycholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Taurochenodeoxycholic acid.
Tauroursodeoxycholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Tauroursodeoxycholic acid.
Bamet-UD2 The risk or severity of adverse effects can be increased when Tranilast is combined with Bamet-UD2.
Dehydrocholic acid The risk or severity of adverse effects can be increased when Tranilast is combined with Dehydrocholic acid.
Hyodeoxycholic Acid The risk or severity of adverse effects can be increased when Tranilast is combined with Hyodeoxycholic Acid.
Glucosamine Glucosamine may increase the antiplatelet activities of Tranilast.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Tranilast is combined with Ibritumomab tiuxetan.
Ibrutinib The risk or severity of adverse effects can be increased when Ibrutinib is combined with Tranilast.
Obinutuzumab The risk or severity of adverse effects can be increased when Tranilast is combined with Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the antiplatelet activities of Tranilast.
Rivaroxaban Tranilast may increase the anticoagulant activities of Rivaroxaban.
Tipranavir Tipranavir may increase the antiplatelet activities of Tranilast.
Urokinase Tranilast may increase the anticoagulant activities of Urokinase.
Vitamin E Vitamin E may increase the antiplatelet activities of Tranilast.
Ceritinib Tranilast may increase the bradycardic activities of Ceritinib.
Ivabradine Tranilast may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of Tranilast.
Cimetidine The serum concentration of Tranilast can be increased when it is combined with Cimetidine.
Clopidogrel The therapeutic efficacy of Clopidogrel can be decreased when used in combination with Tranilast.
Efavirenz The serum concentration of Tranilast can be decreased when it is combined with Efavirenz.
Melatonin The therapeutic efficacy of Tranilast can be decreased when used in combination with Melatonin.
Nafcillin The therapeutic efficacy of Tranilast can be decreased when used in combination with Nafcillin.
Nitroprusside Tranilast may increase the hypotensive activities of Nitroprusside.
Dantrolene The risk or severity of hyperkalemia can be increased when Dantrolene is combined with Tranilast.
Lithium citrate The risk or severity of adverse effects can be increased when Tranilast is combined with Lithium citrate.
Lithium carbonate The risk or severity of adverse effects can be increased when Tranilast is combined with Lithium carbonate.
Lithium hydroxide The risk or severity of adverse effects can be increased when Tranilast is combined with Lithium hydroxide.
Boceprevir The serum concentration of Tranilast can be increased when it is combined with Boceprevir.
Pentosan polysulfate The risk or severity of adverse effects can be increased when Pentosan polysulfate is combined with Tranilast.
Limaprost Limaprost may increase the antiplatelet activities of Tranilast.
Omega-3 fatty acids Omega-3 fatty acids may increase the antiplatelet activities of Tranilast.
Tositumomab The risk or severity of adverse effects can be increased when Tranilast is combined with Tositumomab.
Ibutilide Ibutilide may increase the arrhythmogenic activities of Tranilast.
Hyoscyamine Hyoscyamine may increase the arrhythmogenic activities of Tranilast.
Atropine Atropine may increase the arrhythmogenic activities of Tranilast.
Adenosine Adenosine may increase the arrhythmogenic activities of Tranilast.
Moricizine Moricizine may increase the arrhythmogenic activities of Tranilast.
Levosimendan Levosimendan may increase the arrhythmogenic activities of Tranilast.
Procainamide Procainamide may increase the arrhythmogenic activities of Tranilast.
Tocainide Tocainide may increase the arrhythmogenic activities of Tranilast.
Encainide Encainide may increase the arrhythmogenic activities of Tranilast.
Ajmaline Ajmaline may increase the arrhythmogenic activities of Tranilast.
Aprindine Aprindine may increase the arrhythmogenic activities of Tranilast.
Azimilide Azimilide may increase the arrhythmogenic activities of Tranilast.
Tedisamil Tedisamil may increase the arrhythmogenic activities of Tranilast.
Vernakalant Vernakalant may increase the arrhythmogenic activities of Tranilast.
Cariporide Cariporide may increase the arrhythmogenic activities of Tranilast.
Xylometazoline Xylometazoline may increase the arrhythmogenic activities of Tranilast.
Sparteine Sparteine may increase the arrhythmogenic activities of Tranilast.
Carteolol Tranilast may increase the arrhythmogenic activities of Carteolol.
Metipranolol Tranilast may increase the arrhythmogenic activities of Metipranolol.
Fasudil Tranilast may increase the arrhythmogenic activities of Fasudil.
Melperone Tranilast may increase the arrhythmogenic activities of Melperone.
Tropisetron Tranilast may increase the arrhythmogenic activities of Tropisetron.
Simendan Tranilast may increase the arrhythmogenic activities of Simendan.
Spiradoline Tranilast may increase the arrhythmogenic activities of Spiradoline.
Pilsicainide Tranilast may increase the arrhythmogenic activities of Pilsicainide.
Cicletanine Tranilast may increase the arrhythmogenic activities of Cicletanine.
Cibenzoline Tranilast may increase the arrhythmogenic activities of Cibenzoline.
Nizofenone Tranilast may increase the arrhythmogenic activities of Nizofenone.
Prajmaline Tranilast may increase the arrhythmogenic activities of Prajmaline.
Tiracizine Tranilast may increase the arrhythmogenic activities of Tiracizine.
Ethacizine Tranilast may increase the arrhythmogenic activities of Ethacizine.
Lorajmine Tranilast may increase the arrhythmogenic activities of Lorajmine.
Bunaftine Tranilast may increase the arrhythmogenic activities of Bunaftine.
Lorcainide Tranilast may increase the arrhythmogenic activities of Lorcainide.
Hydroquinine Tranilast may increase the arrhythmogenic activities of Hydroquinine.
Bioallethrin Tranilast may increase the arrhythmogenic activities of Bioallethrin.
Fosfructose Tranilast may increase the arrhythmogenic activities of Fosfructose.
Hydroquinidine Tranilast may increase the arrhythmogenic activities of Hydroquinidine.
SOR-C13 Tranilast may increase the arrhythmogenic activities of SOR-C13.
Digoxin Digoxin may increase the arrhythmogenic activities of Tranilast.
Acetyldigitoxin Acetyldigitoxin may increase the arrhythmogenic activities of Tranilast.
Deslanoside Deslanoside may increase the arrhythmogenic activities of Tranilast.
Cymarin Tranilast may increase the arrhythmogenic activities of Cymarin.
Metildigoxin Tranilast may increase the arrhythmogenic activities of Metildigoxin.
Acetyldigoxin Tranilast may increase the arrhythmogenic activities of Acetyldigoxin.
Niguldipine Tranilast may increase the arrhythmogenic activities of Niguldipine.
Bretylium Bretylium may increase the arrhythmogenic activities of Tranilast.
Isradipine Isradipine may increase the arrhythmogenic activities of Tranilast.
Diltiazem Diltiazem may increase the arrhythmogenic activities of Tranilast.
Trimethadione Trimethadione may increase the arrhythmogenic activities of Tranilast.
Amlodipine Amlodipine may increase the arrhythmogenic activities of Tranilast.
Nimodipine Nimodipine may increase the arrhythmogenic activities of Tranilast.
Lercanidipine Lercanidipine may increase the arrhythmogenic activities of Tranilast.
Lamotrigine Lamotrigine may increase the arrhythmogenic activities of Tranilast.
Cinnarizine Cinnarizine may increase the arrhythmogenic activities of Tranilast.
Verapamil Verapamil may increase the arrhythmogenic activities of Tranilast.
Losartan Losartan may increase the arrhythmogenic activities of Tranilast.
Levomenthol Levomenthol may increase the arrhythmogenic activities of Tranilast.

Target Protein

Steryl-sulfatase STS
Histamine H1 receptor HRH1
Hematopoietic prostaglandin D synthase HPGDS

Referensi & Sumber

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