Peringatan Keamanan

The most important form of toxicity associated with the use of plicamycin consists of a dose-related bleeding syndrome which usually begins with an episode of epistaxis. Plicamycin crosses the blood-brain barrier; the concentration found in brain tissue is low but it persists longer than in other tissues.

Plicamycin

DB06810

small molecule approved investigational withdrawn

Deskripsi

Plicamycin is an antineoplastic antibiotic produced by Streptomyces plicatus. It has been used in the treatment of testicular cancer, Paget's disease of bone, and, rarely, the management of hypercalcemia. The manufacturer discontinued plicamycin in 2000.

Struktur Molekul 2D

Berat 1085.1454
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Radioautography studies with 3H-labeled plicamycin in mice show that the greatest concentrations of the isotope are in the Kupffer cells of the liver and cells of the renal tubules. Plicamycin is rapidly cleared from the blood within the first 2 hours and excretion is also rapid. 67% percent of measured excretion occurs within 4 hours, 75% within 8 hours, and 90% is recovered in the first 24 hours after injection.

Interaksi Obat

41 Data
Trastuzumab The risk or severity of cardiotoxicity can be increased when Trastuzumab is combined with Plicamycin.
Margetuximab The risk or severity of cardiotoxicity can be increased when Margetuximab is combined with Plicamycin.
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Plicamycin.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Plicamycin.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Plicamycin.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Plicamycin.
Lidocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Quinisocaine.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Plicamycin.
Ambroxol The risk or severity of methemoglobinemia can be increased when Plicamycin is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Plicamycin is combined with Etrasimod.

Target Protein

DNA

Referensi & Sumber

Synthesis reference: Jurgen Rohr, Lily Remsing, Mohammad Nur-e-Alam, Jose Salas, Carmen Mendez, Alfredo Brana, Ana Gonzalez, "Derivatives of mithramycin and methods of making and uses thereof." U.S. Patent US20050192432, issued September 01, 2005.
Artikel (PubMed)
  • PMID: 9917296
    Wohlert SE, Kunzel E, Machinek R, Mendez C, Salas JA, Rohr J: The structure of mithramycin reinvestigated. J Nat Prod. 1999 Jan;62(1):119-21.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Mithracin — Pfizer

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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