Peringatan Keamanan

The major drawback of nonoxynol-9 is its detergent-type action on epithelial cells and the normal vaginal flora. Detergent-type spermicides alter the vaginal flora, possibly leading to an increased risk of opportunistic infections. These are known to enhance the susceptibility of the epithelium of the lower genital tract to HIV and human papillomavirus infection. N-9 can cause vaginal irritation and allergic vaginitis as well as genital irritation in male partners.

Nonoxynol-9

DB06804

small molecule approved withdrawn

Deskripsi

Nonoxynol-9 (N-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives. When present in the vagina during intercourse, they immobilize/inactivate/damage and/or kill sperms without eliciting systemic effects. N-9 has been in use for more than 30 years as an over-the-counter (OTC) drug in creams, gels, foams and condom lubricants. It is the most commonly used spermicidal contraceptive in the UK and the USA. In several European countries, spermicides are no longer on the market.

Struktur Molekul 2D

Berat 616.8235
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

113 Data
Aprepitant The serum concentration of Nonoxynol-9 can be decreased when it is combined with Aprepitant.
Thalidomide Nonoxynol-9 may increase the thrombogenic activities of Thalidomide.
Tranexamic acid Tranexamic acid may increase the thrombogenic activities of Nonoxynol-9.
Lorazepam The metabolism of Nonoxynol-9 can be increased when combined with Lorazepam.
Pregabalin The metabolism of Nonoxynol-9 can be increased when combined with Pregabalin.
Butalbital The metabolism of Nonoxynol-9 can be increased when combined with Butalbital.
Phenytoin The metabolism of Nonoxynol-9 can be increased when combined with Phenytoin.
Topiramate The metabolism of Nonoxynol-9 can be increased when combined with Topiramate.
Pentobarbital The metabolism of Nonoxynol-9 can be increased when combined with Pentobarbital.
Valproic acid The metabolism of Nonoxynol-9 can be increased when combined with Valproic acid.
Trimethadione The metabolism of Nonoxynol-9 can be increased when combined with Trimethadione.
Clobazam The metabolism of Nonoxynol-9 can be increased when combined with Clobazam.
Secobarbital The metabolism of Nonoxynol-9 can be increased when combined with Secobarbital.
Metharbital The metabolism of Nonoxynol-9 can be increased when combined with Metharbital.
Methohexital The metabolism of Nonoxynol-9 can be increased when combined with Methohexital.
Mephenytoin The metabolism of Nonoxynol-9 can be increased when combined with Mephenytoin.
Lamotrigine The metabolism of Nonoxynol-9 can be increased when combined with Lamotrigine.
Carbamazepine The metabolism of Nonoxynol-9 can be increased when combined with Carbamazepine.
Ethosuximide The metabolism of Nonoxynol-9 can be increased when combined with Ethosuximide.
Thiopental The metabolism of Nonoxynol-9 can be increased when combined with Thiopental.
Paramethadione The metabolism of Nonoxynol-9 can be increased when combined with Paramethadione.
Clorazepic acid The metabolism of Nonoxynol-9 can be increased when combined with Clorazepic acid.
Magnesium sulfate The metabolism of Nonoxynol-9 can be increased when combined with Magnesium sulfate.
Tizanidine The metabolism of Nonoxynol-9 can be increased when combined with Tizanidine.
Riluzole The metabolism of Nonoxynol-9 can be increased when combined with Riluzole.
Ethotoin The metabolism of Nonoxynol-9 can be increased when combined with Ethotoin.
Oxcarbazepine The metabolism of Nonoxynol-9 can be increased when combined with Oxcarbazepine.
Primidone The metabolism of Nonoxynol-9 can be increased when combined with Primidone.
Acetazolamide The metabolism of Nonoxynol-9 can be increased when combined with Acetazolamide.
Diazepam The metabolism of Nonoxynol-9 can be increased when combined with Diazepam.
Phensuximide The metabolism of Nonoxynol-9 can be increased when combined with Phensuximide.
Progabide The metabolism of Nonoxynol-9 can be increased when combined with Progabide.
Methylphenobarbital The metabolism of Nonoxynol-9 can be increased when combined with Methylphenobarbital.
Tiagabine The metabolism of Nonoxynol-9 can be increased when combined with Tiagabine.
Zonisamide The metabolism of Nonoxynol-9 can be increased when combined with Zonisamide.
Felbamate The metabolism of Nonoxynol-9 can be increased when combined with Felbamate.
Zaleplon The metabolism of Nonoxynol-9 can be increased when combined with Zaleplon.
Gabapentin The metabolism of Nonoxynol-9 can be increased when combined with Gabapentin.
Clonazepam The metabolism of Nonoxynol-9 can be increased when combined with Clonazepam.
Vigabatrin The metabolism of Nonoxynol-9 can be increased when combined with Vigabatrin.
Phenacemide The metabolism of Nonoxynol-9 can be increased when combined with Phenacemide.
Thiamylal The metabolism of Nonoxynol-9 can be increased when combined with Thiamylal.
Phenobarbital The metabolism of Nonoxynol-9 can be increased when combined with Phenobarbital.
Levetiracetam The metabolism of Nonoxynol-9 can be increased when combined with Levetiracetam.
Estazolam The metabolism of Nonoxynol-9 can be increased when combined with Estazolam.
Fosphenytoin The metabolism of Nonoxynol-9 can be increased when combined with Fosphenytoin.
Amobarbital The metabolism of Nonoxynol-9 can be increased when combined with Amobarbital.
Hexobarbital The metabolism of Nonoxynol-9 can be increased when combined with Hexobarbital.
Barbital The metabolism of Nonoxynol-9 can be increased when combined with Barbital.
Delorazepam The metabolism of Nonoxynol-9 can be increased when combined with Delorazepam.
Nitrazepam The metabolism of Nonoxynol-9 can be increased when combined with Nitrazepam.
7-Nitroindazole The metabolism of Nonoxynol-9 can be increased when combined with 7-Nitroindazole.
Valpromide The metabolism of Nonoxynol-9 can be increased when combined with Valpromide.
Flunarizine The metabolism of Nonoxynol-9 can be increased when combined with Flunarizine.
Ezogabine The metabolism of Nonoxynol-9 can be increased when combined with Ezogabine.
Methsuximide The metabolism of Nonoxynol-9 can be increased when combined with Methsuximide.
Brivaracetam The metabolism of Nonoxynol-9 can be increased when combined with Brivaracetam.
Rufinamide The metabolism of Nonoxynol-9 can be increased when combined with Rufinamide.
Lacosamide The metabolism of Nonoxynol-9 can be increased when combined with Lacosamide.
Remacemide The metabolism of Nonoxynol-9 can be increased when combined with Remacemide.
Clomethiazole The metabolism of Nonoxynol-9 can be increased when combined with Clomethiazole.
Deramciclane The metabolism of Nonoxynol-9 can be increased when combined with Deramciclane.
Tramiprosate The metabolism of Nonoxynol-9 can be increased when combined with Tramiprosate.
Gaboxadol The metabolism of Nonoxynol-9 can be increased when combined with Gaboxadol.
Sulthiame The metabolism of Nonoxynol-9 can be increased when combined with Sulthiame.
Perampanel The metabolism of Nonoxynol-9 can be increased when combined with Perampanel.
Ifenprodil The metabolism of Nonoxynol-9 can be increased when combined with Ifenprodil.
Barbexaclone The metabolism of Nonoxynol-9 can be increased when combined with Barbexaclone.
Beclamide The metabolism of Nonoxynol-9 can be increased when combined with Beclamide.
Cannabidiol The metabolism of Nonoxynol-9 can be increased when combined with Cannabidiol.
Paraldehyde The metabolism of Nonoxynol-9 can be increased when combined with Paraldehyde.
Stiripentol The metabolism of Nonoxynol-9 can be increased when combined with Stiripentol.
Eslicarbazepine acetate The metabolism of Nonoxynol-9 can be increased when combined with Eslicarbazepine acetate.
Doramectin The metabolism of Nonoxynol-9 can be increased when combined with Doramectin.
Tiletamine The metabolism of Nonoxynol-9 can be increased when combined with Tiletamine.
Brexanolone The metabolism of Nonoxynol-9 can be increased when combined with Brexanolone.
Etiracetam The metabolism of Nonoxynol-9 can be increased when combined with Etiracetam.
Vinpocetine The metabolism of Nonoxynol-9 can be increased when combined with Vinpocetine.
Carisbamate The metabolism of Nonoxynol-9 can be increased when combined with Carisbamate.
Pheneturide The metabolism of Nonoxynol-9 can be increased when combined with Pheneturide.
Neocitrullamon The metabolism of Nonoxynol-9 can be increased when combined with Neocitrullamon.
Medazepam The metabolism of Nonoxynol-9 can be increased when combined with Medazepam.
Phenibut The metabolism of Nonoxynol-9 can be increased when combined with Phenibut.
Ethadione The metabolism of Nonoxynol-9 can be increased when combined with Ethadione.
Cannabidivarin The metabolism of Nonoxynol-9 can be increased when combined with Cannabidivarin.
Eslicarbazepine The metabolism of Nonoxynol-9 can be increased when combined with Eslicarbazepine.
JNJ-26489112 The metabolism of Nonoxynol-9 can be increased when combined with JNJ-26489112.
Cenobamate The metabolism of Nonoxynol-9 can be increased when combined with Cenobamate.
St. John's Wort The metabolism of Nonoxynol-9 can be increased when combined with St. John's Wort.
Glimepiride The therapeutic efficacy of Glimepiride can be decreased when used in combination with Nonoxynol-9.
Acetohexamide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Nonoxynol-9.
Chlorpropamide The therapeutic efficacy of Chlorpropamide can be decreased when used in combination with Nonoxynol-9.
Tolazamide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Nonoxynol-9.
Glyburide The therapeutic efficacy of Glyburide can be decreased when used in combination with Nonoxynol-9.
Glipizide The therapeutic efficacy of Glipizide can be decreased when used in combination with Nonoxynol-9.
Gliclazide The therapeutic efficacy of Gliclazide can be decreased when used in combination with Nonoxynol-9.
Tolbutamide The therapeutic efficacy of Tolbutamide can be decreased when used in combination with Nonoxynol-9.
Gliquidone The therapeutic efficacy of Gliquidone can be decreased when used in combination with Nonoxynol-9.
Glisoxepide The therapeutic efficacy of Glisoxepide can be decreased when used in combination with Nonoxynol-9.
Glibornuride The therapeutic efficacy of Glibornuride can be decreased when used in combination with Nonoxynol-9.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 19117251
    Iyer V, Poddar SS: Update on nonoxynol-9 as vaginal spermicide. Eur J Contracept Reprod Health Care. 2008 Dec;13(4):339-50. doi: 10.1080/13625180802263515.

Contoh Produk & Brand

Produk: 8 • International brands: 4
Produk
  • Conceptrol Options
    Gel • 4.0 g/100g • Vaginal • US • OTC
  • ContraSeed
    Suppository • 100 mg/1 • Vaginal • US • OTC
  • Encare
    Insert • 100 mg/1 • Vaginal • US • OTC
  • Gynol II Extra Strength
    Gel • 3.0 g/100g • Vaginal • US • OTC
  • Today Vaginal Contraceptive
    Sponge • 1000 mg/1 • Vaginal • US • OTC • Approved
  • Vcf Contraceptive
    Film, soluble • 280 mg/1 • Vaginal • US • OTC
  • Vcf Contraceptive
    Aerosol, foam • 125 mg/1g • Vaginal • US • OTC
  • Vcf Contraceptive Pre-filled Applicators
    Gel, metered • 4 g/100g • Vaginal • US • OTC
International Brands
  • Advantage 24 — Lake Pharmaceuticals
  • Gynoll — Ortho Options
  • Today — Bliss Pharmaceuticals
  • VCF — Apothecus Pharmaceuticals

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