Peringatan Keamanan

Since mafenide is metabolized to a carbonic anhydrase inhibitor, metabolic acidosis could occur.

Mafenide

DB06795

small molecule approved vet_approved withdrawn

Deskripsi

Mafenide is a sulfonamide-type antimicrobial agent used to treat severe burns. It acts by reducing the bacterial population present in the burn tissue and promotes healing of deep burns.L36773 In 1998, mafenide acetate was approved under the FDA’s accelerated approval regulations. In November 2022, the use of mafenide acetate (powder for 5% topical solution) was withdrawn by the FDA due to an unresolved confirmatory study required to fulfill the accelerated approval requirements.L44251

Struktur Molekul 2D

Berat 186.232
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Mafenide is absorbed through devascularized areas into the systemic circulation following topical administration.

Metabolisme

Metabolized to a carbonic anhydrase inhibitor.

Rute Eliminasi

Renal—Metabolite rapidly excreted in urine in high concentrations; however, the parent compound has not been detected in urine.

Interaksi Obat

22 Data
Prilocaine The risk or severity of methemoglobinemia can be increased when Mafenide is combined with Prilocaine.
Dapsone The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Mafenide.
Magnesium The serum concentration of Magnesium can be decreased when it is combined with Mafenide.
Benzylpenicillin Mafenide may decrease the excretion rate of Benzylpenicillin which could result in a higher serum level.
Estetrol The therapeutic efficacy of Estetrol can be decreased when used in combination with Mafenide.
Allogeneic cultured keratinocytes and dermal fibroblasts in murine collagen The therapeutic efficacy of Allogeneic cultured keratinocytes and dermal fibroblasts in murine collagen can be decreased when used in combination with Mafenide.
Insulin human The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin human.
Insulin lispro The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin lispro.
Insulin glargine The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin glargine.
Insulin pork The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin pork.
Insulin aspart The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin aspart.
Insulin detemir The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin detemir.
Insulin glulisine The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin glulisine.
NN344 The risk or severity of hypoglycemia can be increased when Mafenide is combined with NN344.
Insulin beef The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin beef.
Insulin degludec The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin degludec.
Insulin argine The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin argine.
Insulin peglispro The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin peglispro.
Insulin tregopil The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin tregopil.
Tenofovir alafenamide The serum concentration of Tenofovir alafenamide can be increased when it is combined with Mafenide.
Fecal microbiota The therapeutic efficacy of Fecal microbiota can be decreased when used in combination with Mafenide.
Insulin icodec The risk or severity of hypoglycemia can be increased when Mafenide is combined with Insulin icodec.

Target Protein

Carbonic anhydrase 2 CA2
Carbonic anhydrase 12 CA12
Carbonic anhydrase 14 CA14
Carbonic anhydrase 4 CA4
Carbonic anhydrase 6 CA6

Referensi & Sumber

Synthesis reference: U.S. Patent 2,288,531.
Artikel (PubMed)
  • PMID: 22396671
    Maghsoudi H, Salehi F, Khosrowshahi MK, Baghaei M, Nasirzadeh M, Shams R: Comparison between topical honey and mafenide acetate in treatment of burn wounds. Ann Burns Fire Disasters. 2011 Sep 30;24(3):132-7.

Contoh Produk & Brand

Produk: 8 • International brands: 0
Produk
  • Mafenide acetate
    Powder, for solution • 50 g/1 • Topical • US • Generic • Approved
  • Mafenide Acetate
    Powder, for solution • 50 g/1 • Topical • US • Generic • Approved
  • Mafenide Acetate
    Powder, for solution • 50 g/1 • Topical • US • Generic • Approved
  • Sulfamylon
    Powder, for solution • 50 g/1 • Topical • US • Approved
  • Sulfamylon
    Powder, for solution • 50 g/1 • Topical • US • Approved
  • Sulfamylon
    Cream • 85 mg/1g • Topical • US • Approved
  • Sulfamylon
    Cream • 85 mg/1g • Topical • US • Approved
  • Sulfamylon Cream - 8.5%
    Cream • 8.5 % • Topical • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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