Alcaftadine

DB06766

small molecule approved

Deskripsi

Alcaftadine is a H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis. This drug was approved in July 2010.

Struktur Molekul 2D

Berat 307.3895
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The elimination half-life of the carboxylic acid metabolite is approximately 2 hours following topical ocular administration.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

The metabolism of alcaftadine is mediated by non-CYP450 cytosolic enzymes to the active carboxylic acid metabolite.

Rute Eliminasi

Based on data following oral administration of alcaftadine, the carboxylic acid metabolite is primarily eliminated unchanged in the urine.

Interaksi Obat

27 Data
Trazodone The risk or severity of QTc prolongation can be increased when Trazodone is combined with Alcaftadine.
Pitolisant Alcaftadine may increase the QTc-prolonging activities of Pitolisant.
Lefamulin Lefamulin may increase the QTc-prolonging activities of Alcaftadine.
Hydroxyzine The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Hydroxyzine.
Ziprasidone The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Ziprasidone.
Haloperidol The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Haloperidol.
Fluoxetine The risk or severity of QTc prolongation can be increased when Fluoxetine is combined with Alcaftadine.
Hyoscyamine Alcaftadine may increase the anticholinergic activities of Hyoscyamine.
Ponesimod The risk or severity of bradycardia can be increased when Ponesimod is combined with Alcaftadine.
Fexinidazole The risk or severity of adverse effects can be increased when Alcaftadine is combined with Fexinidazole.
Tenofovir alafenamide The serum concentration of Tenofovir alafenamide can be increased when it is combined with Alcaftadine.
Clozapine The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Clozapine.
Glasdegib The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Glasdegib.
Vilanterol The risk or severity of QTc prolongation and ventricular arrhythmias can be increased when Vilanterol is combined with Alcaftadine.
Oxaliplatin The risk or severity of QTc prolongation can be increased when Oxaliplatin is combined with Alcaftadine.
Quizartinib The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Quizartinib.
Citalopram The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Citalopram.
Pimavanserin The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Pimavanserin.
Gepirone The risk or severity of QTc prolongation can be increased when Gepirone is combined with Alcaftadine.
Etrasimod The risk or severity of QTc prolongation and torsade de pointes can be increased when Etrasimod is combined with Alcaftadine.
Bedaquiline The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Bedaquiline.
Encorafenib The risk or severity of QTc prolongation can be increased when Encorafenib is combined with Alcaftadine.
Givinostat The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Givinostat.
Inotuzumab ozogamicin The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Inotuzumab ozogamicin.
Mavorixafor The risk or severity of QTc prolongation can be increased when Mavorixafor is combined with Alcaftadine.
Ribociclib The risk or severity of QTc prolongation can be increased when Ribociclib is combined with Alcaftadine.
Revumenib The risk or severity of QTc prolongation can be increased when Alcaftadine is combined with Revumenib.

Target Protein

Histamine H1 receptor HRH1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 22811343
    Mahvan TD, Buckley WA, Hornecker JR: Alcaftadine for the prevention of itching associated with allergic conjunctivitis. Ann Pharmacother. 2012 Jul-Aug;46(7-8):1025-32. doi: 10.1345/aph.1Q755. Epub 2012 Jul 17.
  • PMID: 22035879
    Simons FE, Simons KJ: Histamine and H1-antihistamines: celebrating a century of progress. J Allergy Clin Immunol. 2011 Dec;128(6):1139-1150.e4. doi: 10.1016/j.jaci.2011.09.005. Epub 2011 Oct 27.
  • PMID: 21752782
    Hussar DA, Samuel J: Vilazodone hydrochloride, linagliptin, and alcaftadine. J Am Pharm Assoc (2003). 2011 Jul-Aug;51(4):557-9. doi: 10.1331/JAPhA.2011.11534.

Contoh Produk & Brand

Produk: 8 • International brands: 0
Produk
  • Alcaftadine
    Solution / drops • 2.5 mg/1mL • Ophthalmic • US • Generic • OTC • Approved
  • Alcaftadine
    Solution / drops • 2.5 mg/1mL • Ophthalmic • US • Generic • OTC • Approved
  • Alcaftadine
    Solution / drops • 2.5 mg/1mL • Ophthalmic • US • Generic • OTC • Approved
  • Lastacaft
    Solution • 2.5 mg/1mL • Ophthalmic • US • Approved
  • Lastacaft
    Solution / drops • 2.5 mg/1mL • Ophthalmic • US • Approved
  • Lastacaft
    Solution / drops • 2.5 mg/1mL • Ophthalmic • US • Approved
  • Lastacaft
    Solution / drops • 2.5 mg/1mL • Ophthalmic • US • Approved
  • Lastacaft
    Solution / drops • 2.5 mg/1mL • Ophthalmic • US • OTC • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul