Bafilomycin A1

DB06733

small molecule experimental

Deskripsi

The bafilomycins refer to a category of toxic macrolide antibiotics that are derivatives of Streptomyces griseus. These compounds all appear in the same fermentation and have similar biological activity. Bafilomycins are specific inhibitors of vacuolar-type H+-ATPase. (V-ATPase). The most commonly utilized bafilomycin is bafilomycin A1. This is a useful tool as it can prevent the re-acidification of synaptic vesicles once they have undergone exocytosis.

Struktur Molekul 2D

Berat 622.84
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

14 Data
Dicoumarol The therapeutic efficacy of Dicoumarol can be increased when used in combination with Bafilomycin A1.
Phenindione The therapeutic efficacy of Phenindione can be increased when used in combination with Bafilomycin A1.
Warfarin The therapeutic efficacy of Warfarin can be increased when used in combination with Bafilomycin A1.
Phenprocoumon The therapeutic efficacy of Phenprocoumon can be increased when used in combination with Bafilomycin A1.
Acenocoumarol The therapeutic efficacy of Acenocoumarol can be increased when used in combination with Bafilomycin A1.
4-hydroxycoumarin The therapeutic efficacy of 4-hydroxycoumarin can be increased when used in combination with Bafilomycin A1.
Coumarin The therapeutic efficacy of Coumarin can be increased when used in combination with Bafilomycin A1.
(R)-warfarin The therapeutic efficacy of (R)-warfarin can be increased when used in combination with Bafilomycin A1.
Ethyl biscoumacetate The therapeutic efficacy of Ethyl biscoumacetate can be increased when used in combination with Bafilomycin A1.
Fluindione The therapeutic efficacy of Fluindione can be increased when used in combination with Bafilomycin A1.
Clorindione The therapeutic efficacy of Clorindione can be increased when used in combination with Bafilomycin A1.
Diphenadione The therapeutic efficacy of Diphenadione can be increased when used in combination with Bafilomycin A1.
Tioclomarol The therapeutic efficacy of Tioclomarol can be increased when used in combination with Bafilomycin A1.
(S)-Warfarin The therapeutic efficacy of (S)-Warfarin can be increased when used in combination with Bafilomycin A1.

Target Protein

V-type proton ATPase catalytic subunit A ATP6V1A

Referensi & Sumber

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Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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