Sparteine

DB06727

small molecule experimental withdrawn

Deskripsi

Sparteine is a plant alkaloid derived from Cytisus scoparius and Lupinus mutabilis which may chelate calcium and magnesium. It is a sodium channel blocker, so it falls in the category of class 1a antiarrhythmic agents. Sparteine is not currently FDA-approved for human use, and its salt, sparteine sulfate, is one of the products that have been withdrawn or removed from the market for reasons of safety or effectiveness.L43942

Struktur Molekul 2D

Berat 234.387
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

464 Data
Amiodarone Amiodarone may increase the QTc-prolonging activities of Sparteine.
Fingolimod Fingolimod may increase the arrhythmogenic activities of Sparteine.
Propafenone Propafenone may increase the arrhythmogenic activities of Sparteine.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Sparteine.
Mirabegron The serum concentration of Sparteine can be increased when it is combined with Mirabegron.
Dofetilide Dofetilide may increase the arrhythmogenic activities of Sparteine.
Isradipine Isradipine may increase the arrhythmogenic activities of Sparteine.
Disopyramide Disopyramide may increase the arrhythmogenic activities of Sparteine.
Ibutilide Ibutilide may increase the arrhythmogenic activities of Sparteine.
Trimethadione Trimethadione may increase the arrhythmogenic activities of Sparteine.
Digoxin Digoxin may increase the arrhythmogenic activities of Sparteine.
Nimodipine Nimodipine may increase the arrhythmogenic activities of Sparteine.
Nisoldipine Nisoldipine may increase the arrhythmogenic activities of Sparteine.
Hyoscyamine Hyoscyamine may increase the arrhythmogenic activities of Sparteine.
Acetyldigitoxin Acetyldigitoxin may increase the arrhythmogenic activities of Sparteine.
Lamotrigine Lamotrigine may increase the arrhythmogenic activities of Sparteine.
Atropine Atropine may increase the arrhythmogenic activities of Sparteine.
Ethosuximide Ethosuximide may increase the arrhythmogenic activities of Sparteine.
Adenosine Adenosine may increase the arrhythmogenic activities of Sparteine.
Magnesium sulfate Magnesium sulfate may increase the arrhythmogenic activities of Sparteine.
Losartan Losartan may increase the arrhythmogenic activities of Sparteine.
Moricizine Moricizine may increase the arrhythmogenic activities of Sparteine.
Levomenthol Levomenthol may increase the arrhythmogenic activities of Sparteine.
Zonisamide Zonisamide may increase the arrhythmogenic activities of Sparteine.
Levosimendan Levosimendan may increase the arrhythmogenic activities of Sparteine.
Nitrendipine Nitrendipine may increase the arrhythmogenic activities of Sparteine.
Tocainide Tocainide may increase the arrhythmogenic activities of Sparteine.
Deslanoside Deslanoside may increase the arrhythmogenic activities of Sparteine.
Bretylium Bretylium may increase the arrhythmogenic activities of Sparteine.
Digitoxin Digitoxin may increase the arrhythmogenic activities of Sparteine.
Ajmaline Ajmaline may increase the arrhythmogenic activities of Sparteine.
Dexpropranolol Dexpropranolol may increase the arrhythmogenic activities of Sparteine.
Nimesulide Nimesulide may increase the arrhythmogenic activities of Sparteine.
Prenylamine Prenylamine may increase the arrhythmogenic activities of Sparteine.
Cyclandelate Cyclandelate may increase the arrhythmogenic activities of Sparteine.
Fluspirilene Fluspirilene may increase the arrhythmogenic activities of Sparteine.
Azimilide Azimilide may increase the arrhythmogenic activities of Sparteine.
Methsuximide Methsuximide may increase the arrhythmogenic activities of Sparteine.
Seletracetam Seletracetam may increase the arrhythmogenic activities of Sparteine.
Nylidrin Nylidrin may increase the arrhythmogenic activities of Sparteine.
Tedisamil Tedisamil may increase the arrhythmogenic activities of Sparteine.
Ziconotide Ziconotide may increase the arrhythmogenic activities of Sparteine.
Dotarizine Dotarizine may increase the arrhythmogenic activities of Sparteine.
Cariporide Cariporide may increase the arrhythmogenic activities of Sparteine.
Xylometazoline Xylometazoline may increase the arrhythmogenic activities of Sparteine.
Nilvadipine Nilvadipine may increase the arrhythmogenic activities of Sparteine.
Carteolol Sparteine may increase the arrhythmogenic activities of Carteolol.
Metipranolol Sparteine may increase the arrhythmogenic activities of Metipranolol.
Tranilast Sparteine may increase the arrhythmogenic activities of Tranilast.
Fasudil Sparteine may increase the arrhythmogenic activities of Fasudil.
Agmatine Sparteine may increase the arrhythmogenic activities of Agmatine.
Fendiline Sparteine may increase the arrhythmogenic activities of Fendiline.
Eperisone Sparteine may increase the arrhythmogenic activities of Eperisone.
Trimebutine Sparteine may increase the arrhythmogenic activities of Trimebutine.
Pinaverium Sparteine may increase the arrhythmogenic activities of Pinaverium.
Nicorandil Sparteine may increase the arrhythmogenic activities of Nicorandil.
Barnidipine Sparteine may increase the arrhythmogenic activities of Barnidipine.
Aranidipine Sparteine may increase the arrhythmogenic activities of Aranidipine.
Azelnidipine Sparteine may increase the arrhythmogenic activities of Azelnidipine.
Benidipine Sparteine may increase the arrhythmogenic activities of Benidipine.
Cilnidipine Sparteine may increase the arrhythmogenic activities of Cilnidipine.
Darodipine Sparteine may increase the arrhythmogenic activities of Darodipine.
Efonidipine Sparteine may increase the arrhythmogenic activities of Efonidipine.
Lacidipine Sparteine may increase the arrhythmogenic activities of Lacidipine.
Niguldipine Sparteine may increase the arrhythmogenic activities of Niguldipine.
Niludipine Sparteine may increase the arrhythmogenic activities of Niludipine.
Tropisetron Sparteine may increase the arrhythmogenic activities of Tropisetron.
Carboxyamidotriazole Sparteine may increase the arrhythmogenic activities of Carboxyamidotriazole.
Naftopidil Sparteine may increase the arrhythmogenic activities of Naftopidil.
Tetrahydropalmatine Sparteine may increase the arrhythmogenic activities of Tetrahydropalmatine.
Vinpocetine Sparteine may increase the arrhythmogenic activities of Vinpocetine.
Simendan Sparteine may increase the arrhythmogenic activities of Simendan.
Spiradoline Sparteine may increase the arrhythmogenic activities of Spiradoline.
Pilsicainide Sparteine may increase the arrhythmogenic activities of Pilsicainide.
Cicletanine Sparteine may increase the arrhythmogenic activities of Cicletanine.
Gallopamil Sparteine may increase the arrhythmogenic activities of Gallopamil.
Cymarin Sparteine may increase the arrhythmogenic activities of Cymarin.
Cibenzoline Sparteine may increase the arrhythmogenic activities of Cibenzoline.
Metildigoxin Sparteine may increase the arrhythmogenic activities of Metildigoxin.
Bencyclane Sparteine may increase the arrhythmogenic activities of Bencyclane.
Otilonium Sparteine may increase the arrhythmogenic activities of Otilonium.
Nizofenone Sparteine may increase the arrhythmogenic activities of Nizofenone.
Prajmaline Sparteine may increase the arrhythmogenic activities of Prajmaline.
Tiracizine Sparteine may increase the arrhythmogenic activities of Tiracizine.
Ethacizine Sparteine may increase the arrhythmogenic activities of Ethacizine.
Lorajmine Sparteine may increase the arrhythmogenic activities of Lorajmine.
Bunaftine Sparteine may increase the arrhythmogenic activities of Bunaftine.
Lorcainide Sparteine may increase the arrhythmogenic activities of Lorcainide.
Acetyldigoxin Sparteine may increase the arrhythmogenic activities of Acetyldigoxin.
Hydroquinine Sparteine may increase the arrhythmogenic activities of Hydroquinine.
Terodiline Sparteine may increase the arrhythmogenic activities of Terodiline.
Bioallethrin Sparteine may increase the arrhythmogenic activities of Bioallethrin.
Lidoflazine Sparteine may increase the arrhythmogenic activities of Lidoflazine.
Penfluridol Sparteine may increase the arrhythmogenic activities of Penfluridol.
Caroverine Sparteine may increase the arrhythmogenic activities of Caroverine.
Fosfructose Sparteine may increase the arrhythmogenic activities of Fosfructose.
WIN 55212-2 Sparteine may increase the arrhythmogenic activities of WIN 55212-2.
Fish oil Sparteine may increase the arrhythmogenic activities of Fish oil.
Dexverapamil Sparteine may increase the arrhythmogenic activities of Dexverapamil.
Emopamil Sparteine may increase the arrhythmogenic activities of Emopamil.

Referensi & Sumber

Synthesis reference: Bernd Hachmeister, "Process for the production of 17-hydroxysparteine by oxidation of sparteine with a permanganate." U.S. Patent US4237295, issued June, 1975.

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