Calcium carbonate

DB06724

small molecule approved investigational

Deskripsi

Calcium carbonate is an inorganic salt used as an antacid. It is a basic compound that acts by neutralizing hydrochloric acid in gastric secretions. Subsequent increases in pH may inhibit the action of pepsin. An increase in bicarbonate ions and prostaglandins may also confer cytoprotective effects. Calcium carbonate may also be used as a nutritional supplement or to treat hypocalcemia.

Struktur Molekul 2D

Berat 100.087
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi Calcium is rapidly distributed taken up by skeletal tissues following absorption and distribution into extracellular fluids. Bone contains 99% of the body's calcium and the remaining 1% is approximately equally distributed between intracellular and extracellular fluids.
Klirens (Clearance) -

Absorpsi

Maximal absorption occurs at doses of 500 mg or less taken with food. Oral bioavailability depends on intestinal pH, the presence of food and dosage.

Metabolisme

None.

Rute Eliminasi

Excreted mainly in the feces. The majority of renally filtered calcium is reabsorbed in the ascending limb of the loop of Henle and the proximal and distal convoluted tubules. Also secreted by sweat glands.

Interaksi Makanan

1 Data
  • 1. Take with or without food. Food increases the absorption of calcium carbonate, which may be advantageous in its use as a calcium supplement.

Interaksi Obat

364 Data
Atazanavir Calcium carbonate can cause a decrease in the absorption of Atazanavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Bosutinib Calcium carbonate can cause a decrease in the absorption of Bosutinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefditoren The serum concentration of Cefditoren can be decreased when it is combined with Calcium carbonate.
Dabigatran etexilate Calcium carbonate can cause a decrease in the absorption of Dabigatran etexilate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dabrafenib Calcium carbonate can cause a decrease in the absorption of Dabrafenib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dasatinib Calcium carbonate can cause a decrease in the absorption of Dasatinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Delavirdine Calcium carbonate can cause a decrease in the absorption of Delavirdine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Erlotinib Calcium carbonate can cause a decrease in the absorption of Erlotinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gefitinib Calcium carbonate can cause a decrease in the absorption of Gefitinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Itraconazole Calcium carbonate can cause a decrease in the absorption of Itraconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ledipasvir Calcium carbonate can cause a decrease in the absorption of Ledipasvir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Methylphenidate Calcium carbonate can cause an increase in the absorption of Methylphenidate resulting in an increased serum concentration and potentially a worsening of adverse effects.
Pazopanib Calcium carbonate can cause a decrease in the absorption of Pazopanib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Riociguat Calcium carbonate can cause a decrease in the absorption of Riociguat resulting in a reduced serum concentration and potentially a decrease in efficacy.
Grepafloxacin Calcium carbonate can cause a decrease in the absorption of Grepafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Enoxacin Calcium carbonate can cause a decrease in the absorption of Enoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Pefloxacin Calcium carbonate can cause a decrease in the absorption of Pefloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Trovafloxacin Calcium carbonate can cause a decrease in the absorption of Trovafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nalidixic acid Calcium carbonate can cause a decrease in the absorption of Nalidixic acid resulting in a reduced serum concentration and potentially a decrease in efficacy.
Rosoxacin Calcium carbonate can cause a decrease in the absorption of Rosoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cinoxacin Calcium carbonate can cause a decrease in the absorption of Cinoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lomefloxacin Calcium carbonate can cause a decrease in the absorption of Lomefloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gatifloxacin Calcium carbonate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Norfloxacin Calcium carbonate can cause a decrease in the absorption of Norfloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gemifloxacin Calcium carbonate can cause a decrease in the absorption of Gemifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ofloxacin Calcium carbonate can cause a decrease in the absorption of Ofloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sparfloxacin Calcium carbonate can cause a decrease in the absorption of Sparfloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Temafloxacin Calcium carbonate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Fleroxacin Calcium carbonate can cause a decrease in the absorption of Fleroxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Technetium Tc-99m ciprofloxacin Calcium carbonate can cause a decrease in the absorption of Technetium Tc-99m ciprofloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Garenoxacin Calcium carbonate can cause a decrease in the absorption of Garenoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nemonoxacin Calcium carbonate can cause a decrease in the absorption of Nemonoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Flumequine Calcium carbonate can cause a decrease in the absorption of Flumequine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Enrofloxacin Calcium carbonate can cause a decrease in the absorption of Enrofloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Orbifloxacin Calcium carbonate can cause a decrease in the absorption of Orbifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sarafloxacin Calcium carbonate can cause a decrease in the absorption of Sarafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Difloxacin Calcium carbonate can cause a decrease in the absorption of Difloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Pazufloxacin Calcium carbonate can cause a decrease in the absorption of Pazufloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Prulifloxacin Calcium carbonate can cause a decrease in the absorption of Prulifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Delafloxacin Calcium carbonate can cause a decrease in the absorption of Delafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sitafloxacin Calcium carbonate can cause a decrease in the absorption of Sitafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Oxolinic acid Calcium carbonate can cause a decrease in the absorption of Oxolinic acid resulting in a reduced serum concentration and potentially a decrease in efficacy.
Rufloxacin Calcium carbonate can cause a decrease in the absorption of Rufloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Pipemidic acid Calcium carbonate can cause a decrease in the absorption of Pipemidic acid resulting in a reduced serum concentration and potentially a decrease in efficacy.
Deferiprone The serum concentration of Deferiprone can be decreased when it is combined with Calcium carbonate.
Dobutamine The therapeutic efficacy of Dobutamine can be decreased when used in combination with Calcium carbonate.
Dolutegravir The serum concentration of Dolutegravir can be decreased when it is combined with Calcium carbonate.
Eltrombopag The serum concentration of Eltrombopag can be decreased when it is combined with Calcium carbonate.
Estramustine Calcium carbonate can cause a decrease in the absorption of Estramustine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Levothyroxine Calcium carbonate can cause a decrease in the absorption of Levothyroxine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium acetate The risk or severity of adverse effects can be increased when Calcium carbonate is combined with Calcium acetate.
Tolevamer The risk or severity of adverse effects can be increased when Tolevamer is combined with Calcium carbonate.
Bisacodyl The therapeutic efficacy of Bisacodyl can be decreased when used in combination with Calcium carbonate.
Captopril Calcium carbonate can cause a decrease in the absorption of Captopril resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefpodoxime The serum concentration of Cefpodoxime can be decreased when it is combined with Calcium carbonate.
Cefuroxime The serum concentration of Cefuroxime can be decreased when it is combined with Calcium carbonate.
Chloroquine Calcium carbonate can cause a decrease in the absorption of Chloroquine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Elvitegravir Calcium carbonate can cause a decrease in the absorption of Elvitegravir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Hyoscyamine Calcium carbonate can cause a decrease in the absorption of Hyoscyamine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Rifampin Calcium carbonate can cause a decrease in the absorption of Rifampicin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mecamylamine Calcium carbonate may decrease the excretion rate of Mecamylamine which could result in a higher serum level.
Memantine Calcium carbonate may decrease the excretion rate of Memantine which could result in a higher serum level.
Penicillamine Calcium carbonate can cause a decrease in the absorption of Penicillamine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Quinidine Calcium carbonate may decrease the excretion rate of Quinidine which could result in a higher serum level.
Sulpiride The therapeutic efficacy of Sulpiride can be increased when used in combination with Calcium carbonate.
Allopurinol The therapeutic efficacy of Allopurinol can be decreased when used in combination with Calcium carbonate.
Raltegravir The serum concentration of Raltegravir can be decreased when it is combined with Calcium carbonate.
Mesalazine Calcium carbonate can cause a decrease in the absorption of Mesalazine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mycophenolic acid Calcium carbonate can cause a decrease in the absorption of Mycophenolic acid resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cysteamine The bioavailability of Cysteamine can be decreased when combined with Calcium carbonate.
Ketoconazole Calcium carbonate can cause a decrease in the absorption of Ketoconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Acetyldigitoxin Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Acetyldigitoxin.
Deslanoside Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Deslanoside.
Ouabain Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Ouabain.
Digitoxin Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Digitoxin.
Oleandrin Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Oleandrin.
Cymarin Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Cymarin.
Proscillaridin Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Proscillaridin.
Lanatoside C Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Lanatoside C.
Gitoformate Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Gitoformate.
Peruvoside Calcium carbonate may increase the arrhythmogenic and cardiotoxic activities of Peruvoside.
Strontium ranelate The serum concentration of Strontium ranelate can be decreased when it is combined with Calcium carbonate.
Methyclothiazide Methyclothiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Chlorthalidone Chlorthalidone may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Bendroflumethiazide Bendroflumethiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Metolazone Metolazone may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Benzthiazide Benzthiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Hydroflumethiazide Hydroflumethiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Indapamide Indapamide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Chlorothiazide Chlorothiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Hydrochlorothiazide Hydrochlorothiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Trichlormethiazide Trichlormethiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Polythiazide Polythiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Quinethazone Quinethazone may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Cyclopenthiazide Cyclopenthiazide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Epitizide Epitizide may decrease the excretion rate of Calcium carbonate which could result in a higher serum level.
Calcitriol The risk or severity of adverse effects can be increased when Calcitriol is combined with Calcium carbonate.
Calcifediol The risk or severity of adverse effects can be increased when Calcifediol is combined with Calcium carbonate.
Paricalcitol The risk or severity of adverse effects can be increased when Paricalcitol is combined with Calcium carbonate.
Dihydrotachysterol The risk or severity of adverse effects can be increased when Dihydrotachysterol is combined with Calcium carbonate.

Referensi & Sumber

Synthesis reference: Nobuo Someya, Tadao Kitazato, Takao Fujikawa, Yasuo Manabe, "Sintered body of calcium carbonate and process for producing same." U.S. Patent US5187125, issued May, 1940.

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