Peringatan Keamanan

Buserelin may induce early, transient increase in serum testosterone or estradiol which can lead in the exacerbation of signs and symptoms of metastatic prostate cancer or endometriosis. Adverse reactions reported at more than 10% occurrence include headache, loss of libido in patients with prostate cancer, hot flashes, hypermenorrhea, decreased libido in prostate cancer and endometriosis, flatulence, impotence, vaginal dryness, back pain and nasal mucosa irritation.

Buserelin

DB06719

biotech approved investigational

Deskripsi

Buserelin is a synthetic peptide analog of the luteinizing hormone-releasing hormone (LHRH) agonist, which stimulates the pituitary gland's gonadotrophin-releasing hormone receptor (GnRHR). It is used in prostate cancer treatment.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The elimination half-life is approximately 50 to 80 minutes following intravenous administration, 80 minutes after subcutaneous administration and approximately 1 to 2 hours after intranasal administration.
Volume Distribusi Buserelin circulates in serum predominantly in intact active form. Preferred accumulation is preferentially in the liver and kidneys as well as in the anterior pituitary lobe, the biological target organ.
Klirens (Clearance) -

Absorpsi

Buserelin is water soluble and readily absorbed after subcutaneous injection (70% bioavailable). However, bioavailability after oral absorption. When administered correctly via the nasal route, it may be absorbed in the nasal mucosa to achieve sufficient plasma levels.

Metabolisme

It is metabolized and subsequently inactivated by peptidase (pyroglutamyl peptidase and chymotrypsin-like endopeptidase) in the liver and kidneys as well as in the gastrointestinal tract. In the pituitary gland, it is inactivated by membrane-located enzymes.

Rute Eliminasi

Buserelin and its inactive metabolites are excreted via the renal and biliary routes. In man it is excreted in urine at 50% in its intact form.

Interaksi Obat

494 Data
Corifollitropin alfa The therapeutic efficacy of Corifollitropin alfa can be increased when used in combination with Buserelin.
Choline C 11 Buserelin may decrease effectiveness of Choline C 11 as a diagnostic agent.
Capromab pendetide Buserelin may decrease effectiveness of Capromab pendetide as a diagnostic agent.
Insulin human The therapeutic efficacy of Insulin human can be decreased when used in combination with Buserelin.
Insulin lispro The therapeutic efficacy of Insulin lispro can be decreased when used in combination with Buserelin.
Insulin glargine The therapeutic efficacy of Insulin glargine can be decreased when used in combination with Buserelin.
Insulin pork The therapeutic efficacy of Insulin pork can be decreased when used in combination with Buserelin.
Troglitazone The therapeutic efficacy of Troglitazone can be decreased when used in combination with Buserelin.
Glimepiride The therapeutic efficacy of Glimepiride can be decreased when used in combination with Buserelin.
Acarbose The therapeutic efficacy of Acarbose can be decreased when used in combination with Buserelin.
Sulfadiazine The therapeutic efficacy of Sulfadiazine can be decreased when used in combination with Buserelin.
Rosiglitazone The therapeutic efficacy of Rosiglitazone can be decreased when used in combination with Buserelin.
Acetohexamide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Buserelin.
Miglitol The therapeutic efficacy of Miglitol can be decreased when used in combination with Buserelin.
Chlorpropamide The therapeutic efficacy of Chlorpropamide can be decreased when used in combination with Buserelin.
Nateglinide The therapeutic efficacy of Nateglinide can be decreased when used in combination with Buserelin.
Tolazamide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Buserelin.
Repaglinide The therapeutic efficacy of Repaglinide can be decreased when used in combination with Buserelin.
Phenformin The therapeutic efficacy of Phenformin can be decreased when used in combination with Buserelin.
Sulfamethoxazole The therapeutic efficacy of Sulfamethoxazole can be decreased when used in combination with Buserelin.
Glyburide The therapeutic efficacy of Glyburide can be decreased when used in combination with Buserelin.
Glipizide The therapeutic efficacy of Glipizide can be decreased when used in combination with Buserelin.
Gliclazide The therapeutic efficacy of Gliclazide can be decreased when used in combination with Buserelin.
Tolbutamide The therapeutic efficacy of Tolbutamide can be decreased when used in combination with Buserelin.
Pioglitazone The therapeutic efficacy of Pioglitazone can be decreased when used in combination with Buserelin.
Bromocriptine The therapeutic efficacy of Bromocriptine can be decreased when used in combination with Buserelin.
Gliquidone The therapeutic efficacy of Gliquidone can be decreased when used in combination with Buserelin.
Mitiglinide The therapeutic efficacy of Mitiglinide can be decreased when used in combination with Buserelin.
Sitagliptin The therapeutic efficacy of Sitagliptin can be decreased when used in combination with Buserelin.
Sunitinib The therapeutic efficacy of Sunitinib can be decreased when used in combination with Buserelin.
Exenatide The therapeutic efficacy of Exenatide can be decreased when used in combination with Buserelin.
Mecasermin The therapeutic efficacy of Mecasermin can be decreased when used in combination with Buserelin.
Pramlintide The therapeutic efficacy of Pramlintide can be decreased when used in combination with Buserelin.
Glisoxepide The therapeutic efficacy of Glisoxepide can be decreased when used in combination with Buserelin.
Insulin aspart The therapeutic efficacy of Insulin aspart can be decreased when used in combination with Buserelin.
Insulin detemir The therapeutic efficacy of Insulin detemir can be decreased when used in combination with Buserelin.
Insulin glulisine The therapeutic efficacy of Insulin glulisine can be decreased when used in combination with Buserelin.
Glymidine The therapeutic efficacy of Glymidine can be decreased when used in combination with Buserelin.
AICA ribonucleotide The therapeutic efficacy of AICA ribonucleotide can be decreased when used in combination with Buserelin.
Buformin The therapeutic efficacy of Buformin can be decreased when used in combination with Buserelin.
Vildagliptin The therapeutic efficacy of Vildagliptin can be decreased when used in combination with Buserelin.
Voglibose The therapeutic efficacy of Voglibose can be decreased when used in combination with Buserelin.
NN344 The therapeutic efficacy of NN344 can be decreased when used in combination with Buserelin.
AMG-222 The therapeutic efficacy of AMG-222 can be decreased when used in combination with Buserelin.
Bisegliptin The therapeutic efficacy of Bisegliptin can be decreased when used in combination with Buserelin.
Alogliptin The therapeutic efficacy of Alogliptin can be decreased when used in combination with Buserelin.
Dapagliflozin The therapeutic efficacy of Dapagliflozin can be decreased when used in combination with Buserelin.
Saxagliptin The therapeutic efficacy of Saxagliptin can be decreased when used in combination with Buserelin.
Liraglutide The therapeutic efficacy of Liraglutide can be decreased when used in combination with Buserelin.
Gosogliptin The therapeutic efficacy of Gosogliptin can be decreased when used in combination with Buserelin.
Linagliptin The therapeutic efficacy of Linagliptin can be decreased when used in combination with Buserelin.
Canagliflozin The therapeutic efficacy of Canagliflozin can be decreased when used in combination with Buserelin.
Glibornuride The therapeutic efficacy of Glibornuride can be decreased when used in combination with Buserelin.
Benfluorex The therapeutic efficacy of Benfluorex can be decreased when used in combination with Buserelin.
Empagliflozin The therapeutic efficacy of Empagliflozin can be decreased when used in combination with Buserelin.
Albiglutide The therapeutic efficacy of Albiglutide can be decreased when used in combination with Buserelin.
Dulaglutide The therapeutic efficacy of Dulaglutide can be decreased when used in combination with Buserelin.
Lobeglitazone The therapeutic efficacy of Lobeglitazone can be decreased when used in combination with Buserelin.
Netoglitazone The therapeutic efficacy of Netoglitazone can be decreased when used in combination with Buserelin.
Rivoglitazone The therapeutic efficacy of Rivoglitazone can be decreased when used in combination with Buserelin.
Ciglitazone The therapeutic efficacy of Ciglitazone can be decreased when used in combination with Buserelin.
Lixisenatide The therapeutic efficacy of Lixisenatide can be decreased when used in combination with Buserelin.
Insulin beef The therapeutic efficacy of Insulin beef can be decreased when used in combination with Buserelin.
Insulin degludec The therapeutic efficacy of Insulin degludec can be decreased when used in combination with Buserelin.
Insulin peglispro The therapeutic efficacy of Insulin peglispro can be decreased when used in combination with Buserelin.
Insulin tregopil The therapeutic efficacy of Insulin tregopil can be decreased when used in combination with Buserelin.
Ipragliflozin The therapeutic efficacy of Ipragliflozin can be decreased when used in combination with Buserelin.
Dutogliptin The therapeutic efficacy of Dutogliptin can be decreased when used in combination with Buserelin.
Allicin The therapeutic efficacy of Allicin can be decreased when used in combination with Buserelin.
Tofogliflozin The therapeutic efficacy of Tofogliflozin can be decreased when used in combination with Buserelin.
Ertugliflozin The therapeutic efficacy of Ertugliflozin can be decreased when used in combination with Buserelin.
2,4-thiazolidinedione The therapeutic efficacy of 2,4-thiazolidinedione can be decreased when used in combination with Buserelin.
Teneligliptin The therapeutic efficacy of Teneligliptin can be decreased when used in combination with Buserelin.
Omarigliptin The therapeutic efficacy of Omarigliptin can be decreased when used in combination with Buserelin.
Carmegliptin The therapeutic efficacy of Carmegliptin can be decreased when used in combination with Buserelin.
Gemigliptin The therapeutic efficacy of Gemigliptin can be decreased when used in combination with Buserelin.
Anagliptin The therapeutic efficacy of Anagliptin can be decreased when used in combination with Buserelin.
Evogliptin The therapeutic efficacy of Evogliptin can be decreased when used in combination with Buserelin.
Sotagliflozin The therapeutic efficacy of Sotagliflozin can be decreased when used in combination with Buserelin.
Balaglitazone The therapeutic efficacy of Balaglitazone can be decreased when used in combination with Buserelin.
Remogliflozin etabonate The therapeutic efficacy of Remogliflozin etabonate can be decreased when used in combination with Buserelin.
Carbutamide The therapeutic efficacy of Carbutamide can be decreased when used in combination with Buserelin.
Guar gum The therapeutic efficacy of Guar gum can be decreased when used in combination with Buserelin.
Metahexamide The therapeutic efficacy of Metahexamide can be decreased when used in combination with Buserelin.
Semaglutide The therapeutic efficacy of Semaglutide can be decreased when used in combination with Buserelin.
Taspoglutide The therapeutic efficacy of Taspoglutide can be decreased when used in combination with Buserelin.
Englitazone The therapeutic efficacy of Englitazone can be decreased when used in combination with Buserelin.
Tirzepatide The therapeutic efficacy of Tirzepatide can be decreased when used in combination with Buserelin.
Gastric inhibitory polypeptide The therapeutic efficacy of Gastric inhibitory polypeptide can be decreased when used in combination with Buserelin.
Leuprolide The risk or severity of QTc prolongation can be increased when Buserelin is combined with Leuprolide.
Goserelin The risk or severity of QTc prolongation can be increased when Buserelin is combined with Goserelin.
Erythromycin The risk or severity of QTc prolongation can be increased when Buserelin is combined with Erythromycin.
Azithromycin The risk or severity of QTc prolongation can be increased when Buserelin is combined with Azithromycin.
Moxifloxacin The risk or severity of QTc prolongation can be increased when Buserelin is combined with Moxifloxacin.
Ranolazine The risk or severity of QTc prolongation can be increased when Buserelin is combined with Ranolazine.
Sulfisoxazole The therapeutic efficacy of Sulfisoxazole can be decreased when used in combination with Buserelin.
Amitriptyline The risk or severity of QTc prolongation can be increased when Buserelin is combined with Amitriptyline.
Methadone The risk or severity of QTc prolongation can be increased when Buserelin is combined with Methadone.
Diltiazem The risk or severity of QTc prolongation can be increased when Buserelin is combined with Diltiazem.
Clozapine The risk or severity of QTc prolongation can be increased when Buserelin is combined with Clozapine.

Target Protein

Lutropin-choriogonadotropic hormone receptor LHCGR
Gonadotropin-releasing hormone receptor GNRHR

Referensi & Sumber

Link

Contoh Produk & Brand

Produk: 7 • International brands: 1
Produk
  • Suprefact
    Solution • 100 mcg / act • Nasal • Canada • Approved
  • Suprefact
    Solution • 1 mg / mL • Subcutaneous • Canada • Approved
  • Suprefact Depot 2 Months
    Implant • 6.3 mg • Subcutaneous • Canada • Approved
  • Suprefact Depot 3 Months
    Implant • 9.45 mg • Subcutaneous • Canada • Approved
  • Suprefact Inj 1mg/ml
    Liquid • 1 mg / mL • Subcutaneous • Canada • Approved
  • Suprefact Intranasal Solution 1mg/ml
    Spray • 1 mg / mL • Nasal • Canada • Approved
  • Suprefact Liq 1mg/ml
    Liquid • 1 mg / mL • Nasal • Canada • Approved
International Brands
  • Cinnafact — Cinnagen

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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