Peringatan Keamanan

Common side effects of combination artemether/lumefantrine therapy in adults include headache, anorexia, dizziness, and asthenia. Common side effects in children include pyrexia, cough, vomiting, anorexia, and headache. Possible serious adverse effects include QT prolongation, bullous eruption, urticaria, splenomegaly (9%), hepatomegaly (adults, 9%; children, 6%), hypersensitivty reaction, and angioedema.

Lumefantrine

DB06708

small molecule approved

Deskripsi

Lumefantrine is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with artemether for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of Plasmodium spp. and may be used to treat infections caused by P. falciparum and unidentified Plasmodium species, including infections acquired in chloroquine-resistant areas.

Struktur Molekul 2D

Berat 528.94
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) ~ 4.5 days
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Food increases absorption.

Metabolisme

Extensively metabolized in the liver primarily by cytochrome P450 3A4. The major metabolite found in plasma is desbutyl-lumefantrine.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid grapefruit products.
  • 2. Take with food. Food increases absorption.

Interaksi Obat

648 Data
Pyrimethamine The risk or severity of QTc prolongation can be increased when Pyrimethamine is combined with Lumefantrine.
Dapsone The risk or severity of QTc prolongation can be increased when Dapsone is combined with Lumefantrine.
Mefloquine The risk or severity of QTc prolongation can be increased when Mefloquine is combined with Lumefantrine.
Quinine The risk or severity of QTc prolongation can be increased when Quinine is combined with Lumefantrine.
Chloroquine The risk or severity of QTc prolongation can be increased when Chloroquine is combined with Lumefantrine.
Amodiaquine The risk or severity of QTc prolongation can be increased when Amodiaquine is combined with Lumefantrine.
Quinidine The risk or severity of QTc prolongation can be increased when Quinidine is combined with Lumefantrine.
Primaquine The risk or severity of QTc prolongation can be increased when Primaquine is combined with Lumefantrine.
Quinacrine The risk or severity of QTc prolongation can be increased when Quinacrine is combined with Lumefantrine.
Atovaquone The risk or severity of QTc prolongation can be increased when Atovaquone is combined with Lumefantrine.
Proguanil The risk or severity of QTc prolongation can be increased when Proguanil is combined with Lumefantrine.
Sulfadoxine The risk or severity of QTc prolongation can be increased when Sulfadoxine is combined with Lumefantrine.
Hydroxychloroquine The risk or severity of QTc prolongation can be increased when Hydroxychloroquine is combined with Lumefantrine.
Tafenoquine The risk or severity of QTc prolongation can be increased when Tafenoquine is combined with Lumefantrine.
Artesunate The risk or severity of QTc prolongation can be increased when Artesunate is combined with Lumefantrine.
Artenimol The risk or severity of QTc prolongation can be increased when Artenimol is combined with Lumefantrine.
Artefenomel The risk or severity of QTc prolongation can be increased when Artefenomel is combined with Lumefantrine.
Chlorproguanil The risk or severity of QTc prolongation can be increased when Chlorproguanil is combined with Lumefantrine.
Mizoribine The risk or severity of QTc prolongation can be increased when Mizoribine is combined with Lumefantrine.
Pyronaridine The risk or severity of QTc prolongation can be increased when Pyronaridine is combined with Lumefantrine.
Artemisinin The risk or severity of QTc prolongation can be increased when Artemisinin is combined with Lumefantrine.
Artemotil The risk or severity of QTc prolongation can be increased when Artemotil is combined with Lumefantrine.
Piperaquine The risk or severity of QTc prolongation can be increased when Piperaquine is combined with Lumefantrine.
Tetrandrine The risk or severity of QTc prolongation can be increased when Tetrandrine is combined with Lumefantrine.
Cycloguanil The risk or severity of QTc prolongation can be increased when Cycloguanil is combined with Lumefantrine.
Brexpiprazole The metabolism of Brexpiprazole can be decreased when combined with Lumefantrine.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Lumefantrine.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Lumefantrine.
Halofantrine Lumefantrine may increase the QTc-prolonging activities of Halofantrine.
Thiethylperazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Thiethylperazine.
Triflupromazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Triflupromazine.
Fluphenazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Fluphenazine.
Moricizine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Moricizine.
Trifluoperazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Trifluoperazine.
Acetophenazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Acetophenazine.
Alimemazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Alimemazine.
Periciazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Periciazine.
Acepromazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Acepromazine.
Aceprometazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Aceprometazine.
Thioproperazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Thioproperazine.
BL-1020 The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with BL-1020.
Cyamemazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Cyamemazine.
Propiopromazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Propiopromazine.
Perazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Perazine.
Butaperazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Butaperazine.
Chlorproethazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Chlorproethazine.
Thiazinam The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Thiazinam.
Dixyrazine The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Dixyrazine.
Perphenazine enanthate The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Perphenazine enanthate.
St. John's Wort The serum concentration of Lumefantrine can be decreased when it is combined with St. John's Wort.
Leuprolide The risk or severity of QTc prolongation can be increased when Leuprolide is combined with Lumefantrine.
Goserelin The risk or severity of QTc prolongation can be increased when Goserelin is combined with Lumefantrine.
Erythromycin The serum concentration of Lumefantrine can be increased when it is combined with Erythromycin.
Azithromycin The risk or severity of QTc prolongation can be increased when Azithromycin is combined with Lumefantrine.
Moxifloxacin The risk or severity of QTc prolongation can be increased when Moxifloxacin is combined with Lumefantrine.
Sulfisoxazole The risk or severity of QTc prolongation can be increased when Sulfisoxazole is combined with Lumefantrine.
Sulpiride The risk or severity of QTc prolongation can be increased when Sulpiride is combined with Lumefantrine.
Nimodipine The risk or severity of QTc prolongation can be increased when Nimodipine is combined with Lumefantrine.
Droperidol The risk or severity of QTc prolongation can be increased when Droperidol is combined with Lumefantrine.
Oxaliplatin The risk or severity of QTc prolongation can be increased when Oxaliplatin is combined with Lumefantrine.
Ciprofloxacin The risk or severity of QTc prolongation can be increased when Ciprofloxacin is combined with Lumefantrine.
Fluorouracil The risk or severity of QTc prolongation can be increased when Fluorouracil is combined with Lumefantrine.
Perflutren The risk or severity of QTc prolongation can be increased when Perflutren is combined with Lumefantrine.
Atropine The risk or severity of QTc prolongation can be increased when Atropine is combined with Lumefantrine.
Adenosine The risk or severity of QTc prolongation can be increased when Adenosine is combined with Lumefantrine.
Gadobenic acid The risk or severity of QTc prolongation can be increased when Gadobenic acid is combined with Lumefantrine.
Carbinoxamine The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Lumefantrine.
Roxithromycin The risk or severity of QTc prolongation can be increased when Roxithromycin is combined with Lumefantrine.
Nalidixic acid The risk or severity of QTc prolongation can be increased when Nalidixic acid is combined with Lumefantrine.
Cinoxacin The risk or severity of QTc prolongation can be increased when Cinoxacin is combined with Lumefantrine.
Granisetron The risk or severity of QTc prolongation can be increased when Granisetron is combined with Lumefantrine.
Levosimendan The risk or severity of QTc prolongation can be increased when Levosimendan is combined with Lumefantrine.
Desloratadine The risk or severity of QTc prolongation can be increased when Desloratadine is combined with Lumefantrine.
Lomefloxacin The risk or severity of QTc prolongation can be increased when Lomefloxacin is combined with Lumefantrine.
Dimenhydrinate The risk or severity of QTc prolongation can be increased when Dimenhydrinate is combined with Lumefantrine.
Papaverine The risk or severity of QTc prolongation can be increased when Papaverine is combined with Lumefantrine.
Levofloxacin The risk or severity of QTc prolongation can be increased when Levofloxacin is combined with Lumefantrine.
Gemifloxacin The risk or severity of QTc prolongation can be increased when Gemifloxacin is combined with Lumefantrine.
Ofloxacin The risk or severity of QTc prolongation can be increased when Ofloxacin is combined with Lumefantrine.
Mibefradil The risk or severity of QTc prolongation can be increased when Mibefradil is combined with Lumefantrine.
Probucol The risk or severity of QTc prolongation can be increased when Probucol is combined with Lumefantrine.
Terlipressin The risk or severity of QTc prolongation can be increased when Terlipressin is combined with Lumefantrine.
Prenylamine The risk or severity of QTc prolongation can be increased when Prenylamine is combined with Lumefantrine.
Fluspirilene The risk or severity of QTc prolongation can be increased when Fluspirilene is combined with Lumefantrine.
Azimilide The risk or severity of QTc prolongation can be increased when Azimilide is combined with Lumefantrine.
Pracinostat The risk or severity of QTc prolongation can be increased when Pracinostat is combined with Lumefantrine.
Technetium Tc-99m ciprofloxacin The risk or severity of QTc prolongation can be increased when Technetium Tc-99m ciprofloxacin is combined with Lumefantrine.
Garenoxacin The risk or severity of QTc prolongation can be increased when Garenoxacin is combined with Lumefantrine.
Tedisamil The risk or severity of QTc prolongation can be increased when Tedisamil is combined with Lumefantrine.
Tucidinostat The risk or severity of QTc prolongation can be increased when Tucidinostat is combined with Lumefantrine.
Telavancin The risk or severity of QTc prolongation can be increased when Telavancin is combined with Lumefantrine.
Nemonoxacin The risk or severity of QTc prolongation can be increased when Nemonoxacin is combined with Lumefantrine.
Nilvadipine The risk or severity of QTc prolongation can be increased when Nilvadipine is combined with Lumefantrine.
Antazoline The risk or severity of QTc prolongation can be increased when Antazoline is combined with Lumefantrine.
Bedaquiline The risk or severity of QTc prolongation can be increased when Lumefantrine is combined with Bedaquiline.
Fendiline The risk or severity of QTc prolongation can be increased when Fendiline is combined with Lumefantrine.
Eperisone The risk or severity of QTc prolongation can be increased when Eperisone is combined with Lumefantrine.
Butriptyline The risk or severity of QTc prolongation can be increased when Butriptyline is combined with Lumefantrine.
Lenvatinib The risk or severity of QTc prolongation can be increased when Lenvatinib is combined with Lumefantrine.
Melperone The risk or severity of QTc prolongation can be increased when Melperone is combined with Lumefantrine.

Target Protein

Sodium/potassium-transporting ATPase subunit alpha-1 ATP1A1

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 3 • International brands: 0
Produk
  • Coartem
    Tablet • - • Oral • US • Approved
  • Coartem
    Tablet • - • Oral • US • Approved
  • Coartem
    Tablet • - • Oral • US • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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