Peringatan Keamanan

Oral mouse: LD50 = 300 mg/kg;
Oral, rabbit: LD50 = 3200 mg/kg;
Oral, rat: LD50=980 mg/kg.
The most common adverse reactions, dizziness, rash, pruritis, flushing, headache, and injection site hemorrhage occurred in < 1.3% of patients.

Iobenguane

DB06704

small molecule approved investigational

Deskripsi

Synthetic guanethidine derivative that locates phaeochromocytomas and neuroblastomas. The radioisotope used can either be iodine-123 for imaging or iodine-131 for destruction of tissues that metabolize noradrenaline. Iodine 123 is a cyclotron-produced radionuclide that decays to Te 123 by electron capture. Images are produced by a I123 MIBG scintigraphy. FDA approved on September 19, 2008.

Struktur Molekul 2D

Berat 275.0896
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Physical half life = 13.2 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Iobenguane rapidly clears from the blood and is highly retained in adrenergic tissues.

Metabolisme

Less than 10% of the dose is metabolized into m-iodohippuric acid (MIHA). However the mechanism in which this metabolite is produced is unknown.

Rute Eliminasi

Renally excreted unchanged (70%-90%) via glomerular filtration; Fecal (<1%)

Interaksi Obat

138 Data
Cocaine The therapeutic efficacy of Iobenguane can be decreased when used in combination with Cocaine.
Reserpine The therapeutic efficacy of Iobenguane can be decreased when used in combination with Reserpine.
Fluvoxamine Fluvoxamine may decrease effectiveness of Iobenguane as a diagnostic agent.
Citalopram Citalopram may decrease effectiveness of Iobenguane as a diagnostic agent.
Fluoxetine Fluoxetine may decrease effectiveness of Iobenguane as a diagnostic agent.
Duloxetine Duloxetine may decrease effectiveness of Iobenguane as a diagnostic agent.
Trazodone Trazodone may decrease effectiveness of Iobenguane as a diagnostic agent.
Paroxetine Paroxetine may decrease effectiveness of Iobenguane as a diagnostic agent.
Sertraline Sertraline may decrease effectiveness of Iobenguane as a diagnostic agent.
Sibutramine Sibutramine may decrease effectiveness of Iobenguane as a diagnostic agent.
Nefazodone Nefazodone may decrease effectiveness of Iobenguane as a diagnostic agent.
Escitalopram Escitalopram may decrease effectiveness of Iobenguane as a diagnostic agent.
Zimelidine Zimelidine may decrease effectiveness of Iobenguane as a diagnostic agent.
Dapoxetine Dapoxetine may decrease effectiveness of Iobenguane as a diagnostic agent.
Milnacipran Milnacipran may decrease effectiveness of Iobenguane as a diagnostic agent.
Desvenlafaxine Desvenlafaxine may decrease effectiveness of Iobenguane as a diagnostic agent.
Seproxetine Seproxetine may decrease effectiveness of Iobenguane as a diagnostic agent.
Levomilnacipran The therapeutic efficacy of Iobenguane can be decreased when used in combination with Levomilnacipran.
Indalpine Indalpine may decrease effectiveness of Iobenguane as a diagnostic agent.
Ritanserin Ritanserin may decrease effectiveness of Iobenguane as a diagnostic agent.
Alaproclate Alaproclate may decrease effectiveness of Iobenguane as a diagnostic agent.
Amphetamine Amphetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Phentermine Phentermine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Midodrine Midodrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Norepinephrine Norepinephrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Phenylephrine Phenylephrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Phenylpropanolamine Phenylpropanolamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Labetalol Labetalol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Metaraminol Metaraminol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Epinephrine Epinephrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Methoxamine Methoxamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Orciprenaline Orciprenaline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Phenmetrazine Phenmetrazine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dobutamine Dobutamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Pseudoephedrine Pseudoephedrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Benzphetamine Benzphetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ritodrine Ritodrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Terbutaline Terbutaline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Oxymetazoline Oxymetazoline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Diethylpropion Diethylpropion can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dopamine Dopamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Isoprenaline Isoprenaline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Acebutolol Acebutolol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lisdexamfetamine Lisdexamfetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Fenoterol Fenoterol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ephedrine Ephedrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mephentermine Mephentermine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Procaterol Procaterol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Clenbuterol Clenbuterol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
MMDA MMDA can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Midomafetamine Midomafetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tenamfetamine Tenamfetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Chlorphentermine Chlorphentermine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Methylenedioxyethamphetamine Methylenedioxyethamphetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dextroamphetamine Dextroamphetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Metamfetamine Metamfetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Celiprolol Celiprolol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nylidrin Nylidrin can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tetryzoline Tetryzoline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tyramine Tyramine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Isoxsuprine Isoxsuprine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Etilefrine Etilefrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Synephrine Synephrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Iofetamine I-123 Iofetamine I-123 can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Racepinephrine Racepinephrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ritobegron Ritobegron can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Bucindolol Bucindolol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tramazoline Tramazoline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mephedrone Mephedrone can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Fenozolone Fenozolone can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Methoxyphenamine Methoxyphenamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tretoquinol Tretoquinol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gepefrine Gepefrine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Epanolol Epanolol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Prenalterol Prenalterol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mefenorex Mefenorex can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
2,5-Dimethoxy-4-ethylthioamphetamine 2,5-Dimethoxy-4-ethylthioamphetamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Venlafaxine The therapeutic efficacy of Iobenguane can be decreased when used in combination with Venlafaxine.
Reboxetine Reboxetine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Amitriptyline Amitriptyline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Protriptyline Protriptyline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Imipramine Imipramine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nortriptyline Nortriptyline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Amoxapine Amoxapine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mazindol Mazindol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Trimipramine Trimipramine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Maprotiline Maprotiline can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Desipramine Desipramine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tapentadol Tapentadol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dosulepin Dosulepin can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Edivoxetine Edivoxetine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Viloxazine Viloxazine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nisoxetine Nisoxetine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lortalamine Lortalamine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Talopram Talopram can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Esreboxetine Esreboxetine can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Solriamfetol Solriamfetol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Doxepin Doxepin may decrease effectiveness of Iobenguane as a diagnostic agent.

Target Protein

Sodium-dependent noradrenaline transporter SLC6A2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 8082671
    Wafelman AR, Hoefnagel CA, Maes RA, Beijnen JH: Radioiodinated metaiodobenzylguanidine: a review of its biodistribution and pharmacokinetics, drug interactions, cytotoxicity and dosimetry. Eur J Nucl Med. 1994 Jun;21(6):545-59.

Contoh Produk & Brand

Produk: 3 • International brands: 0
Produk
  • AdreView
    Injection • 2 mCi/1mL • Intravenous • US • Approved
  • Azedra
    Injection, solution • 15 mCi/1mL • Intravenous • US • Approved
  • Iobenguane Sulfate I 131 Injection
    Injection • 2.3 mCi/2mL • Intravenous • US • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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