Peringatan Keamanan

The signs and symptoms that are produced after the acute overdosage of Mepyramine include Convulsions, Coma, Ataxia, Hyperpyrexia, Tremor, Extrapyramidal effects, Excitement.

Mepyramine

DB06691

small molecule approved vet_approved

Deskripsi

Mepyramine, or pyrilamine, targets the H1 receptor. It is a first generation antihistamine. However, it rapidly permeates the brain and so often causes drowsiness as a side effect. It has been found in over-the-counter combination products for colds and menstrual symptoms, but is considered to be an unapproved prescription medication used for cough, cold, or allergic conditions.

Struktur Molekul 2D

Berat 285.384
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food.

Interaksi Obat

1039 Data
Buprenorphine Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Magnesium sulfate The therapeutic efficacy of Mepyramine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Mepyramine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Mirtazapine Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Orphenadrine Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Pramipexole Mepyramine may increase the sedative activities of Pramipexole.
Ropinirole Mepyramine may increase the sedative activities of Ropinirole.
Rotigotine Mepyramine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Mepyramine.
Suvorexant Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Thalidomide Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Benzylpenicilloyl polylysine Mepyramine may decrease effectiveness of Benzylpenicilloyl polylysine as a diagnostic agent.
Betahistine The therapeutic efficacy of Betahistine can be decreased when used in combination with Mepyramine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Mepyramine.
Sodium oxybate Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Mepyramine.
Ethanol Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Mepyramine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Mepyramine.
Sibutramine The risk or severity of adverse effects can be increased when Mepyramine is combined with Sibutramine.
Zimelidine The risk or severity of adverse effects can be increased when Mepyramine is combined with Zimelidine.
Milnacipran The risk or severity of adverse effects can be increased when Mepyramine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Mepyramine is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Mepyramine is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Mepyramine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Mepyramine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Mepyramine is combined with Alaproclate.
Fluvoxamine The risk or severity of adverse effects can be increased when Mepyramine is combined with Fluvoxamine.
Citalopram The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Mepyramine is combined with Duloxetine.
Paroxetine The risk or severity of adverse effects can be increased when Mepyramine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Mepyramine is combined with Sertraline.
Nefazodone The risk or severity of adverse effects can be increased when Mepyramine is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Mepyramine is combined with Escitalopram.
Dapoxetine The risk or severity of adverse effects can be increased when Mepyramine is combined with Dapoxetine.
Amphetamine Amphetamine may decrease the sedative activities of Mepyramine.
Phentermine Phentermine may decrease the sedative activities of Mepyramine.
Benzphetamine Benzphetamine may decrease the sedative activities of Mepyramine.
Diethylpropion Diethylpropion may decrease the sedative activities of Mepyramine.
Lisdexamfetamine The serum concentration of dextroamphetamine, an active metabolite of Lisdexamfetamine, can be increased when used in combination with Mepyramine.
Mephentermine Mephentermine may decrease the sedative activities of Mepyramine.
MMDA MMDA may decrease the sedative activities of Mepyramine.
Midomafetamine Midomafetamine may decrease the sedative activities of Mepyramine.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the sedative activities of Mepyramine.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the sedative activities of Mepyramine.
Tenamfetamine Tenamfetamine may decrease the sedative activities of Mepyramine.
Chlorphentermine Chlorphentermine may decrease the sedative activities of Mepyramine.
Methylenedioxyethamphetamine Methylenedioxyethamphetamine may decrease the sedative activities of Mepyramine.
Dextroamphetamine Dextroamphetamine may decrease the sedative activities of Mepyramine.
Metamfetamine Metamfetamine may decrease the sedative activities of Mepyramine.
Iofetamine I-123 Iofetamine I-123 may decrease the sedative activities of Mepyramine.
Ritobegron Ritobegron may decrease the sedative activities of Mepyramine.
Mephedrone Mephedrone may decrease the sedative activities of Mepyramine.
Methoxyphenamine Methoxyphenamine may decrease the sedative activities of Mepyramine.
Gepefrine Gepefrine may decrease the sedative activities of Mepyramine.
2,5-Dimethoxy-4-ethylthioamphetamine 2,5-Dimethoxy-4-ethylthioamphetamine may decrease the sedative activities of Mepyramine.
Phendimetrazine Phendimetrazine may decrease the sedative activities of Mepyramine.
Buclizine The risk or severity of QTc prolongation can be increased when Buclizine is combined with Mepyramine.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Mepyramine.
Gallamine triethiodide The risk or severity of CNS depression can be increased when Gallamine triethiodide is combined with Mepyramine.
Triflupromazine The risk or severity of CNS depression can be increased when Triflupromazine is combined with Mepyramine.
Lamotrigine The risk or severity of CNS depression can be increased when Lamotrigine is combined with Mepyramine.
Nicardipine The risk or severity of QTc prolongation can be increased when Nicardipine is combined with Mepyramine.
Rocuronium The risk or severity of CNS depression can be increased when Rocuronium is combined with Mepyramine.
Scopolamine The risk or severity of CNS depression can be increased when Scopolamine is combined with Mepyramine.
Clidinium The risk or severity of CNS depression can be increased when Clidinium is combined with Mepyramine.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Mepyramine.
Brompheniramine The risk or severity of CNS depression can be increased when Brompheniramine is combined with Mepyramine.
Doxacurium The risk or severity of CNS depression can be increased when Doxacurium is combined with Mepyramine.
Mivacurium The risk or severity of CNS depression can be increased when Mivacurium is combined with Mepyramine.
Chlorprothixene The risk or severity of CNS depression can be increased when Chlorprothixene is combined with Mepyramine.
Metocurine The risk or severity of CNS depression can be increased when Metocurine is combined with Mepyramine.
Pancuronium The risk or severity of CNS depression can be increased when Pancuronium is combined with Mepyramine.
Pipecuronium The risk or severity of CNS depression can be increased when Pipecuronium is combined with Mepyramine.
Rapacuronium The risk or severity of CNS depression can be increased when Rapacuronium is combined with Mepyramine.
Pizotifen The risk or severity of CNS depression can be increased when Pizotifen is combined with Mepyramine.
Benactyzine The risk or severity of CNS depression can be increased when Mepyramine is combined with Benactyzine.
Trimebutine The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Trimebutine.
Emepronium The risk or severity of CNS depression can be increased when Mepyramine is combined with Emepronium.
Doxepin The risk or severity of CNS depression can be increased when Doxepin is combined with Mepyramine.
Zopiclone The risk or severity of adverse effects can be increased when Mepyramine is combined with Zopiclone.
Leuprolide The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Leuprolide.
Goserelin The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Goserelin.
Erythromycin The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Erythromycin.
Azithromycin The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Azithromycin.
Moxifloxacin The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Moxifloxacin.
Sulfisoxazole The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Sulfisoxazole.
Sulpiride The risk or severity of CNS depression can be increased when Sulpiride is combined with Mepyramine.
Nimodipine The risk or severity of QTc prolongation can be increased when Mepyramine is combined with Nimodipine.
Oxaliplatin The risk or severity of QTc prolongation can be increased when Oxaliplatin is combined with Mepyramine.

Target Protein

Histamine H1 receptor HRH1

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 226 • International brands: 0
Produk
  • A-Tan 12X Suspension
    Suspension • - • Oral • US
  • Acetaminophen 500mg Caffeine 60mg Pyrilamine maleate 15mg
    Tablet • - • Oral • US • OTC
  • Acetaminophen 500mg Caffeine 60mg Pyrilamine maleate 15mg
    Tablet • - • Oral • US • OTC
  • Acetaminophen 500mg Caffeine 60mg Pyrilamine maleate 15mg
    Tablet • - • Oral • US • OTC
  • Acetaminophen 500mg Caffeine 60mg Pyrilamine maleate 15mg
    Tablet • - • Oral • US • OTC
  • Acetaminophen,Caffeine and Pyrilamine Maleate
    Tablet • - • Oral • US • OTC
  • Aldex D
    Suspension • - • Oral • US • OTC
  • Antitussive Decong Antihistamine Syr
    Syrup • - • Oral • Canada • OTC • Approved
Menampilkan 8 dari 226 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul