Deramciclane

DB06512

small molecule investigational

Deskripsi

Deramciclane (EGIS-3886) is used for the treatment of a number of anxiety disorders. Deramciclane differs from other anti anxiety medications in that it is not a benzodiazepine and so has a different structure and target. It antagonizes 5-HT2A receptors, agonizes 5-HT2C receptors, and functions as a GABA reuptake inhibitor.

Struktur Molekul 2D

Berat 301.474
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

961 Data
Buprenorphine Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Hydrocodone Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Magnesium sulfate The therapeutic efficacy of Deramciclane can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Deramciclane may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Mirtazapine Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Orphenadrine Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Pramipexole Deramciclane may increase the sedative activities of Pramipexole.
Ropinirole Deramciclane may increase the sedative activities of Ropinirole.
Rotigotine Deramciclane may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Deramciclane.
Sodium oxybate Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Thalidomide Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Yohimbine The therapeutic efficacy of Deramciclane can be increased when used in combination with Yohimbine.
Mefloquine The therapeutic efficacy of Deramciclane can be decreased when used in combination with Mefloquine.
Mianserin The therapeutic efficacy of Deramciclane can be decreased when used in combination with Mianserin.
Orlistat Orlistat can cause a decrease in the absorption of Deramciclane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Topotecan Deramciclane may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Deramciclane.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Deramciclane.
Dicoumarol The risk or severity of adverse effects can be increased when Deramciclane is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Deramciclane is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when Deramciclane is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Deramciclane is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Deramciclane is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Deramciclane is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when Deramciclane is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Deramciclane is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Deramciclane is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Deramciclane is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Deramciclane is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Deramciclane is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when Deramciclane is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when Deramciclane is combined with (S)-Warfarin.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Deramciclane.
Ethanol Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Deramciclane may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Zimelidine The risk or severity of adverse effects can be increased when Deramciclane is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Deramciclane is combined with Dapoxetine.
Seproxetine The risk or severity of adverse effects can be increased when Deramciclane is combined with Seproxetine.
Fluvoxamine The risk or severity of adverse effects can be increased when Deramciclane is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Deramciclane is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Deramciclane is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Deramciclane is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Deramciclane is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Deramciclane is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Deramciclane is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Deramciclane is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Deramciclane is combined with Escitalopram.
Milnacipran The risk or severity of adverse effects can be increased when Deramciclane is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Deramciclane is combined with Desvenlafaxine.
Levomilnacipran The risk or severity of adverse effects can be increased when Deramciclane is combined with Levomilnacipran.
Indalpine The risk or severity of adverse effects can be increased when Deramciclane is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Deramciclane is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Deramciclane is combined with Alaproclate.
Benzatropine The metabolism of Benzatropine can be decreased when combined with Deramciclane.
Terfenadine The metabolism of Terfenadine can be decreased when combined with Deramciclane.
Darifenacin The metabolism of Darifenacin can be decreased when combined with Deramciclane.
Cocaine The risk or severity of methemoglobinemia can be increased when Deramciclane is combined with Cocaine.
Quinidine The therapeutic efficacy of Deramciclane can be decreased when used in combination with Quinidine.
Tolterodine The metabolism of Tolterodine can be decreased when combined with Deramciclane.
Tiotropium The metabolism of Tiotropium can be decreased when combined with Deramciclane.
Solifenacin The metabolism of Solifenacin can be decreased when combined with Deramciclane.
Fesoterodine The metabolism of Fesoterodine can be decreased when combined with Deramciclane.
Umeclidinium The metabolism of Umeclidinium can be decreased when combined with Deramciclane.
Revefenacin The metabolism of Revefenacin can be decreased when combined with Deramciclane.
Doxepin The risk or severity of CNS depression can be increased when Doxepin is combined with Deramciclane.
Zopiclone The risk or severity of adverse effects can be increased when Deramciclane is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Deramciclane.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Deramciclane.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Deramciclane.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Deramciclane.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Deramciclane.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Deramciclane.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with Deramciclane.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with Deramciclane.
Butalbital The risk or severity of CNS depression can be increased when Butalbital is combined with Deramciclane.
Methysergide The risk or severity of CNS depression can be increased when Methysergide is combined with Deramciclane.
Cabergoline The risk or severity of CNS depression can be increased when Cabergoline is combined with Deramciclane.
Phenytoin The risk or severity of CNS depression can be increased when Phenytoin is combined with Deramciclane.
Topiramate The risk or severity of CNS depression can be increased when Topiramate is combined with Deramciclane.
Clemastine The risk or severity of CNS depression can be increased when Clemastine is combined with Deramciclane.
Etomidate The risk or severity of CNS depression can be increased when Etomidate is combined with Deramciclane.
Morphine The risk or severity of CNS depression can be increased when Morphine is combined with Deramciclane.
Talbutal The risk or severity of CNS depression can be increased when Talbutal is combined with Deramciclane.
Pentobarbital The risk or severity of CNS depression can be increased when Pentobarbital is combined with Deramciclane.
Zolmitriptan The risk or severity of CNS depression can be increased when Zolmitriptan is combined with Deramciclane.
Codeine The risk or severity of CNS depression can be increased when Codeine is combined with Deramciclane.

Target Protein

5-hydroxytryptamine receptor 2A HTR2A
5-hydroxytryptamine receptor 2C HTR2C

Referensi & Sumber

Artikel (PubMed)
  • PMID: 2502985
    Kovacs I, Maksay G, Simonyi M: Inhibition of high-affinity synaptosomal uptake of gamma-aminobutyric acid by a bicyclo-heptane derivative. Arzneimittelforschung. 1989 Mar;39(3):295-7.

Contoh Produk & Brand

Produk: 0 • International brands: 0
Belum ada data produk/brand untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field produk/brand.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul