Muraglitazar (Bristol-Myers Squibb/Merck) is a new agent under investigation for the treatment of patients with type 2 diabetes. It belongs to a novel class of drugs that target the peroxisome proliferator-activated receptors, both alpha and gamma subtypes. In addition to improvements in blood glucose and hemoglobin A1c (HbA1c), muraglitazar treatment is associated with a substantial reduction in triglycerides (TGs), an increase in HDL-C, and a modest decrease in LDL-C levels.
Fitur visualisasi ini dikembangkan menggunakan pendekatan Graph Theory untuk memetakan hubungan polifarmasi dan molekuler. Entitas (Obat, Target, Gen) direpresentasikan sebagai Simpul (Nodes), sedangkan hubungan biologisnya sebagai Sisi (Edges).
drugbank-id dan name pada skema XML DrugBank.targets/target yang memuat polipeptida sasaran.gene-name dan varian snp-effects.Tata letak grafik menggunakan algoritma Force-Directed Graph (Barnes-Hut). Model fisika ini menerapkan gaya tolak-menolak antar simpul (Gravitasi: -3000) agar tidak tumpang tindih, serta gaya pegas (Spring: 0.04) pada garis penghubung untuk fleksibilitas interaksi.
| Mifepristone | The serum concentration of Muraglitazar can be increased when it is combined with Mifepristone. |
| Nelfinavir | The metabolism of Muraglitazar can be increased when combined with Nelfinavir. |
| Desogestrel | The metabolism of Muraglitazar can be increased when combined with Desogestrel. |
| Zidovudine | The metabolism of Muraglitazar can be increased when combined with Zidovudine. |
| Lamotrigine | The metabolism of Muraglitazar can be increased when combined with Lamotrigine. |
| Carbamazepine | The metabolism of Muraglitazar can be increased when combined with Carbamazepine. |
| Efavirenz | The metabolism of Muraglitazar can be increased when combined with Efavirenz. |
| Tipranavir | The metabolism of Muraglitazar can be increased when combined with Tipranavir. |
| Ethinylestradiol | The metabolism of Muraglitazar can be increased when combined with Ethinylestradiol. |
| Testosterone propionate | The metabolism of Muraglitazar can be increased when combined with Testosterone propionate. |
| Primidone | The metabolism of Muraglitazar can be increased when combined with Primidone. |
| Secobarbital | The metabolism of Muraglitazar can be increased when combined with Secobarbital. |
| Rifampin | The metabolism of Muraglitazar can be increased when combined with Rifampicin. |
| Phenobarbital | The metabolism of Muraglitazar can be increased when combined with Phenobarbital. |
| Bexarotene | The metabolism of Muraglitazar can be decreased when combined with Bexarotene. |
| Diltiazem | The metabolism of Muraglitazar can be decreased when combined with Diltiazem. |
| Levothyroxine | The metabolism of Muraglitazar can be decreased when combined with Levothyroxine. |
| Loratadine | The metabolism of Muraglitazar can be decreased when combined with Loratadine. |
| Quinine | The metabolism of Muraglitazar can be decreased when combined with Quinine. |
| Medroxyprogesterone acetate | The metabolism of Muraglitazar can be decreased when combined with Medroxyprogesterone acetate. |
| Nicardipine | The metabolism of Muraglitazar can be decreased when combined with Nicardipine. |
| Tamoxifen | The metabolism of Muraglitazar can be decreased when combined with Tamoxifen. |
| Irbesartan | The metabolism of Muraglitazar can be decreased when combined with Irbesartan. |
| Oxybutynin | The metabolism of Muraglitazar can be decreased when combined with Oxybutynin. |
| Fluvastatin | The metabolism of Muraglitazar can be decreased when combined with Fluvastatin. |
| Pioglitazone | The metabolism of Muraglitazar can be decreased when combined with Pioglitazone. |
| Saquinavir | The metabolism of Muraglitazar can be decreased when combined with Saquinavir. |
| Genistein | The metabolism of Muraglitazar can be decreased when combined with Genistein. |
| Topiroxostat | The metabolism of Muraglitazar can be decreased when combined with Topiroxostat. |
| Abiraterone | The metabolism of Muraglitazar can be decreased when combined with Abiraterone. |
| Teriflunomide | The metabolism of Muraglitazar can be decreased when combined with Teriflunomide. |
| Enzalutamide | The metabolism of Muraglitazar can be decreased when combined with Enzalutamide. |
| Trimethoprim | The metabolism of Muraglitazar can be decreased when combined with Trimethoprim. |
| Ritonavir | The metabolism of Muraglitazar can be decreased when combined with Ritonavir. |
| Fluticasone propionate | The metabolism of Muraglitazar can be decreased when combined with Fluticasone propionate. |
| Clopidogrel | The metabolism of Muraglitazar can be decreased when combined with Clopidogrel. |
| Candesartan cilexetil | The metabolism of Muraglitazar can be decreased when combined with Candesartan cilexetil. |
| Salmeterol | The metabolism of Muraglitazar can be decreased when combined with Salmeterol. |
| Felodipine | The metabolism of Muraglitazar can be decreased when combined with Felodipine. |
| Gemfibrozil | The metabolism of Muraglitazar can be decreased when combined with Gemfibrozil. |
| Fluticasone | The metabolism of Muraglitazar can be decreased when combined with Fluticasone. |
| Mometasone furoate | The metabolism of Muraglitazar can be decreased when combined with Mometasone furoate. |
| Adenine | The metabolism of Muraglitazar can be decreased when combined with Adenine. |
| Indinavir | The metabolism of Muraglitazar can be decreased when combined with Indinavir. |
| Valproic acid | The metabolism of Muraglitazar can be decreased when combined with Valproic acid. |
| Amitriptyline | The metabolism of Muraglitazar can be decreased when combined with Amitriptyline. |
| Indomethacin | The metabolism of Muraglitazar can be decreased when combined with Indomethacin. |
| Flurbiprofen | The metabolism of Muraglitazar can be decreased when combined with Flurbiprofen. |
| Propofol | The metabolism of Muraglitazar can be decreased when combined with Propofol. |
| Ketoconazole | The metabolism of Muraglitazar can be decreased when combined with Ketoconazole. |
| Probenecid | The metabolism of Muraglitazar can be decreased when combined with Probenecid. |
| Atazanavir | The metabolism of Muraglitazar can be decreased when combined with Atazanavir. |
| Flunitrazepam | The metabolism of Muraglitazar can be decreased when combined with Flunitrazepam. |
| Deferasirox | The metabolism of Muraglitazar can be decreased when combined with Deferasirox. |
| Nilotinib | The metabolism of Muraglitazar can be decreased when combined with Nilotinib. |
| Eltrombopag | The metabolism of Muraglitazar can be decreased when combined with Eltrombopag. |
| Regorafenib | The metabolism of Muraglitazar can be decreased when combined with Regorafenib. |
| Dasabuvir | The metabolism of Muraglitazar can be decreased when combined with Dasabuvir. |
| Sodium aurothiomalate | The metabolism of Muraglitazar can be decreased when combined with Sodium aurothiomalate. |
| Ombitasvir | The metabolism of Muraglitazar can be decreased when combined with Ombitasvir. |
| Paritaprevir | The metabolism of Muraglitazar can be decreased when combined with Paritaprevir. |
| Silibinin | The metabolism of Muraglitazar can be decreased when combined with Silibinin. |
| Dacomitinib | The metabolism of Muraglitazar can be decreased when combined with Dacomitinib. |
| Fostamatinib | The metabolism of Muraglitazar can be decreased when combined with Fostamatinib. |
| Pibrentasvir | The metabolism of Muraglitazar can be decreased when combined with Pibrentasvir. |
| Glecaprevir | The metabolism of Muraglitazar can be decreased when combined with Glecaprevir. |
| Pexidartinib | The metabolism of Muraglitazar can be decreased when combined with Pexidartinib. |
| Pyrimethamine | The metabolism of Muraglitazar can be decreased when combined with Pyrimethamine. |
| Ticlopidine | The metabolism of Muraglitazar can be decreased when combined with Ticlopidine. |
| Cimetidine | The metabolism of Muraglitazar can be decreased when combined with Cimetidine. |
| Rofecoxib | The metabolism of Muraglitazar can be decreased when combined with Rofecoxib. |
| Quinidine | The metabolism of Muraglitazar can be decreased when combined with Quinidine. |
| Ketoprofen | The metabolism of Muraglitazar can be decreased when combined with Ketoprofen. |
| Fenofibrate | The metabolism of Muraglitazar can be decreased when combined with Fenofibrate. |
| Tegaserod | The metabolism of Muraglitazar can be decreased when combined with Tegaserod. |
| Cabozantinib | The metabolism of Muraglitazar can be decreased when combined with Cabozantinib. |
| Diethylstilbestrol | The metabolism of Muraglitazar can be decreased when combined with Diethylstilbestrol. |
| Terfenadine | The metabolism of Muraglitazar can be decreased when combined with Terfenadine. |
| Cerivastatin | The metabolism of Muraglitazar can be decreased when combined with Cerivastatin. |
| Raloxifene | The metabolism of Muraglitazar can be decreased when combined with Raloxifene. |
| Simvastatin | The metabolism of Muraglitazar can be decreased when combined with Simvastatin. |
| Nilutamide | The metabolism of Muraglitazar can be decreased when combined with Nilutamide. |
| Metronidazole | The metabolism of Muraglitazar can be decreased when combined with Metronidazole. |
| Bezafibrate | The metabolism of Muraglitazar can be decreased when combined with Bezafibrate. |
| Quercetin | The metabolism of Muraglitazar can be decreased when combined with Quercetin. |
| Licofelone | The metabolism of Muraglitazar can be decreased when combined with Licofelone. |
| Nilvadipine | The metabolism of Muraglitazar can be decreased when combined with Nilvadipine. |
| Sulfaphenazole | The metabolism of Muraglitazar can be decreased when combined with Sulfaphenazole. |
| Vemurafenib | The metabolism of Muraglitazar can be decreased when combined with Vemurafenib. |
| Lumacaftor | The metabolism of Muraglitazar can be decreased when combined with Lumacaftor. |
| Isavuconazole | The metabolism of Muraglitazar can be decreased when combined with Isavuconazole. |
| Alpelisib | The metabolism of Muraglitazar can be decreased when combined with Alpelisib. |
| Letermovir | The metabolism of Muraglitazar can be decreased when combined with Letermovir. |
| Triclabendazole | The metabolism of Muraglitazar can be decreased when combined with Triclabendazole. |
| Candesartan | The metabolism of Muraglitazar can be decreased when combined with Candesartan. |
| Favipiravir | The metabolism of Muraglitazar can be decreased when combined with Favipiravir. |
| Methylene blue | The metabolism of Muraglitazar can be decreased when combined with Methylene blue. |
| Mometasone | The metabolism of Muraglitazar can be decreased when combined with Mometasone. |
| Pralsetinib | The metabolism of Muraglitazar can be decreased when combined with Pralsetinib. |
| Miconazole | The metabolism of Muraglitazar can be decreased when combined with Miconazole. |