Human C1-esterase inhibitor

DB06404

biotech approved

Deskripsi

C1 Esterase Inhibitor (Human) is composed of purified endogenous complement component-1 esterase inhibitor (hC1INH) isolated from human plasma. The primary function of endogenous C1INH is to regulate the activation of the complement and contact system pathways.L16586, L16606

This drug is indicated for prophylaxis and treatment of Hereditary Angioedema (HAE), a human genetic disorder caused by a shortage of C1 inhibitor activity that results in an overreaction of the immune system. The disease is characterized by acute attacks of painful, and in some cases, fatal swelling of several soft tissues or edema, which may last up to five days when untreated.L16586, L16606

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Following intravenous administration of a single dose, the half-life was 56 ± 36 hours.[L16586] Subcutaneous administration produces a half-life of 199.6 hours.[A19661]
Volume Distribusi -
Klirens (Clearance) Following intravenous administration of a single dose, the clearance rate was 0.85 ± 1.07 mL/min.[L16586]

Absorpsi

Following intravenous administration of a single dose, the Cmax was 0.68 ± 0.08 U/mL and Tmax was 3.9 ± 7.3 hours.L16586

Metabolisme

Protein drugs are expected to be degraded by proteases and other catalytic enzymes to smaller peptides and amino acids.A182009

Rute Eliminasi

After nonspecific proteolysis, the amino acids from protein drugs are reused for protein synthesis or further broken down and eliminated by the kidneys.A182009

Interaksi Obat

37 Data
Etonogestrel The risk or severity of thromboembolism can be increased when Etonogestrel is combined with Human C1-esterase inhibitor.
Desogestrel The risk or severity of thromboembolism can be increased when Desogestrel is combined with Human C1-esterase inhibitor.
Megestrol acetate The risk or severity of thromboembolism can be increased when Megestrol acetate is combined with Human C1-esterase inhibitor.
Levonorgestrel The risk or severity of thromboembolism can be increased when Levonorgestrel is combined with Human C1-esterase inhibitor.
Dydrogesterone The risk or severity of thromboembolism can be increased when Dydrogesterone is combined with Human C1-esterase inhibitor.
Progesterone The risk or severity of thromboembolism can be increased when Progesterone is combined with Human C1-esterase inhibitor.
Medroxyprogesterone acetate The risk or severity of thromboembolism can be increased when Medroxyprogesterone acetate is combined with Human C1-esterase inhibitor.
Norethisterone The risk or severity of thromboembolism can be increased when Norethisterone is combined with Human C1-esterase inhibitor.
Ethynodiol diacetate The risk or severity of thromboembolism can be increased when Ethynodiol diacetate is combined with Human C1-esterase inhibitor.
Norgestimate The risk or severity of thromboembolism can be increased when Norgestimate is combined with Human C1-esterase inhibitor.
Drospirenone The risk or severity of thromboembolism can be increased when Drospirenone is combined with Human C1-esterase inhibitor.
Allylestrenol The risk or severity of thromboembolism can be increased when Allylestrenol is combined with Human C1-esterase inhibitor.
Cyproterone acetate The risk or severity of thromboembolism can be increased when Cyproterone acetate is combined with Human C1-esterase inhibitor.
Norelgestromin The risk or severity of thromboembolism can be increased when Norelgestromin is combined with Human C1-esterase inhibitor.
Gestodene The risk or severity of thromboembolism can be increased when Gestodene is combined with Human C1-esterase inhibitor.
Hydroxyprogesterone caproate The risk or severity of thromboembolism can be increased when Hydroxyprogesterone caproate is combined with Human C1-esterase inhibitor.
Dienogest The risk or severity of thromboembolism can be increased when Dienogest is combined with Human C1-esterase inhibitor.
Medrogestone The risk or severity of thromboembolism can be increased when Medrogestone is combined with Human C1-esterase inhibitor.
Norethynodrel The risk or severity of thromboembolism can be increased when Norethynodrel is combined with Human C1-esterase inhibitor.
Norgestrel The risk or severity of thromboembolism can be increased when Norgestrel is combined with Human C1-esterase inhibitor.
Altrenogest The risk or severity of thromboembolism can be increased when Altrenogest is combined with Human C1-esterase inhibitor.
Gestrinone The risk or severity of thromboembolism can be increased when Gestrinone is combined with Human C1-esterase inhibitor.
Nomegestrol The risk or severity of thromboembolism can be increased when Nomegestrol is combined with Human C1-esterase inhibitor.
Lynestrenol The risk or severity of thromboembolism can be increased when Lynestrenol is combined with Human C1-esterase inhibitor.
Gestonorone The risk or severity of thromboembolism can be increased when Gestonorone is combined with Human C1-esterase inhibitor.
Chlormadinone The risk or severity of thromboembolism can be increased when Chlormadinone is combined with Human C1-esterase inhibitor.
Methylestrenolone The risk or severity of thromboembolism can be increased when Methylestrenolone is combined with Human C1-esterase inhibitor.
Norgestrienone The risk or severity of thromboembolism can be increased when Norgestrienone is combined with Human C1-esterase inhibitor.
Promegestone The risk or severity of thromboembolism can be increased when Promegestone is combined with Human C1-esterase inhibitor.
Quingestanol The risk or severity of thromboembolism can be increased when Quingestanol is combined with Human C1-esterase inhibitor.
Demegestone The risk or severity of thromboembolism can be increased when Demegestone is combined with Human C1-esterase inhibitor.
Etynodiol The risk or severity of thromboembolism can be increased when Etynodiol is combined with Human C1-esterase inhibitor.
Nomegestrol acetate The risk or severity of thromboembolism can be increased when Nomegestrol acetate is combined with Human C1-esterase inhibitor.
Hydroxyprogesterone The risk or severity of thromboembolism can be increased when Hydroxyprogesterone is combined with Human C1-esterase inhibitor.
Norethindrone enanthate The risk or severity of thromboembolism can be increased when Norethindrone enanthate is combined with Human C1-esterase inhibitor.
Quingestanol acetate The risk or severity of thromboembolism can be increased when Quingestanol acetate is combined with Human C1-esterase inhibitor.
Algestone acetophenide The risk or severity of thromboembolism can be increased when Algestone acetophenide is combined with Human C1-esterase inhibitor.

Target Protein

Complement C1r subcomponent C1R
Complement C1s subcomponent C1S
Plasma kallikrein KLKB1
Coagulation factor XII F12
Coagulation factor XI F11
Tissue-type plasminogen activator PLAT
Prothrombin F2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 21698655
    Katsila T, Siskos AP, Tamvakopoulos C: Peptide and protein drugs: the study of their metabolism and catabolism by mass spectrometry. Mass Spectrom Rev. 2012 Jan-Feb;31(1):110-33. doi: 10.1002/mas.20340. Epub 2011 Jun 22.
  • PMID: 24266596
    Martinez-Saguer I, Cicardi M, Suffritti C, Rusicke E, Aygoren-Pursun E, Stoll H, Rossmanith T, Feussner A, Kalina U, Kreuz W: Pharmacokinetics of plasma-derived C1-esterase inhibitor after subcutaneous versus intravenous administration in subjects with mild or moderate hereditary angioedema: the PASSION study. Transfusion. 2014 Jun;54(6):1552-61. doi: 10.1111/trf.12501. Epub 2013 Nov 24.

Contoh Produk & Brand

Produk: 11 • International brands: 0
Produk
  • Berinert
    Injection, powder, lyophilized, for solution; Kit • 500 [iU]/10mL • Intravenous • US • Approved
  • Berinert 1500
    Kit; Powder, for solution • 1500 unit / vial • Intravenous • Canada • Approved
  • Berinert 500
    Kit; Powder, for solution • 500 unit / vial • Intravenous • Canada • Approved
  • Cinryze
    Injection, powder, lyophilized, for solution; Kit • 500 [iU]/5mL • Intravenous • US • Approved
  • Cinryze
    Powder, for solution • 500 unit / vial • Intravenous • Canada • Approved
  • Cinryze
    Injection, powder, for solution • 500 U • Intravenous • EU • Approved
  • Cinryze
    Injection, powder, lyophilized, for solution • 500 [iU]/5mL • Intravenous • US • Approved
  • Haegarda
    Kit; Powder, for solution • 2000 unit / vial • Subcutaneous • Canada • Approved
Menampilkan 8 dari 11 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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