Tolperisone

DB06264

small molecule investigational

Deskripsi

Tolperisone is an oral, centrally acting muscle relaxant. Its precise mechanism is not completely understood, though it blocks sodium and calcium channels. It possesses a high affinity for nervous system tissue, reaching highest concentrations in brain stem, spinal cord and peripheral nerves. Based on existing clinical data, Tolperisone is not sedating and does not interact with alcohol.

Struktur Molekul 2D

Berat 245.366
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

668 Data
Buprenorphine Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Hydrocodone Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Magnesium sulfate The therapeutic efficacy of Tolperisone can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Tolperisone may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Mirtazapine Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Orphenadrine Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Pramipexole Tolperisone may increase the sedative activities of Pramipexole.
Ropinirole Tolperisone may increase the sedative activities of Ropinirole.
Rotigotine Tolperisone may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Tolperisone.
Sodium oxybate Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Thalidomide Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Tolperisone.
Ethanol Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Tolperisone may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Fluvoxamine The risk or severity of adverse effects can be increased when Tolperisone is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Tolperisone is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Tolperisone is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Tolperisone is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Tolperisone is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Tolperisone is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Tolperisone is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Tolperisone is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Tolperisone is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Tolperisone is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Tolperisone is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Tolperisone is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Tolperisone is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Tolperisone is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Tolperisone is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Tolperisone is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Tolperisone is combined with Alaproclate.
Amitriptyline The risk or severity of CNS depression can be increased when Amitriptyline is combined with Tolperisone.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Tolperisone.
Imipramine The risk or severity of CNS depression can be increased when Imipramine is combined with Tolperisone.
Nortriptyline The risk or severity of CNS depression can be increased when Nortriptyline is combined with Tolperisone.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Tolperisone.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Tolperisone.
Maprotiline The risk or severity of CNS depression can be increased when Maprotiline is combined with Tolperisone.
Doxepin The risk or severity of CNS depression can be increased when Doxepin is combined with Tolperisone.
Desipramine The risk or severity of CNS depression can be increased when Desipramine is combined with Tolperisone.
Pizotifen The risk or severity of CNS depression can be increased when Pizotifen is combined with Tolperisone.
Dosulepin The risk or severity of CNS depression can be increased when Tolperisone is combined with Dosulepin.
Zopiclone The risk or severity of adverse effects can be increased when Tolperisone is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Tolperisone.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Tolperisone.
Tryptophan The risk or severity of CNS depression can be increased when Tryptophan is combined with Tolperisone.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Tolperisone.
Lorazepam The risk or severity of CNS depression can be increased when Lorazepam is combined with Tolperisone.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Tolperisone.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Tolperisone.
Reserpine The risk or severity of CNS depression can be increased when Reserpine is combined with Tolperisone.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Tolperisone.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with Tolperisone.
Temazepam The risk or severity of CNS depression can be increased when Temazepam is combined with Tolperisone.
Reboxetine The risk or severity of CNS depression can be increased when Reboxetine is combined with Tolperisone.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with Tolperisone.
Butalbital The risk or severity of CNS depression can be increased when Butalbital is combined with Tolperisone.
Methysergide The risk or severity of CNS depression can be increased when Methysergide is combined with Tolperisone.
Cabergoline The risk or severity of CNS depression can be increased when Cabergoline is combined with Tolperisone.
Phenytoin The risk or severity of CNS depression can be increased when Phenytoin is combined with Tolperisone.
Topiramate The risk or severity of CNS depression can be increased when Topiramate is combined with Tolperisone.
Clemastine The risk or severity of CNS depression can be increased when Clemastine is combined with Tolperisone.
Venlafaxine The risk or severity of CNS depression can be increased when Venlafaxine is combined with Tolperisone.
Etomidate The risk or severity of CNS depression can be increased when Etomidate is combined with Tolperisone.
Morphine The risk or severity of CNS depression can be increased when Morphine is combined with Tolperisone.
Talbutal The risk or severity of CNS depression can be increased when Talbutal is combined with Tolperisone.
Pentobarbital The risk or severity of CNS depression can be increased when Pentobarbital is combined with Tolperisone.
Valproic acid The risk or severity of CNS depression can be increased when Valproic acid is combined with Tolperisone.
Zolmitriptan The risk or severity of CNS depression can be increased when Zolmitriptan is combined with Tolperisone.
Codeine The risk or severity of CNS depression can be increased when Codeine is combined with Tolperisone.
Dihydroergotamine The risk or severity of CNS depression can be increased when Dihydroergotamine is combined with Tolperisone.
Tolcapone The risk or severity of CNS depression can be increased when Tolcapone is combined with Tolperisone.
Hydromorphone The risk or severity of CNS depression can be increased when Hydromorphone is combined with Tolperisone.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with Tolperisone.
Cetirizine The risk or severity of CNS depression can be increased when Cetirizine is combined with Tolperisone.
Protriptyline The risk or severity of CNS depression can be increased when Protriptyline is combined with Tolperisone.
Trimethadione The risk or severity of CNS depression can be increased when Trimethadione is combined with Tolperisone.
Clobazam The risk or severity of sedation, somnolence, and CNS depression can be increased when Clobazam is combined with Tolperisone.
Chlorzoxazone The risk or severity of CNS depression can be increased when Chlorzoxazone is combined with Tolperisone.
Clozapine The risk or severity of CNS depression can be increased when Clozapine is combined with Tolperisone.
Meprobamate The risk or severity of CNS depression can be increased when Meprobamate is combined with Tolperisone.
Thiethylperazine The risk or severity of CNS depression can be increased when Thiethylperazine is combined with Tolperisone.
Palonosetron The risk or severity of CNS depression can be increased when Palonosetron is combined with Tolperisone.
Sulpiride The risk or severity of CNS depression can be increased when Sulpiride is combined with Tolperisone.
Alprazolam The risk or severity of CNS depression can be increased when Alprazolam is combined with Tolperisone.
Dexbrompheniramine The risk or severity of CNS depression can be increased when Dexbrompheniramine is combined with Tolperisone.

Target Protein

Sodium channel protein type 11 subunit alpha SCN11A

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 0 • International brands: 2
International Brands
  • Musclex
  • Viveo

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