YKP-1358

DB06109

small molecule investigational

Deskripsi

YKP1358 is a novel serotonin (5-HT2A) and dopamine (D2) antagonist that has demonstrated potent activity in animals that relates to both positive and negative symptoms of schizophrenia. In addition, the YKP1358 pharmacological profile suggests a very low potential for extrapyramidal side effects.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

714 Data
Buprenorphine YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Hydrocodone YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Magnesium sulfate The therapeutic efficacy of YKP-1358 can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine YKP-1358 may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Orphenadrine YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Rotigotine YKP-1358 may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with YKP-1358.
Sodium oxybate YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Thalidomide YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with YKP-1358.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with YKP-1358.
Dicoumarol The risk or severity of adverse effects can be increased when YKP-1358 is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when YKP-1358 is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when YKP-1358 is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when YKP-1358 is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when YKP-1358 is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when YKP-1358 is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when YKP-1358 is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when YKP-1358 is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when YKP-1358 is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when YKP-1358 is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when YKP-1358 is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when YKP-1358 is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when YKP-1358 is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when YKP-1358 is combined with (S)-Warfarin.
Mirtazapine YKP-1358 may increase the serotonergic activities of Mirtazapine.
Ethanol YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine YKP-1358 may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Fluvoxamine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when YKP-1358 is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Duloxetine.
Paroxetine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when YKP-1358 is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when YKP-1358 is combined with Nefazodone.
Zimelidine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when YKP-1358 is combined with Milnacipran.
Desvenlafaxine The risk or severity of serotonin syndrome can be increased when Desvenlafaxine is combined with YKP-1358.
Seproxetine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Seproxetine.
Levomilnacipran The risk or severity of serotonin syndrome can be increased when YKP-1358 is combined with Levomilnacipran.
Indalpine The risk or severity of adverse effects can be increased when YKP-1358 is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when YKP-1358 is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when YKP-1358 is combined with Alaproclate.
Methylene blue YKP-1358 may increase the serotonergic activities of Methylene blue.
Zopiclone The risk or severity of adverse effects can be increased when YKP-1358 is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with YKP-1358.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with YKP-1358.
Tryptophan The risk or severity of CNS depression can be increased when Tryptophan is combined with YKP-1358.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of YKP-1358.
Lorazepam The risk or severity of CNS depression can be increased when Lorazepam is combined with YKP-1358.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with YKP-1358.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with YKP-1358.
Reserpine The risk or severity of CNS depression can be increased when Reserpine is combined with YKP-1358.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with YKP-1358.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with YKP-1358.
Temazepam The risk or severity of CNS depression can be increased when Temazepam is combined with YKP-1358.
Reboxetine The risk or severity of CNS depression can be increased when Reboxetine is combined with YKP-1358.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with YKP-1358.
Butalbital The risk or severity of CNS depression can be increased when Butalbital is combined with YKP-1358.
Methysergide The risk or severity of CNS depression can be increased when Methysergide is combined with YKP-1358.
Cabergoline The risk or severity of CNS depression can be increased when Cabergoline is combined with YKP-1358.
Phenytoin The risk or severity of CNS depression can be increased when Phenytoin is combined with YKP-1358.
Topiramate The risk or severity of CNS depression can be increased when Topiramate is combined with YKP-1358.
Clemastine The risk or severity of CNS depression can be increased when Clemastine is combined with YKP-1358.
Venlafaxine The risk or severity of serotonin syndrome can be increased when YKP-1358 is combined with Venlafaxine.
Etomidate The risk or severity of CNS depression can be increased when Etomidate is combined with YKP-1358.
Morphine The risk or severity of CNS depression can be increased when Morphine is combined with YKP-1358.
Talbutal The risk or severity of CNS depression can be increased when Talbutal is combined with YKP-1358.
Pentobarbital The risk or severity of CNS depression can be increased when Pentobarbital is combined with YKP-1358.
Valproic acid The risk or severity of CNS depression can be increased when Valproic acid is combined with YKP-1358.
Zolmitriptan The risk or severity of CNS depression can be increased when Zolmitriptan is combined with YKP-1358.
Codeine The risk or severity of CNS depression can be increased when Codeine is combined with YKP-1358.
Dihydroergotamine The risk or severity of CNS depression can be increased when Dihydroergotamine is combined with YKP-1358.
Amitriptyline The risk or severity of CNS depression can be increased when Amitriptyline is combined with YKP-1358.
Tolcapone The risk or severity of CNS depression can be increased when Tolcapone is combined with YKP-1358.
Hydromorphone The risk or severity of CNS depression can be increased when Hydromorphone is combined with YKP-1358.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with YKP-1358.
Cetirizine The risk or severity of CNS depression can be increased when Cetirizine is combined with YKP-1358.
Protriptyline The risk or severity of CNS depression can be increased when Protriptyline is combined with YKP-1358.
Trimethadione The risk or severity of CNS depression can be increased when Trimethadione is combined with YKP-1358.
Clobazam The risk or severity of sedation, somnolence, and CNS depression can be increased when Clobazam is combined with YKP-1358.
Chlorzoxazone The risk or severity of CNS depression can be increased when Chlorzoxazone is combined with YKP-1358.
Clozapine The risk or severity of CNS depression can be increased when Clozapine is combined with YKP-1358.
Meprobamate The risk or severity of CNS depression can be increased when Meprobamate is combined with YKP-1358.
Thiethylperazine The risk or severity of CNS depression can be increased when Thiethylperazine is combined with YKP-1358.
Palonosetron The risk or severity of CNS depression can be increased when Palonosetron is combined with YKP-1358.

Target Protein

5-hydroxytryptamine receptor 2A HTR2A
D(2) dopamine receptor DRD2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 17259948
    Lim KS, Kwon JS, Jang IJ, Jeong JM, Lee JS, Kim HW, Kang WJ, Kim JR, Cho JY, Kim E, Yoo SY, Shin SG, Yu KS: Modeling of brain D2 receptor occupancy-plasma concentration relationships with a novel antipsychotic, YKP1358, using serial PET scans in healthy volunteers. Clin Pharmacol Ther. 2007 Feb;81(2):252-8.

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Sekuens Gen/Protein (FASTA)

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