Peringatan Keamanan

Infusion-related reactions may occur during or after the administration which include bronchospasm, flushing, hypotension, anaphylactic shock, or cardiac arrest. Olaratumab may cause embryo-fetal toxicity based on animal data and its mechanism of action. Other reported adverse effects include neutropenia, leukopenia, anemia, nausea and musculoskeletal pain.

Olaratumab

DB06043

biotech approved investigational

Deskripsi

Olaratumab (IMC-3G3) is a fully human IgG1 monoclonal antibody with antitumor activity that selectively binds the external domain of human platelet-derived growth factor receptor (PDGFR)-? with high affinity and blocks ligand binding. It is composed of two heavy chain molecule fragments and 2 light chain fragments. Studies show that the treatment of olaratumab in combination with doxorubicin resulted in significant reduction of cancer cell proliferation and tumor growth. Olaratumab was granted accelerated approval (as Lartruvo) as initial therapy to treat adults with certain types of soft tissue sarcoma (STS) in October, 2016.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Estimated value of 11 days
Volume Distribusi 7.7 L at steady state.
Klirens (Clearance) Mean value of 0.56L/day

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Mainly degraded nonspecifically by proteolytic enzymes

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

411 Data
Diethylstilbestrol Diethylstilbestrol may increase the thrombogenic activities of Olaratumab.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Olaratumab.
Conjugated estrogens Conjugated estrogens may increase the thrombogenic activities of Olaratumab.
Estrone Estrone may increase the thrombogenic activities of Olaratumab.
Estradiol Estradiol may increase the thrombogenic activities of Olaratumab.
Dienestrol Dienestrol may increase the thrombogenic activities of Olaratumab.
Ethinylestradiol Ethinylestradiol may increase the thrombogenic activities of Olaratumab.
Mestranol Mestranol may increase the thrombogenic activities of Olaratumab.
Estriol Estriol may increase the thrombogenic activities of Olaratumab.
Estrone sulfate Estrone sulfate may increase the thrombogenic activities of Olaratumab.
Quinestrol Quinestrol may increase the thrombogenic activities of Olaratumab.
Hexestrol Hexestrol may increase the thrombogenic activities of Olaratumab.
Tibolone Tibolone may increase the thrombogenic activities of Olaratumab.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Olaratumab.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Olaratumab.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Olaratumab.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Olaratumab.
Zeranol Zeranol may increase the thrombogenic activities of Olaratumab.
Equol Equol may increase the thrombogenic activities of Olaratumab.
Promestriene Promestriene may increase the thrombogenic activities of Olaratumab.
Methallenestril Methallenestril may increase the thrombogenic activities of Olaratumab.
Epimestrol Epimestrol may increase the thrombogenic activities of Olaratumab.
Moxestrol Moxestrol may increase the thrombogenic activities of Olaratumab.
Estradiol acetate Estradiol acetate may increase the thrombogenic activities of Olaratumab.
Estradiol benzoate Estradiol benzoate may increase the thrombogenic activities of Olaratumab.
Estradiol cypionate Estradiol cypionate may increase the thrombogenic activities of Olaratumab.
Estradiol valerate Estradiol valerate may increase the thrombogenic activities of Olaratumab.
Biochanin A Biochanin A may increase the thrombogenic activities of Olaratumab.
Formononetin Formononetin may increase the thrombogenic activities of Olaratumab.
Estetrol Estetrol may increase the thrombogenic activities of Olaratumab.
Cetuximab The risk or severity of adverse effects can be increased when Cetuximab is combined with Olaratumab.
Human immunoglobulin G The risk or severity of adverse effects can be increased when Human immunoglobulin G is combined with Olaratumab.
Omalizumab The risk or severity of adverse effects can be increased when Omalizumab is combined with Olaratumab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Olaratumab.
Abciximab The risk or severity of adverse effects can be increased when Abciximab is combined with Olaratumab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Olaratumab.
Indium In-111 satumomab pendetide The risk or severity of adverse effects can be increased when Indium In-111 satumomab pendetide is combined with Olaratumab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Olaratumab.
Trastuzumab The risk or severity of adverse effects can be increased when Trastuzumab is combined with Olaratumab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Olaratumab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Olaratumab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Olaratumab.
Digoxin Immune Fab (Ovine) The risk or severity of adverse effects can be increased when Digoxin Immune Fab (Ovine) is combined with Olaratumab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Olaratumab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Olaratumab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Olaratumab.
Capromab pendetide The risk or severity of adverse effects can be increased when Capromab pendetide is combined with Olaratumab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Olaratumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Olaratumab.
Natalizumab The risk or severity of adverse effects can be increased when Natalizumab is combined with Olaratumab.
Palivizumab The risk or severity of adverse effects can be increased when Palivizumab is combined with Olaratumab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Olaratumab.
Bevacizumab The risk or severity of adverse effects can be increased when Bevacizumab is combined with Olaratumab.
Technetium Tc-99m arcitumomab The risk or severity of adverse effects can be increased when Technetium Tc-99m arcitumomab is combined with Olaratumab.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Olaratumab.
Panitumumab The risk or severity of adverse effects can be increased when Panitumumab is combined with Olaratumab.
Ranibizumab The risk or severity of adverse effects can be increased when Ranibizumab is combined with Olaratumab.
Galiximab The risk or severity of adverse effects can be increased when Galiximab is combined with Olaratumab.
Pexelizumab The risk or severity of adverse effects can be increased when Pexelizumab is combined with Olaratumab.
Afelimomab The risk or severity of adverse effects can be increased when Afelimomab is combined with Olaratumab.
Epratuzumab The risk or severity of adverse effects can be increased when Epratuzumab is combined with Olaratumab.
Bectumomab The risk or severity of adverse effects can be increased when Bectumomab is combined with Olaratumab.
Oregovomab The risk or severity of adverse effects can be increased when Oregovomab is combined with Olaratumab.
IGN311 The risk or severity of adverse effects can be increased when IGN311 is combined with Olaratumab.
Adecatumumab The risk or severity of adverse effects can be increased when Adecatumumab is combined with Olaratumab.
Labetuzumab The risk or severity of adverse effects can be increased when Labetuzumab is combined with Olaratumab.
Matuzumab The risk or severity of adverse effects can be increased when Matuzumab is combined with Olaratumab.
Fontolizumab The risk or severity of adverse effects can be increased when Fontolizumab is combined with Olaratumab.
Bavituximab The risk or severity of adverse effects can be increased when Bavituximab is combined with Olaratumab.
CR002 The risk or severity of adverse effects can be increased when CR002 is combined with Olaratumab.
Rozrolimupab The risk or severity of adverse effects can be increased when Rozrolimupab is combined with Olaratumab.
Girentuximab The risk or severity of adverse effects can be increased when Girentuximab is combined with Olaratumab.
Obiltoxaximab The risk or severity of adverse effects can be increased when Obiltoxaximab is combined with Olaratumab.
XTL-001 The risk or severity of adverse effects can be increased when XTL-001 is combined with Olaratumab.
NAV 1800 The risk or severity of adverse effects can be increased when NAV 1800 is combined with Olaratumab.
Briakinumab The risk or severity of adverse effects can be increased when Briakinumab is combined with Olaratumab.
Otelixizumab The risk or severity of adverse effects can be increased when Otelixizumab is combined with Olaratumab.
AMG 108 The risk or severity of adverse effects can be increased when AMG 108 is combined with Olaratumab.
Iratumumab The risk or severity of adverse effects can be increased when Iratumumab is combined with Olaratumab.
Enokizumab The risk or severity of adverse effects can be increased when Enokizumab is combined with Olaratumab.
Ramucirumab The risk or severity of adverse effects can be increased when Ramucirumab is combined with Olaratumab.
Farletuzumab The risk or severity of adverse effects can be increased when Farletuzumab is combined with Olaratumab.
Veltuzumab The risk or severity of adverse effects can be increased when Veltuzumab is combined with Olaratumab.
Ustekinumab The risk or severity of adverse effects can be increased when Ustekinumab is combined with Olaratumab.
Trastuzumab emtansine The risk or severity of adverse effects can be increased when Trastuzumab emtansine is combined with Olaratumab.
PRO-542 The risk or severity of adverse effects can be increased when PRO-542 is combined with Olaratumab.
TNX-901 The risk or severity of adverse effects can be increased when TNX-901 is combined with Olaratumab.
Inotuzumab ozogamicin The risk or severity of adverse effects can be increased when Inotuzumab ozogamicin is combined with Olaratumab.
RI 624 The risk or severity of adverse effects can be increased when RI 624 is combined with Olaratumab.
Stamulumab The risk or severity of adverse effects can be increased when MYO-029 is combined with Olaratumab.
CT-011 The risk or severity of adverse effects can be increased when CT-011 is combined with Olaratumab.
Leronlimab The risk or severity of adverse effects can be increased when Leronlimab is combined with Olaratumab.
Glembatumumab vedotin The risk or severity of adverse effects can be increased when Glembatumumab vedotin is combined with Olaratumab.
IPH 2101 The risk or severity of adverse effects can be increased when Olaratumab is combined with IPH 2101.
TB-402 The risk or severity of adverse effects can be increased when Olaratumab is combined with TB-402.
Caplacizumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Caplacizumab.
IMC-1C11 The risk or severity of adverse effects can be increased when Olaratumab is combined with IMC-1C11.
Eldelumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Eldelumab.
Lumiliximab The risk or severity of adverse effects can be increased when Olaratumab is combined with Lumiliximab.
Canakinumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Canakinumab.

Target Protein

Platelet-derived growth factor receptor alpha PDGFRA

Referensi & Sumber

Artikel (PubMed)
  • PMID: 17234763
    Dolloff NG, Russell MR, Loizos N, Fatatis A: Human bone marrow activates the Akt pathway in metastatic prostate cells through transactivation of the alpha-platelet-derived growth factor receptor. Cancer Res. 2007 Jan 15;67(2):555-62.
  • PMID: 27995580
    Shirley M: Olaratumab: First Global Approval. Drugs. 2016 Dec 19.
  • PMID: 24816152
    Doi T, Ma Y, Dontabhaktuni A, Nippgen C, Nippgen J, Ohtsu A: Phase I study of olaratumab in Japanese patients with advanced solid tumors. Cancer Sci. 2014 Jul;105(7):862-9. doi: 10.1111/cas.12444. Epub 2014 Jun 27.
  • PMID: 28205191
    Knepper TC, Saller J, Walko CM: Novel and Expanded Oncology Drug Approvals of 2016-PART 1: New Options in Solid Tumor Management. Oncology (Williston Park). 2017 Feb 15;31(2):110-21.
  • PMID: 28426120
    Wagner AJ, Kindler H, Gelderblom H, Schoffski P, Bauer S, Hohenberger P, Kopp HG, Lopez-Martin JA, Peeters M, Reichardt P, Qin A, Nippgen J, Ilaria RL, Rutkowski P: A phase II study of a human anti-PDGFRalpha monoclonal antibody (olaratumab, IMC-3G3) in previously treated patients with metastatic gastrointestinal stromal tumors. Ann Oncol. 2017 Mar 1;28(3):541-546. doi: 10.1093/annonc/mdw659.
  • PMID: 27291997
    Tap WD, Jones RL, Van Tine BA, Chmielowski B, Elias AD, Adkins D, Agulnik M, Cooney MM, Livingston MB, Pennock G, Hameed MR, Shah GD, Qin A, Shahir A, Cronier DM, Ilaria R Jr, Conti I, Cosaert J, Schwartz GK: Olaratumab and doxorubicin versus doxorubicin alone for treatment of soft-tissue sarcoma: an open-label phase 1b and randomised phase 2 trial. Lancet. 2016 Jul 30;388(10043):488-97. doi: 10.1016/S0140-6736(16)30587-6. Epub 2016 Jun 9.

Contoh Produk & Brand

Produk: 7 • International brands: 0
Produk
  • Lartruvo
    Injection, solution, concentrate • 10 mg/ml • Intravenous • EU
  • Lartruvo
    Injection, solution, concentrate • 10 mg/ml • Intravenous • EU
  • Lartruvo
    Injection, solution, concentrate • 10 mg/ml • Intravenous • EU
  • Lartruvo
    Solution • 500 mg / 50 mL • Intravenous • Canada • Approved
  • Lartruvo
    Injection, solution • 10 mg/1mL • Intravenous • US • Approved
  • Lartruvo
    Injection, solution • 10 mg/1mL • Intravenous • US • Approved
  • Lartruvo
    Solution • 190 mg / 19 mL • Intravenous • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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