Dovitinib

DB05928

small molecule investigational

Deskripsi

Dovitinib is an orally active small molecule that exhibits potent inhibitory activity against multiple RTKs involved in tumor growth and angiogenesis. Preclinical data show that dovitinib works to inhibit multiple kinases associated with different cancers, including acute myeloid leukemia (AML) and multiple myeloma. Chiron currently has three ongoing Phase I clinical trials for dovitinib.

Struktur Molekul 2D

Berat 392.438
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

563 Data
Lomitapide The metabolism of Lomitapide can be decreased when combined with Dovitinib.
Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Dovitinib.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Dovitinib.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Dovitinib.
Colchicine The metabolism of Colchicine can be decreased when combined with Dovitinib.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Dovitinib.
Retapamulin The metabolism of Retapamulin can be decreased when combined with Dovitinib.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with Dovitinib.
Vardenafil The metabolism of Vardenafil can be decreased when combined with Dovitinib.
Eszopiclone The metabolism of Eszopiclone can be decreased when combined with Dovitinib.
Zopiclone The metabolism of Zopiclone can be decreased when combined with Dovitinib.
Lovastatin The metabolism of Lovastatin can be decreased when combined with Dovitinib.
Acetaminophen The serum concentration of Acetaminophen can be increased when it is combined with Dovitinib.
Propacetamol The serum concentration of Propacetamol can be increased when it is combined with Dovitinib.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with Dovitinib.
Alprazolam The metabolism of Alprazolam can be decreased when combined with Dovitinib.
Warfarin The serum concentration of Warfarin can be increased when it is combined with Dovitinib.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with Dovitinib.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with Dovitinib.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with Dovitinib.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with Dovitinib.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with Dovitinib.
Midazolam The serum concentration of Midazolam can be increased when it is combined with Dovitinib.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with Dovitinib.
Atorvastatin The metabolism of Atorvastatin can be decreased when combined with Dovitinib.
Eluxadoline The serum concentration of Eluxadoline can be increased when it is combined with Dovitinib.
Folic acid Dovitinib may decrease the excretion rate of Folic acid which could result in a higher serum level.
Allopurinol Dovitinib may decrease the excretion rate of Allopurinol which could result in a higher serum level.
Raloxifene Dovitinib may decrease the excretion rate of Raloxifene which could result in a higher serum level.
Celecoxib Dovitinib may decrease the excretion rate of Celecoxib which could result in a higher serum level.
Oxaliplatin Dovitinib may decrease the excretion rate of Oxaliplatin which could result in a higher serum level.
Testosterone Dovitinib may decrease the excretion rate of Testosterone which could result in a higher serum level.
Clofarabine Dovitinib may decrease the excretion rate of Clofarabine which could result in a higher serum level.
Nitrofurantoin Dovitinib may decrease the excretion rate of Nitrofurantoin which could result in a higher serum level.
Riluzole Dovitinib may decrease the excretion rate of Riluzole which could result in a higher serum level.
Sulfasalazine Dovitinib may decrease the excretion rate of Sulfasalazine which could result in a higher serum level.
Glyburide Dovitinib may decrease the excretion rate of Glyburide which could result in a higher serum level.
Tegaserod Dovitinib may decrease the excretion rate of Tegaserod which could result in a higher serum level.
Leflunomide Dovitinib may decrease the excretion rate of Leflunomide which could result in a higher serum level.
Rosuvastatin Dovitinib may decrease the excretion rate of Rosuvastatin which could result in a higher serum level.
Alvocidib Dovitinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Teriflunomide Dovitinib may decrease the excretion rate of Teriflunomide which could result in a higher serum level.
Riociguat Dovitinib may decrease the excretion rate of Riociguat which could result in a higher serum level.
Fimasartan Dovitinib may decrease the excretion rate of Fimasartan which could result in a higher serum level.
Delafloxacin Dovitinib may decrease the excretion rate of Delafloxacin which could result in a higher serum level.
Glasdegib Dovitinib may decrease the excretion rate of Glasdegib which could result in a higher serum level.
Testosterone cypionate Dovitinib may decrease the excretion rate of Testosterone cypionate which could result in a higher serum level.
Testosterone enanthate Dovitinib may decrease the excretion rate of Testosterone enanthate which could result in a higher serum level.
Darolutamide Dovitinib may decrease the excretion rate of Darolutamide which could result in a higher serum level.
Tazemetostat Dovitinib may decrease the excretion rate of Tazemetostat which could result in a higher serum level.
Conjugated estrogens Dovitinib may decrease the excretion rate of Conjugated estrogens which could result in a higher serum level.
Gefitinib Dovitinib may decrease the excretion rate of Gefitinib which could result in a higher serum level.
Cerivastatin Dovitinib may decrease the excretion rate of Cerivastatin which could result in a higher serum level.
Prazosin Dovitinib may decrease the excretion rate of Prazosin which could result in a higher serum level.
Zidovudine Dovitinib may decrease the excretion rate of Zidovudine which could result in a higher serum level.
Ritonavir Dovitinib may decrease the excretion rate of Ritonavir which could result in a higher serum level.
Ivermectin Dovitinib may decrease the excretion rate of Ivermectin which could result in a higher serum level.
Sumatriptan Dovitinib may decrease the excretion rate of Sumatriptan which could result in a higher serum level.
Mycophenolate mofetil Dovitinib may decrease the excretion rate of Mycophenolate mofetil which could result in a higher serum level.
Lamivudine Dovitinib may decrease the excretion rate of Lamivudine which could result in a higher serum level.
Donepezil Dovitinib may decrease the excretion rate of Donepezil which could result in a higher serum level.
Ezetimibe Dovitinib may decrease the excretion rate of Ezetimibe which could result in a higher serum level.
Topotecan Dovitinib may decrease the excretion rate of Topotecan which could result in a higher serum level.
Mitoxantrone Dovitinib may decrease the excretion rate of Mitoxantrone which could result in a higher serum level.
Camptothecin Dovitinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Pitavastatin The metabolism of Pitavastatin can be decreased when combined with Dovitinib.
Afatinib Dovitinib may decrease the excretion rate of Afatinib which could result in a higher serum level.
Tenofovir alafenamide The serum concentration of Tenofovir alafenamide can be increased when it is combined with Dovitinib.
Pravastatin Dovitinib may decrease the excretion rate of Pravastatin which could result in a higher serum level.
Dactinomycin Dovitinib may decrease the excretion rate of Dactinomycin which could result in a higher serum level.
Simeprevir Dovitinib may decrease the excretion rate of Simeprevir which could result in a higher serum level.
Apixaban Dovitinib may decrease the excretion rate of Apixaban which could result in a higher serum level.
Dolutegravir Dovitinib may decrease the excretion rate of Dolutegravir which could result in a higher serum level.
Sofosbuvir Dovitinib may decrease the excretion rate of Sofosbuvir which could result in a higher serum level.
Lenvatinib Dovitinib may decrease the excretion rate of Lenvatinib which could result in a higher serum level.
Ombitasvir Dovitinib may decrease the excretion rate of Ombitasvir which could result in a higher serum level.
Velpatasvir Dovitinib may decrease the excretion rate of Velpatasvir which could result in a higher serum level.
Talazoparib The serum concentration of Talazoparib can be increased when it is combined with Dovitinib.
Duvelisib Dovitinib may decrease the excretion rate of Duvelisib which could result in a higher serum level.
Voxilaprevir Dovitinib may decrease the excretion rate of Voxilaprevir which could result in a higher serum level.
Rucaparib Dovitinib may decrease the excretion rate of Rucaparib which could result in a higher serum level.
Lusutrombopag Dovitinib may decrease the excretion rate of Lusutrombopag which could result in a higher serum level.
Pibrentasvir Dovitinib may decrease the excretion rate of Pibrentasvir which could result in a higher serum level.
Glecaprevir Dovitinib may decrease the excretion rate of Glecaprevir which could result in a higher serum level.
Tucatinib Dovitinib may decrease the excretion rate of Tucatinib which could result in a higher serum level.
Rivaroxaban Dovitinib may decrease the excretion rate of Rivaroxaban which could result in a higher serum level.
Selumetinib Dovitinib may decrease the excretion rate of Selumetinib which could result in a higher serum level.
Pralatrexate Dovitinib may decrease the excretion rate of Pralatrexate which could result in a higher serum level.
Ripretinib Dovitinib may decrease the excretion rate of Ripretinib which could result in a higher serum level.
Daunorubicin Dovitinib may decrease the excretion rate of Daunorubicin which could result in a higher serum level.
Fostemsavir Dovitinib may decrease the excretion rate of Fostemsavir which could result in a higher serum level.
Pralsetinib Dovitinib may decrease the excretion rate of Pralsetinib which could result in a higher serum level.
Trilaciclib Dovitinib may decrease the excretion rate of Trilaciclib which could result in a higher serum level.
Aripiprazole The metabolism of Aripiprazole can be decreased when combined with Dovitinib.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be decreased when combined with Dovitinib.
Valsartan The excretion of Valsartan can be decreased when combined with Dovitinib.
Torasemide The excretion of Torasemide can be decreased when combined with Dovitinib.
Caspofungin The excretion of Caspofungin can be decreased when combined with Dovitinib.
Bosentan The excretion of Bosentan can be decreased when combined with Dovitinib.
Enalapril The excretion of Enalapril can be decreased when combined with Dovitinib.

Target Protein

Nuclear receptor subfamily 1 group I member 2 NR1I2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16914579
    Xin X, Abrams TJ, Hollenbach PW, Rendahl KG, Tang Y, Oei YA, Embry MG, Swinarski DE, Garrett EN, Pryer NK, Trudel S, Jallal B, Mendel DB, Heise CC: CHIR-258 is efficacious in a newly developed fibroblast growth factor receptor 3-expressing orthotopic multiple myeloma model in mice. Clin Cancer Res. 2006 Aug 15;12(16):4908-15.
  • PMID: 15598814
    Trudel S, Li ZH, Wei E, Wiesmann M, Chang H, Chen C, Reece D, Heise C, Stewart AK: CHIR-258, a novel, multitargeted tyrosine kinase inhibitor for the potential treatment of t(4;14) multiple myeloma. Blood. 2005 Apr 1;105(7):2941-8. Epub 2004 Dec 14.

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