Sar9, Met (O2)11-Substance P

DB05875

small molecule investigational

Deskripsi

Sar9, Met (O2)11-Substance P is a neurokinin-1 receptor agonist. It is an analog of the naturally occurring human neuropeptide Substance P, which can be found throughout the body, including in the airways of humans and many other species.

Struktur Molekul 2D

Berat 1393.68
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

75 Data
Pegvisomant Pegvisomant may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Mefloquine Mefloquine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Tacrine Tacrine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Sulpiride Sulpiride may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Profenamine Profenamine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Chlorpromazine Chlorpromazine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Gallamine triethiodide Gallamine triethiodide may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Triflupromazine Triflupromazine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Cisplatin Cisplatin may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Cinchocaine Cinchocaine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Pyridostigmine Pyridostigmine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Nizatidine Nizatidine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Galantamine Galantamine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Isoflurophate Isoflurophate may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Diethylcarbamazine Diethylcarbamazine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Procaine Procaine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Minaprine Minaprine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Donepezil Donepezil may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Terbutaline Terbutaline may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Mechlorethamine Mechlorethamine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Hexafluronium Hexafluronium may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Demecarium Demecarium may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Physostigmine Physostigmine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Rivastigmine Rivastigmine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Edrophonium Edrophonium may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Procainamide Procainamide may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Memantine Memantine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Ambenonium Ambenonium may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Tubocurarine Tubocurarine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Ketamine Ketamine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Metoclopramide Metoclopramide may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Decamethonium Decamethonium may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Pancuronium Pancuronium may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Pipecuronium Pipecuronium may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Ginkgo biloba Ginkgo biloba may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Neostigmine Neostigmine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Bambuterol Bambuterol may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
1,10-Phenanthroline 1,10-Phenanthroline may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Thiotepa Thiotepa may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Huperzine A Huperzine A may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Phenserine Phenserine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Regramostim Regramostim may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Aprotinin Aprotinin may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Betaine Betaine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Capsaicin Capsaicin may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Coumaphos Coumaphos may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Dichlorvos Dichlorvos may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Fenthion Fenthion may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Metrifonate Metrifonate may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Acotiamide Acotiamide may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Methanesulfonyl Fluoride Methanesulfonyl Fluoride may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Paraoxon Paraoxon may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Tyrothricin Tyrothricin may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Ipidacrine Ipidacrine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Distigmine Distigmine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Tretamine Tretamine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Posiphen Posiphen may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Methylphosphinic Acid Methylphosphinic Acid may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Succinylcholine The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Succinylcholine.
Cocaine The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Cocaine.
Trimethaphan The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Trimethaphan.
Doxacurium The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Doxacurium.
Chloroprocaine The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Chloroprocaine.
Ephedrine The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Ephedrine.
Clevidipine The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Clevidipine.
Mirabegron The serum concentration of Mirabegron can be increased when it is combined with Sar9, Met (O2)11-Substance P.
Aclidinium The serum concentration of Aclidinium can be increased when it is combined with Sar9, Met (O2)11-Substance P.
Moxisylyte The serum concentration of Moxisylyte can be increased when it is combined with Sar9, Met (O2)11-Substance P.
Propacetamol The serum concentration of Propacetamol can be increased when it is combined with Sar9, Met (O2)11-Substance P.
Butyrylthiocholine The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Butyrylthiocholine.
Oxybuprocaine The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Oxybuprocaine.
Benzonatate The serum concentration of Sar9, Met (O2)11-Substance P can be increased when it is combined with Benzonatate.
Isoprenaline Isoprenaline may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Isavuconazonium The serum concentration of Isavuconazonium can be increased when it is combined with Sar9, Met (O2)11-Substance P.
Benzgalantamine Benzgalantamine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 18289674
    Grimsholm O, Rantapaa-Dahlqvist S, Dalen T, Forsgren S: Observations favouring the occurrence of local production and marked effects of bombesin/gastrin-releasing peptide in the synovial tissue of the human knee joint--comparisons with substance P and the NK-1 receptor. Neuropeptides. 2008 Apr;42(2):133-45. doi: 10.1016/j.npep.2007.12.008.
  • PMID: 2476938
    Rothstein RD, Johnson E, Ouyang A: Substance P: mechanism of action and receptor distribution at the feline ileocecal sphincter region. Am J Physiol. 1989 Sep;257(3 Pt 1):G447-53.
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