GPI-1485

DB05814

small molecule investigational

Deskripsi

GPI 1485 is a product candidate that belongs to a class of small molecule compounds called neuroimmunophilin ligands.
In preclinical experiments, neuroimmunophilin ligands have been shown to repair and regenerate damaged nerves without affecting normal, healthy nerves.
GPI 1485 is being studied in phase 2 clinical trials for the treatment of Parkinson's disease and post-prostatectomy erectile dysfunction and in pre-clinical development for HIV related dementia and neuropathy.

Struktur Molekul 2D

Berat 241.287
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

174 Data
Eliglustat The metabolism of Eliglustat can be decreased when combined with GPI-1485.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with GPI-1485.
Cilostazol The metabolism of Cilostazol can be decreased when combined with GPI-1485.
Colchicine The metabolism of Colchicine can be decreased when combined with GPI-1485.
Iloperidone The metabolism of Iloperidone can be decreased when combined with GPI-1485.
Retapamulin The metabolism of Retapamulin can be decreased when combined with GPI-1485.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with GPI-1485.
Vardenafil The metabolism of Vardenafil can be decreased when combined with GPI-1485.
Eszopiclone The metabolism of Eszopiclone can be decreased when combined with GPI-1485.
Zopiclone The metabolism of Zopiclone can be decreased when combined with GPI-1485.
Lovastatin The metabolism of Lovastatin can be decreased when combined with GPI-1485.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with GPI-1485.
Alprazolam The metabolism of Alprazolam can be decreased when combined with GPI-1485.
Warfarin The serum concentration of Warfarin can be increased when it is combined with GPI-1485.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with GPI-1485.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with GPI-1485.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with GPI-1485.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with GPI-1485.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with GPI-1485.
Midazolam The serum concentration of Midazolam can be increased when it is combined with GPI-1485.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with GPI-1485.
Atorvastatin The metabolism of Atorvastatin can be decreased when combined with GPI-1485.
Aripiprazole The metabolism of Aripiprazole can be decreased when combined with GPI-1485.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be decreased when combined with GPI-1485.
Azithromycin The metabolism of Azithromycin can be decreased when combined with GPI-1485.
Ziprasidone The metabolism of Ziprasidone can be decreased when combined with GPI-1485.
Chlorpromazine The metabolism of Chlorpromazine can be decreased when combined with GPI-1485.
Albendazole The metabolism of Albendazole can be decreased when combined with GPI-1485.
Cephalexin The metabolism of Cephalexin can be decreased when combined with GPI-1485.
Doxazosin The metabolism of Doxazosin can be decreased when combined with GPI-1485.
Norethisterone The metabolism of Norethisterone can be decreased when combined with GPI-1485.
Fenofibrate The metabolism of Fenofibrate can be decreased when combined with GPI-1485.
Atazanavir The metabolism of Atazanavir can be decreased when combined with GPI-1485.
Rosuvastatin The metabolism of Rosuvastatin can be decreased when combined with GPI-1485.
Drospirenone The metabolism of Drospirenone can be decreased when combined with GPI-1485.
Allylestrenol The metabolism of Allylestrenol can be decreased when combined with GPI-1485.
Zuclopenthixol The metabolism of Zuclopenthixol can be decreased when combined with GPI-1485.
Roflumilast The serum concentration of Roflumilast can be increased when it is combined with GPI-1485.
Lacosamide The metabolism of Lacosamide can be decreased when combined with GPI-1485.
Linagliptin The metabolism of Linagliptin can be decreased when combined with GPI-1485.
Vorapaxar The metabolism of Vorapaxar can be decreased when combined with GPI-1485.
Suvorexant The metabolism of Suvorexant can be decreased when combined with GPI-1485.
Netupitant The metabolism of Netupitant can be decreased when combined with GPI-1485.
Tasimelteon The metabolism of Tasimelteon can be decreased when combined with GPI-1485.
Nintedanib The metabolism of Nintedanib can be decreased when combined with GPI-1485.
Tenofovir alafenamide The metabolism of Tenofovir alafenamide can be decreased when combined with GPI-1485.
Dihydroergocornine The metabolism of Dihydroergocornine can be decreased when combined with GPI-1485.
Duvelisib The metabolism of Duvelisib can be decreased when combined with GPI-1485.
Gilteritinib The metabolism of Gilteritinib can be decreased when combined with GPI-1485.
9-aminocamptothecin The metabolism of 9-aminocamptothecin can be decreased when combined with GPI-1485.
Methylprednisone The metabolism of Methylprednisone can be decreased when combined with GPI-1485.
Dihydroergocristine The metabolism of Dihydroergocristine can be decreased when combined with GPI-1485.
Dihydroergocryptine The metabolism of Dihydroergocryptine can be decreased when combined with GPI-1485.
Medical Cannabis The metabolism of Medical Cannabis can be decreased when combined with GPI-1485.
Elexacaftor The metabolism of Elexacaftor can be decreased when combined with GPI-1485.
Tazemetostat The metabolism of Tazemetostat can be decreased when combined with GPI-1485.
Fosaprepitant The metabolism of Fosaprepitant can be decreased when combined with GPI-1485.
Lefamulin The metabolism of Lefamulin can be decreased when combined with GPI-1485.
Methysergide The metabolism of Methysergide can be decreased when combined with GPI-1485.
Meperidine The metabolism of Meperidine can be decreased when combined with GPI-1485.
Ebastine The metabolism of Ebastine can be decreased when combined with GPI-1485.
Terfenadine The metabolism of Terfenadine can be decreased when combined with GPI-1485.
Cisapride The metabolism of Cisapride can be decreased when combined with GPI-1485.
Isavuconazole The metabolism of Isavuconazole can be decreased when combined with GPI-1485.
Pretomanid The metabolism of Pretomanid can be decreased when combined with GPI-1485.
Pimavanserin The metabolism of Pimavanserin can be decreased when combined with GPI-1485.
Estetrol The metabolism of Estetrol can be decreased when combined with GPI-1485.
Infigratinib The metabolism of Infigratinib can be decreased when combined with GPI-1485.
Cyclosporine The serum concentration of Cyclosporine can be increased when it is combined with GPI-1485.
Dofetilide The serum concentration of Dofetilide can be increased when it is combined with GPI-1485.
Theophylline The serum concentration of Theophylline can be increased when it is combined with GPI-1485.
Carbamazepine The serum concentration of Carbamazepine can be increased when it is combined with GPI-1485.
Sirolimus The serum concentration of Sirolimus can be increased when it is combined with GPI-1485.
Quinidine The serum concentration of Quinidine can be increased when it is combined with GPI-1485.
Phenprocoumon The serum concentration of Phenprocoumon can be increased when it is combined with GPI-1485.
Busulfan The serum concentration of Busulfan can be increased when it is combined with GPI-1485.
Pimozide The serum concentration of Pimozide can be increased when it is combined with GPI-1485.
Amiodarone The serum concentration of Amiodarone can be increased when it is combined with GPI-1485.
Aminophylline The serum concentration of Aminophylline can be increased when it is combined with GPI-1485.
Paclitaxel The serum concentration of Paclitaxel can be increased when it is combined with GPI-1485.
Dasatinib The serum concentration of Dasatinib can be increased when it is combined with GPI-1485.
Fosphenytoin The serum concentration of Fosphenytoin can be increased when it is combined with GPI-1485.
Digitoxin The serum concentration of Digitoxin can be increased when it is combined with GPI-1485.
Everolimus The serum concentration of Everolimus can be increased when it is combined with GPI-1485.
Dronedarone The serum concentration of Dronedarone can be increased when it is combined with GPI-1485.
Cobimetinib The serum concentration of Cobimetinib can be increased when it is combined with GPI-1485.
Temsirolimus The serum concentration of Temsirolimus can be increased when it is combined with GPI-1485.
Idelalisib The serum concentration of Idelalisib can be increased when it is combined with GPI-1485.
Ceritinib The serum concentration of Ceritinib can be increased when it is combined with GPI-1485.
Tianeptine The serum concentration of Tianeptine can be increased when it is combined with GPI-1485.
Osimertinib The serum concentration of Osimertinib can be increased when it is combined with GPI-1485.
Ribociclib The serum concentration of Ribociclib can be increased when it is combined with GPI-1485.
Dacomitinib The serum concentration of Dacomitinib can be increased when it is combined with GPI-1485.
Alpelisib The serum concentration of Alpelisib can be increased when it is combined with GPI-1485.
Astemizole The serum concentration of Astemizole can be increased when it is combined with GPI-1485.
Lomitapide The serum concentration of Lomitapide can be increased when it is combined with GPI-1485.
Siponimod The serum concentration of Siponimod can be increased when it is combined with GPI-1485.
Methotrexate The serum concentration of Methotrexate can be increased when it is combined with GPI-1485.
Vinorelbine The serum concentration of Vinorelbine can be increased when it is combined with GPI-1485.
Vincristine The serum concentration of Vincristine can be increased when it is combined with GPI-1485.

Target Protein

Peptidyl-prolyl cis-trans isomerase FKBP1A FKBP1A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 17200487
    Authors unspecified: A randomized clinical trial of coenzyme Q10 and GPI-1485 in early Parkinson disease. Neurology. 2007 Jan 2;68(1):20-8.
  • PMID: 14983983
    Marshall VL, Grosset DG: GPI-1485 (Guilford). Curr Opin Investig Drugs. 2004 Jan;5(1):107-12.

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