Irofulven

DB05786

small molecule investigational

Deskripsi

A novel anti-cancer compound synthesized by scientists at the University of California, San Diego more than a decade ago from toxins of the poisonous jack-o-lantern mushroom, has been granted “fast track” status by the U.S. Food and Drug Administration (FDA) after demonstrating promise against one of the most deadly cancers.

MGI-114 (Irofulven) is currently being developed by MGI PHARMA, Inc., an emerging oncology-focused pharmaceutical company based in Minneapolis. Phase III clinical trials involving the drug have been underway since early 2001 at sites in the U.S. and Europe.

Struktur Molekul 2D

Berat 246.3016
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

39 Data
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Irofulven.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Irofulven.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Irofulven.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Irofulven.
Lidocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Quinisocaine.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Irofulven.
Ambroxol The risk or severity of methemoglobinemia can be increased when Irofulven is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Irofulven is combined with Etrasimod.

Target Protein

Serine/threonine-protein kinase Chk2 CHEK2
Far upstream element-binding protein 1 FUBP1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 10637489
    Kelner MJ, McMorris TC, Estes L, Samson KM, Trani NA, MacDonald JR: Anti-leukemic action of the novel agent MGI 114 (HMAF) and synergistic action with topotecan. Leukemia. 2000 Jan;14(1):136-41.
  • PMID: 12231547
    Leggas M, Stewart CF, Woo MH, Fouladi M, Cheshire PJ, Peterson JK, Friedman HS, Billups C, Houghton PJ: Relation between Irofulven (MGI-114) systemic exposure and tumor response in human solid tumor xenografts. Clin Cancer Res. 2002 Sep;8(9):3000-7.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Irofulven

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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