SN-38

DB05482

small molecule investigational

Deskripsi

7-ethyl-10-hydroxycamptothecin (SN 38) is a liposomal formulation of the active metabolite of Irinotecan DB00762, a chemotherapeutic pro-drug approved for the treatment of advanced colorectal cancer. SN 38 has been used in trials studying the treatment of Cancer, Advanced Solid Tumors, Small Cell Lung Cancer, Metastatic Colorectal Cancer, and Triple Negative Breast Cancer, among others.

Struktur Molekul 2D

Berat 392.4046
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

297 Data
Eliglustat The metabolism of Eliglustat can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Cilostazol The metabolism of Cilostazol can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Colchicine The metabolism of Colchicine can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Iloperidone The metabolism of Iloperidone can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Retapamulin The metabolism of Retapamulin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Vardenafil The metabolism of Vardenafil can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Eszopiclone The metabolism of Eszopiclone can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Zopiclone The metabolism of Zopiclone can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Lovastatin The metabolism of Lovastatin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Alprazolam The metabolism of Alprazolam can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Warfarin The serum concentration of Warfarin can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Midazolam The serum concentration of Midazolam can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Atorvastatin The metabolism of Atorvastatin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Pitolisant The serum concentration of 7-ethyl-10-hydroxycamptothecin can be decreased when it is combined with Pitolisant.
Aripiprazole The metabolism of Aripiprazole can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Metreleptin The metabolism of 7-ethyl-10-hydroxycamptothecin can be increased when combined with Metreleptin.
Azithromycin The metabolism of Azithromycin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Chlorpromazine The metabolism of Chlorpromazine can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Albendazole The metabolism of Albendazole can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Cephalexin The metabolism of Cephalexin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Doxazosin The metabolism of Doxazosin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Norethisterone The metabolism of Norethisterone can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Fenofibrate The metabolism of Fenofibrate can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Rosuvastatin The metabolism of Rosuvastatin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Allylestrenol The metabolism of Allylestrenol can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Zuclopenthixol The metabolism of Zuclopenthixol can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Roflumilast The serum concentration of Roflumilast can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Lacosamide The metabolism of Lacosamide can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Vorapaxar The metabolism of Vorapaxar can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Suvorexant The metabolism of Suvorexant can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Tasimelteon The metabolism of Tasimelteon can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Nintedanib The metabolism of Nintedanib can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Tenofovir alafenamide The metabolism of Tenofovir alafenamide can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Dihydroergocornine The metabolism of Dihydroergocornine can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Duvelisib The metabolism of Duvelisib can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Gilteritinib The metabolism of Gilteritinib can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
9-aminocamptothecin The metabolism of 9-aminocamptothecin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Methylprednisone The metabolism of Methylprednisone can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Dihydroergocristine The metabolism of Dihydroergocristine can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Dihydroergocryptine The metabolism of Dihydroergocryptine can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Medical Cannabis The metabolism of Medical Cannabis can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Drospirenone The metabolism of Drospirenone can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Ziprasidone The metabolism of 7-ethyl-10-hydroxycamptothecin can be decreased when combined with Ziprasidone.
Linagliptin The metabolism of 7-ethyl-10-hydroxycamptothecin can be decreased when combined with Linagliptin.
Netupitant The metabolism of 7-ethyl-10-hydroxycamptothecin can be decreased when combined with Netupitant.
Elexacaftor The metabolism of Elexacaftor can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Tazemetostat The metabolism of Tazemetostat can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Fosaprepitant The metabolism of Fosaprepitant can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Lefamulin The metabolism of Lefamulin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Methysergide The metabolism of Methysergide can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Meperidine The metabolism of Meperidine can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Ebastine The metabolism of Ebastine can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Cisapride The metabolism of Cisapride can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Isavuconazole The metabolism of 7-ethyl-10-hydroxycamptothecin can be decreased when combined with Isavuconazole.
Pretomanid The metabolism of Pretomanid can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Pimavanserin The metabolism of Pimavanserin can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Estetrol The metabolism of Estetrol can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Infigratinib The metabolism of Infigratinib can be decreased when combined with 7-ethyl-10-hydroxycamptothecin.
Cobimetinib The serum concentration of Cobimetinib can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Ceritinib The serum concentration of Ceritinib can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Dacomitinib The serum concentration of Dacomitinib can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Alpelisib The serum concentration of Alpelisib can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Cyclosporine The serum concentration of Cyclosporine can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Dofetilide The serum concentration of Dofetilide can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Theophylline The serum concentration of Theophylline can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Carbamazepine The serum concentration of Carbamazepine can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Sirolimus The serum concentration of Sirolimus can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Quinidine The serum concentration of Quinidine can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Phenprocoumon The serum concentration of Phenprocoumon can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Busulfan The serum concentration of Busulfan can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Pimozide The serum concentration of Pimozide can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Aminophylline The serum concentration of Aminophylline can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Paclitaxel The serum concentration of Paclitaxel can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Dasatinib The serum concentration of Dasatinib can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Digitoxin The serum concentration of Digitoxin can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Everolimus The serum concentration of Everolimus can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Dronedarone The serum concentration of Dronedarone can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Temsirolimus The serum concentration of Temsirolimus can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Tianeptine The serum concentration of Tianeptine can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Fosphenytoin The serum concentration of Fosphenytoin can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Idelalisib The serum concentration of Idelalisib can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Osimertinib The serum concentration of Osimertinib can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Astemizole The serum concentration of Astemizole can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Lomitapide The serum concentration of Lomitapide can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Siponimod The serum concentration of Siponimod can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Methotrexate The serum concentration of Methotrexate can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Vinorelbine The serum concentration of Vinorelbine can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Vincristine The serum concentration of Vincristine can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Vinblastine The serum concentration of Vinblastine can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.
Doxorubicin The serum concentration of Doxorubicin can be increased when it is combined with 7-ethyl-10-hydroxycamptothecin.

Target Protein

DNA topoisomerase 1 TOP1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16386867
    Xuan T, Zhang JA, Ahmad I: HPLC method for determination of SN-38 content and SN-38 entrapment efficiency in a novel liposome-based formulation, LE-SN38. J Pharm Biomed Anal. 2006 May 3;41(2):582-8. Epub 2006 Jan 18.
  • PMID: 15996839
    Peikov V, Ugwu S, Parmar M, Zhang A, Ahmad I: pH-dependent association of SN-38 with lipid bilayers of a novel liposomal formulation. Int J Pharm. 2005 Aug 11;299(1-2):92-9.
  • PMID: 15816556
    Pal A, Khan S, Wang YF, Kamath N, Sarkar AK, Ahmad A, Sheikh S, Ali S, Carbonaro D, Zhang A, Ahmad I: Preclinical safety, pharmacokinetics and antitumor efficacy profile of liposome-entrapped SN-38 formulation. Anticancer Res. 2005 Jan-Feb;25(1A):331-41.
  • PMID: 15664753
    Khan S, Ahmad A, Guo W, Wang YF, Abu-Qare A, Ahmad I: A simple and sensitive LC/MS/MS assay for 7-ethyl-10-hydroxycamptothecin (SN-38) in mouse plasma and tissues: application to pharmacokinetic study of liposome entrapped SN-38 (LE-SN38). J Pharm Biomed Anal. 2005 Feb 7;37(1):135-42.
  • PMID: 15494639
    Lei S, Chien PY, Sheikh S, Zhang A, Ali S, Ahmad I: Enhanced therapeutic efficacy of a novel liposome-based formulation of SN-38 against human tumor models in SCID mice. Anticancer Drugs. 2004 Sep;15(8):773-8.
  • PMID: 14726126
    Zhang JA, Xuan T, Parmar M, Ma L, Ugwu S, Ali S, Ahmad I: Development and characterization of a novel liposome-based formulation of SN-38. Int J Pharm. 2004 Feb 11;270(1-2):93-107.
  • PMID: 14648604
    Khan S, Ahmad A, Ahmad I: A sensitive and rapid liquid chromatography tandem mass spectrometry method for quantitative determination of 7-ethyl-10-hydroxycamptothecin (SN-38) in human plasma containing liposome-based SN-38 (LE-SN38). Biomed Chromatogr. 2003 Dec;17(8):493-9.
  • PMID: 12798168
    Guo W, Ahmad A, Khan S, Dahhani F, Wang YF, Ahmad I: Determination by liquid chromatography with fluorescence detection of total 7-ethyl-10-hydroxy-camptothecin (SN-38) in beagle dog plasma after intravenous administration of liposome-based SN-38 (LE-SN38). J Chromatogr B Analyt Technol Biomed Life Sci. 2003 Jul 5;791(1-2):85-92.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • NeoLipid Camptosar

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul