Motexafin gadolinium

DB05428

small molecule investigational

Deskripsi

Motexafin gadolinium is studied in the treatment of cancer by Pharmacyclics. It may make tumor cells more sensitive to radiation therapy, improve tumor images using magnetic resonance imaging (MRI), and kill cancer cells. It belongs to the family of drugs called metalloporphyrin complexes. Also called gadolinium texaphyrin.

Struktur Molekul 2D

Berat 1148.4
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

43 Data
Porfimer sodium Motexafin gadolinium may increase the photosensitizing activities of Porfimer sodium.
Verteporfin Motexafin gadolinium may increase the photosensitizing activities of Verteporfin.
Tretinoin The risk or severity of adverse effects can be increased when Tretinoin is combined with Motexafin gadolinium.
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Motexafin gadolinium.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Motexafin gadolinium.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Motexafin gadolinium.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Motexafin gadolinium.
Padeliporfin Motexafin gadolinium may increase the photosensitizing activities of Padeliporfin.
Lidocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Quinisocaine.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Motexafin gadolinium.
Ambroxol The risk or severity of methemoglobinemia can be increased when Motexafin gadolinium is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Motexafin gadolinium is combined with Etrasimod.

Target Protein

Peroxiredoxin-5, mitochondrial PRDX5
Thioredoxin reductase 1, cytoplasmic TXNRD1
Thioredoxin reductase 2, mitochondrial TXNRD2
Ribonucleoside-diphosphate reductase subunit M2 RRM2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15627019
    Evens AM: Motexafin gadolinium: a redox-active tumor selective agent for the treatment of cancer. Curr Opin Oncol. 2004 Nov;16(6):576-80.
  • PMID: 17555388
    Forouzannia A, Richards GM, Khuntia D, Mehta MP: Motexafin gadolinium: a novel radiosensitizer for brain tumors. Expert Rev Anticancer Ther. 2007 Jun;7(6):785-94.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Xcytrin

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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