Canertinib

DB05424

small molecule investigational

Deskripsi

Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squamous cell carcinoma in vitro and in vivo. Canertinib treatment significantly affects tumour metabolism, proliferation and hypoxia as determined by PET.

Struktur Molekul 2D

Berat 485.938
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

66 Data
Acetaminophen The serum concentration of Acetaminophen can be increased when it is combined with Canertinib.
Propacetamol The serum concentration of Propacetamol can be increased when it is combined with Canertinib.
Salmon calcitonin The therapeutic efficacy of Salmon calcitonin can be decreased when used in combination with Canertinib.
Thyrotropin alfa The therapeutic efficacy of Thyrotropin alfa can be decreased when used in combination with Canertinib.
Follitropin The therapeutic efficacy of Follitropin can be decreased when used in combination with Canertinib.
Liothyronine The therapeutic efficacy of Liothyronine can be decreased when used in combination with Canertinib.
Carbimazole The therapeutic efficacy of Carbimazole can be decreased when used in combination with Canertinib.
Levothyroxine The therapeutic efficacy of Levothyroxine can be decreased when used in combination with Canertinib.
Propylthiouracil The therapeutic efficacy of Propylthiouracil can be decreased when used in combination with Canertinib.
Methimazole The therapeutic efficacy of Methimazole can be decreased when used in combination with Canertinib.
Liotrix The therapeutic efficacy of Liotrix can be decreased when used in combination with Canertinib.
3,5-Diiodotyrosine The therapeutic efficacy of 3,5-Diiodotyrosine can be decreased when used in combination with Canertinib.
Tiratricol The therapeutic efficacy of Tiratricol can be decreased when used in combination with Canertinib.
Parathyroid hormone The therapeutic efficacy of Parathyroid hormone can be decreased when used in combination with Canertinib.
Teriparatide The therapeutic efficacy of Teriparatide can be decreased when used in combination with Canertinib.
Potassium Iodide The therapeutic efficacy of Potassium Iodide can be decreased when used in combination with Canertinib.
Dibromotyrosine The therapeutic efficacy of Dibromotyrosine can be decreased when used in combination with Canertinib.
Thyroid, porcine The therapeutic efficacy of Thyroid, porcine can be decreased when used in combination with Canertinib.
Potassium perchlorate The therapeutic efficacy of Potassium perchlorate can be decreased when used in combination with Canertinib.
Protirelin The therapeutic efficacy of Protirelin can be decreased when used in combination with Canertinib.
3,5-diiodothyropropionic acid The therapeutic efficacy of 3,5-diiodothyropropionic acid can be decreased when used in combination with Canertinib.
Methylthiouracil The therapeutic efficacy of Methylthiouracil can be decreased when used in combination with Canertinib.
Elcatonin The therapeutic efficacy of Elcatonin can be decreased when used in combination with Canertinib.
Benzylthiouracil The therapeutic efficacy of Benzylthiouracil can be decreased when used in combination with Canertinib.
Thyrotropin The therapeutic efficacy of Thyrotropin can be decreased when used in combination with Canertinib.
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Canertinib.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Canertinib.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Canertinib.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Canertinib.
Lidocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Quinisocaine.
Voriconazole The serum concentration of Canertinib can be increased when it is combined with Voriconazole.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Canertinib.
Ambroxol The risk or severity of methemoglobinemia can be increased when Canertinib is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Canertinib is combined with Etrasimod.
Palopegteriparatide The therapeutic efficacy of Palopegteriparatide can be decreased when used in combination with Canertinib.

Target Protein

Receptor tyrosine-protein kinase erbB-2 ERBB2
RAC-alpha serine/threonine-protein kinase AKT1
Receptor tyrosine-protein kinase erbB-4 ERBB4
Epidermal growth factor receptor EGFR

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16899614
    Simon GR, Garrett CR, Olson SC, Langevin M, Eiseman IA, Mahany JJ, Williams CC, Lush R, Daud A, Munster P, Chiappori A, Fishman M, Bepler G, Lenehan PF, Sullivan DM: Increased bioavailability of intravenous versus oral CI-1033, a pan erbB tyrosine kinase inhibitor: results of a phase I pharmacokinetic study. Clin Cancer Res. 2006 Aug 1;12(15):4645-51.
  • PMID: 17405897
    Sequist LV: Second-generation epidermal growth factor receptor tyrosine kinase inhibitors in non-small cell lung cancer. Oncologist. 2007 Mar;12(3):325-30.

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Sekuens Gen/Protein (FASTA)

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