Pimagedine

DB05383

small molecule investigational

Deskripsi

Pimagedine has been developed by Synvista Therapeutics, Inc for the treatment of diabetic kidney disease. It is an advanced glycation end product inhibitor which manages diabetic nephropathy, either alone or in combination with other therapies. It is beneficial in treating patients with diabetic nephropathy.

Struktur Molekul 2D

Berat 74.0851
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

27 Data
Tipiracil The excretion of Tipiracil can be decreased when combined with Pimagedine.
Varenicline The excretion of Varenicline can be decreased when combined with Pimagedine.
Prazosin The serum concentration of Prazosin can be increased when it is combined with Pimagedine.
Solriamfetol The serum concentration of Solriamfetol can be increased when it is combined with Pimagedine.
Ranitidine The serum concentration of Ranitidine can be increased when it is combined with Pimagedine.
Linagliptin The serum concentration of Linagliptin can be increased when it is combined with Pimagedine.
Choline salicylate The serum concentration of Choline salicylate can be increased when it is combined with Pimagedine.
Choline The serum concentration of Choline can be increased when it is combined with Pimagedine.
Metformin The serum concentration of Metformin can be increased when it is combined with Pimagedine.
Norepinephrine The serum concentration of Norepinephrine can be increased when it is combined with Pimagedine.
Reserpine The serum concentration of Reserpine can be increased when it is combined with Pimagedine.
Pramipexole The serum concentration of Pramipexole can be increased when it is combined with Pimagedine.
Epinephrine The serum concentration of Epinephrine can be increased when it is combined with Pimagedine.
Lamivudine The serum concentration of Lamivudine can be increased when it is combined with Pimagedine.
Amantadine The serum concentration of Amantadine can be increased when it is combined with Pimagedine.
Dopamine The serum concentration of Dopamine can be increased when it is combined with Pimagedine.
Memantine The serum concentration of Memantine can be increased when it is combined with Pimagedine.
Histamine The serum concentration of Histamine can be increased when it is combined with Pimagedine.
Agmatine The serum concentration of Agmatine can be increased when it is combined with Pimagedine.
Nafamostat The serum concentration of Nafamostat can be increased when it is combined with Pimagedine.
Dofetilide The serum concentration of Dofetilide can be increased when it is combined with Pimagedine.
Cisplatin The serum concentration of Cisplatin can be increased when it is combined with Pimagedine.
Oxaliplatin The serum concentration of Oxaliplatin can be increased when it is combined with Pimagedine.
Procainamide The serum concentration of Procainamide can be increased when it is combined with Pimagedine.
Dalfampridine The serum concentration of Dalfampridine can be increased when it is combined with Pimagedine.
Clofarabine The serum concentration of Clofarabine can be increased when it is combined with Pimagedine.
Gentamicin The serum concentration of Gentamicin can be increased when it is combined with Pimagedine.

Target Protein

Nitric oxide synthase, inducible NOS2
C-C chemokine receptor type 2 CCR2
Diamine oxidase [copper-containing] AOC1
Aldo-keto reductase family 1 member B1 AKR1B1
Metalloproteinase inhibitor 3 TIMP3

Referensi & Sumber

Artikel (PubMed)
  • PMID: 11922864
    Abdel-Rahman E, Bolton WK: Pimagedine: a novel therapy for diabetic nephropathy. Expert Opin Investig Drugs. 2002 Apr;11(4):565-74.
  • PMID: 1727735
    Edelstein D, Brownlee M: Mechanistic studies of advanced glycosylation end product inhibition by aminoguanidine. Diabetes. 1992 Jan;41(1):26-9.

Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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