Peringatan Keamanan

LD50=807 mg/kg (mouse, oral). Side effects can lead to hypertension, hypotension, headache, dizziness, nervousness and tachycardia. Large overdoses can lead to seizures.

Histamine

DB05381

small molecule approved investigational

Deskripsi

A depressor amine derived by enzymatic decarboxylation of histidine. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscle, a vasodilator, and also a centrally acting neurotransmitter.

Struktur Molekul 2D

Berat 111.1451
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Readily absorbed after parenteral administration.

Metabolisme

Primarily hepatic. Histamine is rapidly metabolized by methylation and oxidation. Methylation involves ring methylation and catalyzation by the enzyme histamine-N-methyltransferase, producing N-methylhistamine, which is mostly converted to N-methyl imidazole acetic acid. 2 to 3% excreted as free histamine, 4 to 8% as N-methylhistamine, 42 to 47% as N-methyl imidazole acetic acid, 9 to 11% as imidazole acetic acid, and 16 to 23% as imidazole acetic acid riboside.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

107 Data
Bupropion The excretion of Histamine can be decreased when combined with Bupropion.
Tipiracil The excretion of Tipiracil can be decreased when combined with Histamine.
Varenicline The excretion of Varenicline can be decreased when combined with Histamine.
Prazosin The serum concentration of Prazosin can be increased when it is combined with Histamine.
Solriamfetol The serum concentration of Solriamfetol can be increased when it is combined with Histamine.
Choline The serum concentration of Histamine can be increased when it is combined with Choline.
Thiamine The serum concentration of Histamine can be increased when it is combined with Thiamine.
Nicotine The serum concentration of Histamine can be increased when it is combined with Nicotine.
Ranolazine The serum concentration of Histamine can be increased when it is combined with Ranolazine.
Metoprolol The serum concentration of Histamine can be increased when it is combined with Metoprolol.
Disopyramide The serum concentration of Histamine can be increased when it is combined with Disopyramide.
Metformin The serum concentration of Histamine can be increased when it is combined with Metformin.
Aminohippuric acid The serum concentration of Histamine can be increased when it is combined with Aminohippuric acid.
Grepafloxacin The serum concentration of Histamine can be increased when it is combined with Grepafloxacin.
Norepinephrine The serum concentration of Histamine can be increased when it is combined with Norepinephrine.
Progesterone The serum concentration of Histamine can be increased when it is combined with Progesterone.
Imipramine The serum concentration of Histamine can be increased when it is combined with Imipramine.
Quinine The serum concentration of Histamine can be increased when it is combined with Quinine.
Cimetidine The serum concentration of Histamine can be increased when it is combined with Cimetidine.
Guanidine The serum concentration of Histamine can be increased when it is combined with Guanidine.
Lamotrigine The serum concentration of Histamine can be increased when it is combined with Lamotrigine.
Propranolol The serum concentration of Histamine can be increased when it is combined with Propranolol.
Amiloride The serum concentration of Histamine can be increased when it is combined with Amiloride.
Imatinib The serum concentration of Histamine can be increased when it is combined with Imatinib.
Epinephrine The serum concentration of Histamine can be increased when it is combined with Epinephrine.
Flurazepam The serum concentration of Histamine can be increased when it is combined with Flurazepam.
Clopidogrel The serum concentration of Histamine can be increased when it is combined with Clopidogrel.
Estradiol The serum concentration of Histamine can be increased when it is combined with Estradiol.
Ranitidine The serum concentration of Histamine can be increased when it is combined with Ranitidine.
Quinidine The serum concentration of Histamine can be increased when it is combined with Quinidine.
Phenformin The serum concentration of Histamine can be increased when it is combined with Phenformin.
Amantadine The serum concentration of Histamine can be increased when it is combined with Amantadine.
Dinoprostone The serum concentration of Histamine can be increased when it is combined with Dinoprostone.
Phenoxybenzamine The serum concentration of Histamine can be increased when it is combined with Phenoxybenzamine.
Famotidine The serum concentration of Histamine can be increased when it is combined with Famotidine.
Salmeterol The serum concentration of Histamine can be increased when it is combined with Salmeterol.
Dopamine The serum concentration of Histamine can be increased when it is combined with Dopamine.
Probenecid The serum concentration of Histamine can be increased when it is combined with Probenecid.
Diphenhydramine The serum concentration of Histamine can be increased when it is combined with Diphenhydramine.
Quinacrine The serum concentration of Histamine can be increased when it is combined with Quinacrine.
Chlorpheniramine The serum concentration of Histamine can be increased when it is combined with Chlorpheniramine.
Amiodarone The serum concentration of Histamine can be increased when it is combined with Amiodarone.
Desipramine The serum concentration of Histamine can be increased when it is combined with Desipramine.
Oxprenolol The serum concentration of Histamine can be increased when it is combined with Oxprenolol.
Dronedarone The serum concentration of Histamine can be increased when it is combined with Dronedarone.
Vandetanib The serum concentration of Histamine can be increased when it is combined with Vandetanib.
Reserpine The serum concentration of Reserpine can be increased when it is combined with Histamine.
Pramipexole The serum concentration of Pramipexole can be increased when it is combined with Histamine.
Lamivudine The serum concentration of Lamivudine can be increased when it is combined with Histamine.
Memantine The serum concentration of Memantine can be increased when it is combined with Histamine.
Agmatine The serum concentration of Agmatine can be increased when it is combined with Histamine.
Linagliptin The serum concentration of Linagliptin can be increased when it is combined with Histamine.
Nafamostat The serum concentration of Nafamostat can be increased when it is combined with Histamine.
Choline salicylate The serum concentration of Choline salicylate can be increased when it is combined with Histamine.
Pimagedine The serum concentration of Histamine can be increased when it is combined with Pimagedine.
Tafenoquine The serum concentration of Histamine can be increased when it is combined with Tafenoquine.
Crizotinib The serum concentration of Histamine can be increased when it is combined with Crizotinib.
Dolutegravir The serum concentration of Histamine can be increased when it is combined with Dolutegravir.
Lenvatinib The serum concentration of Histamine can be increased when it is combined with Lenvatinib.
Dexchlorpheniramine maleate The serum concentration of Histamine can be increased when it is combined with Dexchlorpheniramine maleate.
Isavuconazole The serum concentration of Histamine can be increased when it is combined with Isavuconazole.
Tucatinib The serum concentration of Histamine can be increased when it is combined with Tucatinib.
Apalutamide The serum concentration of Histamine can be increased when it is combined with Apalutamide.
Erdafitinib The serum concentration of Histamine can be increased when it is combined with Erdafitinib.
Enasidenib The serum concentration of Histamine can be increased when it is combined with Enasidenib.
Estradiol acetate The serum concentration of Histamine can be increased when it is combined with Estradiol acetate.
Estradiol benzoate The serum concentration of Histamine can be increased when it is combined with Estradiol benzoate.
Estradiol cypionate The serum concentration of Histamine can be increased when it is combined with Estradiol cypionate.
Estradiol dienanthate The serum concentration of Histamine can be increased when it is combined with Estradiol dienanthate.
Estradiol valerate The serum concentration of Histamine can be increased when it is combined with Estradiol valerate.
Methylene blue The serum concentration of Histamine can be increased when it is combined with Methylene blue.
Trilaciclib The serum concentration of Histamine can be increased when it is combined with Trilaciclib.
Codeine The risk or severity of adverse effects can be increased when Codeine is combined with Histamine.
Doxazosin The risk or severity of adverse effects can be increased when Doxazosin is combined with Histamine.
Rocuronium The risk or severity of adverse effects can be increased when Rocuronium is combined with Histamine.
Acyclovir The risk or severity of adverse effects can be increased when Acyclovir is combined with Histamine.
Ganciclovir The risk or severity of adverse effects can be increased when Ganciclovir is combined with Histamine.
Pancuronium The risk or severity of adverse effects can be increased when Pancuronium is combined with Histamine.
Palbociclib The risk or severity of adverse effects can be increased when Palbociclib is combined with Histamine.
Dacomitinib The risk or severity of adverse effects can be increased when Dacomitinib is combined with Histamine.
Gilteritinib The risk or severity of adverse effects can be increased when Gilteritinib is combined with Histamine.
Nelfinavir The risk or severity of adverse effects can be increased when Nelfinavir is combined with Histamine.
Indinavir The risk or severity of adverse effects can be increased when Indinavir is combined with Histamine.
Nevirapine The risk or severity of adverse effects can be increased when Nevirapine is combined with Histamine.
Efavirenz The risk or severity of adverse effects can be increased when Efavirenz is combined with Histamine.
Verapamil The risk or severity of adverse effects can be increased when Verapamil is combined with Histamine.
Saquinavir The risk or severity of adverse effects can be increased when Saquinavir is combined with Histamine.
Pitolisant The risk or severity of adverse effects can be increased when Pitolisant is combined with Histamine.
Formoterol The risk or severity of adverse effects can be increased when Formoterol is combined with Histamine.
Guanfacine The risk or severity of adverse effects can be increased when Guanfacine is combined with Histamine.
Cisplatin The serum concentration of Cisplatin can be increased when it is combined with Histamine.
Procainamide The serum concentration of Procainamide can be increased when it is combined with Histamine.
Oxaliplatin The serum concentration of Oxaliplatin can be increased when it is combined with Histamine.
Dalfampridine The serum concentration of Dalfampridine can be increased when it is combined with Histamine.
Dofetilide The serum concentration of Dofetilide can be increased when it is combined with Histamine.
Clofarabine The serum concentration of Clofarabine can be increased when it is combined with Histamine.
Gentamicin The serum concentration of Gentamicin can be increased when it is combined with Histamine.
Pentagastrin The serum concentration of Histamine can be increased when it is combined with Pentagastrin.
Fexinidazole The serum concentration of Histamine can be increased when it is combined with Fexinidazole.
Levoketoconazole The serum concentration of Histamine can be increased when it is combined with Levoketoconazole.

Target Protein

Histamine H1 receptor HRH1
Histamine H2 receptor HRH2
Histamine H3 receptor HRH3
Histamine H4 receptor HRH4
Synaptic vesicular amine transporter SLC18A2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 12092744
    Middleton M, Sarno M, Agarwala SS, Glaspy J, Laurent A, McMasters K, Naredi P, O'Day S, Whitman E, Danson S, Cosford R, Gehlsen K: Pharmacokinetics of histamine dihydrochloride in healthy volunteers and cancer patients: implications for combined immunotherapy with interleukin-2. J Clin Pharmacol. 2002 Jul;42(7):774-81.
  • PMID: 26252585
    Silberstein SD: Preventive Migraine Treatment. Continuum (Minneap Minn). 2015 Aug;21(4 Headache):973-89. doi: 10.1212/CON.0000000000000199.

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