Fibrinolysin

DB05254

biotech investigational

Deskripsi

Fibrinolysin consists of two polypeptide chains, one light and one heavy, linked by a disulfide bond. The light chain has a molecular weight of approximately 27,000 Da and contains the active center of Fibrinolysin; the heavy chain has a molecular weight of approximately 57,000 Da. Fibrinolysin is used as a local healing ointment when combined together with the enzyme deoxyribonuclease I (extracted from bovine pancreas). Fibrinolysin and deoxyribonuclease both act as lytic enzymes. The combination is available as ointment containing 1 BU (Biological Unit) Fibrinolysin and 666 BUs desoxyribonuclease per gram. The ointment is marketed by Pfizer under the brand name Fibrolan in a variety of countries (e.g. Switzerland). It is currently not approved in the USA.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Almost completely inactivated after 24 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

local inactivation

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

10 Data
Citalopram The risk or severity of bleeding can be increased when Fibrinolysin is combined with Citalopram.
Desvenlafaxine The risk or severity of adverse effects can be increased when Desvenlafaxine is combined with Fibrinolysin.
Levomilnacipran The risk or severity of bleeding can be increased when Fibrinolysin is combined with Levomilnacipran.
Venlafaxine The risk or severity of bleeding can be increased when Fibrinolysin is combined with Venlafaxine.
Oxaliplatin The risk or severity of hemorrhage can be increased when Oxaliplatin is combined with Fibrinolysin.
Padeliporfin The risk or severity of bleeding can be increased when Fibrinolysin is combined with Padeliporfin.
Soybean oil The therapeutic efficacy of Fibrinolysin can be decreased when used in combination with Soybean oil.
Olive oil The therapeutic efficacy of Fibrinolysin can be decreased when used in combination with Olive oil.
Inotersen The risk or severity of thrombocytopenia can be increased when Inotersen is combined with Fibrinolysin.
Iloprost Iloprost may increase the anticoagulant activities of Fibrinolysin.

Target Protein

Plasminogen activator inhibitor 1 SERPINE1
Urokinase-type plasminogen activator PLAU

Referensi & Sumber

Synthesis reference: U.S. Patent 2,624,691; U.S. Patent 3,136,703; U.S. Patent 3,234,106.
Artikel (PubMed)
  • PMID: 6226244
    Birk Y, Khalef S, Jibson MD: Purification and properties of protease F, a bacterial enzyme with chymotrypsin and elastase specificities. Arch Biochem Biophys. 1983 Sep;225(2):451-7.

Contoh Produk & Brand

Produk: 0 • International brands: 2
International Brands
  • Elase — Pfizer
  • Fibrolan — Pfizer

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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