Peringatan Keamanan

Acute overdoses may produce nausea, vomiting, and CNS depression including coma with respiratory depression. Levels greater than 40 µg/mL have caused toxicity and coma has been seen at levels of 150 µg/mL.

Methsuximide

DB05246

small molecule approved

Deskripsi

Mesuximide (or methsuximide) is an anticonvulsant medication. It is sold by Pfizer under the name Petinutin.

Struktur Molekul 2D

Berat 203.2371
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 1.4-2.6 hours for mesuximide and 28-38 hours for the active metabolite.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food.

Interaksi Obat

1640 Data
Ceritinib Methsuximide may increase the bradycardic activities of Ceritinib.
Ivabradine Methsuximide may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of Methsuximide.
Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Methsuximide.
Buprenorphine Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Hydrocodone Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Magnesium sulfate The therapeutic efficacy of Methsuximide can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Methsuximide may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Mirtazapine Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Orphenadrine Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Pramipexole Methsuximide may increase the sedative activities of Pramipexole.
Ropinirole Methsuximide may increase the sedative activities of Ropinirole.
Rotigotine Methsuximide may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Methsuximide.
Sodium oxybate Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Thalidomide Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Dabrafenib The serum concentration of Methsuximide can be decreased when it is combined with Dabrafenib.
Luliconazole The serum concentration of Methsuximide can be increased when it is combined with Luliconazole.
Mefloquine The therapeutic efficacy of Methsuximide can be decreased when used in combination with Mefloquine.
Mianserin The therapeutic efficacy of Methsuximide can be decreased when used in combination with Mianserin.
Orlistat Orlistat can cause a decrease in the absorption of Methsuximide resulting in a reduced serum concentration and potentially a decrease in efficacy.
Topotecan Methsuximide may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Cimetidine The serum concentration of Methsuximide can be increased when it is combined with Cimetidine.
Clopidogrel The therapeutic efficacy of Clopidogrel can be decreased when used in combination with Methsuximide.
Efavirenz The serum concentration of Methsuximide can be decreased when it is combined with Efavirenz.
Melatonin The therapeutic efficacy of Methsuximide can be decreased when used in combination with Melatonin.
Nafcillin The therapeutic efficacy of Methsuximide can be decreased when used in combination with Nafcillin.
Nitroprusside Methsuximide may increase the hypotensive activities of Nitroprusside.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Methsuximide.
Dantrolene The risk or severity of hyperkalemia can be increased when Dantrolene is combined with Methsuximide.
Lithium citrate The risk or severity of adverse effects can be increased when Methsuximide is combined with Lithium citrate.
Lithium carbonate The risk or severity of adverse effects can be increased when Methsuximide is combined with Lithium carbonate.
Lithium hydroxide The risk or severity of adverse effects can be increased when Methsuximide is combined with Lithium hydroxide.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Methsuximide.
Boceprevir The serum concentration of Methsuximide can be increased when it is combined with Boceprevir.
Ethanol Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Methsuximide may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Methsuximide.
Duloxetine The risk or severity of adverse effects can be increased when Methsuximide is combined with Duloxetine.
Paroxetine The risk or severity of adverse effects can be increased when Methsuximide is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Methsuximide is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Methsuximide is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Methsuximide is combined with Nefazodone.
Zimelidine The risk or severity of adverse effects can be increased when Methsuximide is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Methsuximide is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Methsuximide is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Methsuximide is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Methsuximide is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Methsuximide is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Methsuximide is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Methsuximide is combined with Alaproclate.
Escitalopram The risk or severity of adverse effects can be increased when Methsuximide is combined with Escitalopram.
Lumacaftor The serum concentration of Methsuximide can be decreased when it is combined with Lumacaftor.
Mexiletine Mexiletine may increase the arrhythmogenic activities of Methsuximide.
Tocainide Tocainide may increase the arrhythmogenic activities of Methsuximide.
Aprindine Aprindine may increase the arrhythmogenic activities of Methsuximide.
Carteolol Methsuximide may increase the arrhythmogenic activities of Carteolol.
Metipranolol Methsuximide may increase the arrhythmogenic activities of Metipranolol.
Xylometazoline Methsuximide may increase the arrhythmogenic activities of Xylometazoline.
Sparteine Methsuximide may increase the arrhythmogenic activities of Sparteine.
Fasudil Methsuximide may increase the arrhythmogenic activities of Fasudil.
Spiradoline Methsuximide may increase the arrhythmogenic activities of Spiradoline.
Tiracizine Methsuximide may increase the arrhythmogenic activities of Tiracizine.
Ethacizine Methsuximide may increase the arrhythmogenic activities of Ethacizine.
Hydroquinine Methsuximide may increase the arrhythmogenic activities of Hydroquinine.
Bioallethrin Methsuximide may increase the arrhythmogenic activities of Bioallethrin.
Fosfructose Methsuximide may increase the arrhythmogenic activities of Fosfructose.
Hydroquinidine Methsuximide may increase the arrhythmogenic activities of Hydroquinidine.
SOR-C13 Methsuximide may increase the arrhythmogenic activities of SOR-C13.
Digoxin Digoxin may increase the arrhythmogenic activities of Methsuximide.
Acetyldigitoxin Acetyldigitoxin may increase the arrhythmogenic activities of Methsuximide.
Deslanoside Deslanoside may increase the arrhythmogenic activities of Methsuximide.
Digitoxin Digitoxin may increase the arrhythmogenic activities of Methsuximide.
Cymarin Methsuximide may increase the arrhythmogenic activities of Cymarin.
Metildigoxin Methsuximide may increase the arrhythmogenic activities of Metildigoxin.
Acetyldigoxin Methsuximide may increase the arrhythmogenic activities of Acetyldigoxin.
Hyoscyamine Hyoscyamine may increase the arrhythmogenic activities of Methsuximide.
Nicardipine Nicardipine may increase the arrhythmogenic activities of Methsuximide.
Verapamil Verapamil may increase the arrhythmogenic activities of Methsuximide.
Niguldipine Methsuximide may increase the arrhythmogenic activities of Niguldipine.
Diltiazem Diltiazem may increase the arrhythmogenic activities of Methsuximide.
Nimodipine Nimodipine may increase the arrhythmogenic activities of Methsuximide.
Cinnarizine Cinnarizine may increase the arrhythmogenic activities of Methsuximide.
Atropine Atropine may increase the arrhythmogenic activities of Methsuximide.
Adenosine Adenosine may increase the arrhythmogenic activities of Methsuximide.
Loperamide Loperamide may increase the arrhythmogenic activities of Methsuximide.
Levosimendan Levosimendan may increase the arrhythmogenic activities of Methsuximide.
Nifedipine Nifedipine may increase the arrhythmogenic activities of Methsuximide.
Flecainide Flecainide may increase the arrhythmogenic activities of Methsuximide.

Target Protein

Voltage-dependent T-type calcium channel subunit alpha-1G CACNA1G

Referensi & Sumber

Artikel (PubMed)
  • PMID: 8777552
    Hurst DL: Methsuximide therapy of juvenile myoclonic epilepsy. Seizure. 1996 Mar;5(1):47-50.
  • PMID: 10802770
    Besag FM, Berry DJ, Pool F: Methsuximide lowers lamotrigine blood levels: A pharmacokinetic antiepileptic drug interaction. Epilepsia. 2000 May;41(5):624-7.
  • PMID: 7640152
    Wright JD, Helsby NA, Ward SA: The role of S-mephenytoin hydroxylase (CYP2C19) in the metabolism of the antimalarial biguanides. Br J Clin Pharmacol. 1995 Apr;39(4):441-4.

Contoh Produk & Brand

Produk: 5 • International brands: 1
Produk
  • Celontin
    Capsule • 300 mg/1 • Oral • US • Approved
  • Celontin
    Capsule • 300 mg/1 • Oral • US • Approved
  • Celontin
    Capsule • 150 mg/1 • Oral • US • Approved
  • Celontin Cap 300mg
    Capsule • 300 mg • Oral • Canada • Approved
  • Methsuximide
    Capsule • 300 mg/1 • Oral • US • Generic • Approved
International Brands
  • Petinutin

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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