Afelimomab

DB04956

biotech investigational

Deskripsi

Afelimomab (also known as Fab 2 or MAK 195F) is an anti-TNF-? monoclonal antibody. Administration of 195F reduces the concentration of interleukin-6 in patients with sepsis.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 44.7 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1333 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Afelimomab.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Afelimomab.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Afelimomab.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Afelimomab.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Afelimomab.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Afelimomab.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Afelimomab.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Afelimomab.
Aldesleukin The risk or severity of adverse effects can be increased when Aldesleukin is combined with Afelimomab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Afelimomab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Afelimomab.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Afelimomab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Afelimomab.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Afelimomab.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Afelimomab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Afelimomab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Afelimomab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Afelimomab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Afelimomab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Afelimomab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Afelimomab.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Afelimomab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Afelimomab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Afelimomab.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Afelimomab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Afelimomab.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Afelimomab.
Cladribine Afelimomab may increase the immunosuppressive activities of Cladribine.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Afelimomab.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Afelimomab.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Afelimomab.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Afelimomab.
Mitomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Afelimomab.
Floxuridine The risk or severity of adverse effects can be increased when Floxuridine is combined with Afelimomab.
Tioguanine The risk or severity of adverse effects can be increased when Tioguanine is combined with Afelimomab.
Dexrazoxane The risk or severity of adverse effects can be increased when Dexrazoxane is combined with Afelimomab.
Streptozocin The risk or severity of adverse effects can be increased when Streptozocin is combined with Afelimomab.
Trifluridine The risk or severity of adverse effects can be increased when Trifluridine is combined with Afelimomab.
Gemcitabine The risk or severity of adverse effects can be increased when Gemcitabine is combined with Afelimomab.
Epirubicin The risk or severity of adverse effects can be increased when Epirubicin is combined with Afelimomab.
Chloramphenicol The risk or severity of adverse effects can be increased when Chloramphenicol is combined with Afelimomab.
Lenalidomide The risk or severity of adverse effects can be increased when Lenalidomide is combined with Afelimomab.
Altretamine The risk or severity of adverse effects can be increased when Altretamine is combined with Afelimomab.
Cisplatin The risk or severity of adverse effects can be increased when Cisplatin is combined with Afelimomab.
Oxaliplatin The risk or severity of adverse effects can be increased when Oxaliplatin is combined with Afelimomab.
Propylthiouracil The risk or severity of adverse effects can be increased when Propylthiouracil is combined with Afelimomab.
Pentostatin The risk or severity of adverse effects can be increased when Pentostatin is combined with Afelimomab.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Afelimomab.
Clofarabine The risk or severity of adverse effects can be increased when Clofarabine is combined with Afelimomab.
Methimazole The risk or severity of adverse effects can be increased when Methimazole is combined with Afelimomab.
Sulfasalazine The risk or severity of adverse effects can be increased when Sulfasalazine is combined with Afelimomab.
Temozolomide The risk or severity of adverse effects can be increased when Temozolomide is combined with Afelimomab.
Penicillamine The risk or severity of adverse effects can be increased when Penicillamine is combined with Afelimomab.
Mechlorethamine The risk or severity of adverse effects can be increased when Mechlorethamine is combined with Afelimomab.
Azacitidine The risk or severity of adverse effects can be increased when Azacitidine is combined with Afelimomab.
Carboplatin The risk or severity of adverse effects can be increased when Carboplatin is combined with Afelimomab.
Dactinomycin The risk or severity of adverse effects can be increased when Dactinomycin is combined with Afelimomab.
Hydroxyurea The risk or severity of adverse effects can be increased when Hydroxyurea is combined with Afelimomab.
Mycophenolic acid The risk or severity of adverse effects can be increased when Mycophenolic acid is combined with Afelimomab.
Topotecan The risk or severity of adverse effects can be increased when Topotecan is combined with Afelimomab.
Mercaptopurine The risk or severity of adverse effects can be increased when Mercaptopurine is combined with Afelimomab.
Melphalan The risk or severity of adverse effects can be increased when Melphalan is combined with Afelimomab.
Fludarabine The risk or severity of adverse effects can be increased when Fludarabine is combined with Afelimomab.
Flucytosine The risk or severity of adverse effects can be increased when Flucytosine is combined with Afelimomab.
Procarbazine The risk or severity of adverse effects can be increased when Procarbazine is combined with Afelimomab.
Arsenic trioxide The risk or severity of adverse effects can be increased when Arsenic trioxide is combined with Afelimomab.
Mitoxantrone The risk or severity of adverse effects can be increased when Mitoxantrone is combined with Afelimomab.
Lomustine The risk or severity of adverse effects can be increased when Lomustine is combined with Afelimomab.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Afelimomab.
Decitabine The risk or severity of adverse effects can be increased when Decitabine is combined with Afelimomab.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Afelimomab.
Stepronin The risk or severity of adverse effects can be increased when Stepronin is combined with Afelimomab.
Castanospermine The risk or severity of adverse effects can be increased when Castanospermine is combined with Afelimomab.
Vorinostat The risk or severity of adverse effects can be increased when Vorinostat is combined with Afelimomab.
2-Methoxyethanol The risk or severity of adverse effects can be increased when 2-Methoxyethanol is combined with Afelimomab.
Brequinar The risk or severity of adverse effects can be increased when Brequinar is combined with Afelimomab.
Interferon alfa The risk or severity of adverse effects can be increased when Afelimomab is combined with Interferon alfa.
Glatiramer The risk or severity of adverse effects can be increased when Afelimomab is combined with Glatiramer.
Briakinumab The risk or severity of adverse effects can be increased when Afelimomab is combined with Briakinumab.
Human interferon omega-1 The risk or severity of adverse effects can be increased when Afelimomab is combined with Human interferon omega-1.
Mepolizumab The risk or severity of adverse effects can be increased when Afelimomab is combined with Mepolizumab.
Abetimus The risk or severity of adverse effects can be increased when Afelimomab is combined with Abetimus.
Golimumab The risk or severity of adverse effects can be increased when Afelimomab is combined with Golimumab.
Belatacept The risk or severity of adverse effects can be increased when Afelimomab is combined with Belatacept.
Pralatrexate The risk or severity of adverse effects can be increased when Afelimomab is combined with Pralatrexate.
Wortmannin The risk or severity of adverse effects can be increased when Afelimomab is combined with Wortmannin.
Eribulin The risk or severity of adverse effects can be increased when Afelimomab is combined with Eribulin.
Belimumab The risk or severity of adverse effects can be increased when Afelimomab is combined with Belimumab.
Teriflunomide The risk or severity of adverse effects can be increased when Afelimomab is combined with Teriflunomide.
Carfilzomib The risk or severity of adverse effects can be increased when Afelimomab is combined with Carfilzomib.
Dimethyl fumarate The risk or severity of adverse effects can be increased when Afelimomab is combined with Dimethyl fumarate.
Obinutuzumab The risk or severity of adverse effects can be increased when Afelimomab is combined with Obinutuzumab.
Secukinumab The risk or severity of adverse effects can be increased when Afelimomab is combined with Secukinumab.
Siltuximab The risk or severity of adverse effects can be increased when Afelimomab is combined with Siltuximab.
Blinatumomab The risk or severity of adverse effects can be increased when Afelimomab is combined with Blinatumomab.
Dinutuximab The risk or severity of adverse effects can be increased when Afelimomab is combined with Dinutuximab.
Tixocortol The risk or severity of adverse effects can be increased when Afelimomab is combined with Tixocortol.
Peginterferon beta-1a The risk or severity of adverse effects can be increased when Afelimomab is combined with Peginterferon beta-1a.
Antilymphocyte immunoglobulin (horse) The risk or severity of adverse effects can be increased when Afelimomab is combined with Antilymphocyte immunoglobulin (horse).
Tepoxalin The risk or severity of adverse effects can be increased when Afelimomab is combined with Tepoxalin.

Target Protein

Tumor necrosis factor TNF

Referensi & Sumber

Artikel (PubMed)
  • PMID: 10829362
    Vincent JL: Afelimomab. Int J Clin Pract. 2000 Apr;54(3):190-3.
  • PMID: 11534565
    Gallagher J, Fisher C, Sherman B, Munger M, Meyers B, Ellison T, Fischkoff S, Barchuk WT, Teoh L, Velagapudi R: A multicenter, open-label, prospective, randomized, dose-ranging pharmacokinetic study of the anti-TNF-alpha antibody afelimomab in patients with sepsis syndrome. Intensive Care Med. 2001 Jul;27(7):1169-78.

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Sekuens Gen/Protein (FASTA)

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