Peringatan Keamanan

Most common adverse reactions associated with the use of lucinactant are endotracheal tube reflux, pallor, endotracheal tube obstruction, and need for
dose interruption.

Lucinactant

DB04897

biotech approved investigational

Deskripsi

Lucinactant is a new synthetic peptide-containing surfactant for intratracheal use. It contains sinapultide, a novel, hydrophobic, 21-amino acid peptide (leucine and lysine repeating units, KL4 peptide) designed to mimic human surfactant protein-B (SB-P). More specifically, it mimics the C-terminal amphipathic helical domain of this protein. It also consists of phospholipids (dipalmitoylphosphatidylcholine, DPPC and palmitoyloleoyl phosphatidylglycerol, POPG) and a fatty acid (palmitic acid). It is completely devoid of animal-derived components. FDA approved on March 6, 2012.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

141 Data
Ceritinib Lucinactant may increase the bradycardic activities of Ceritinib.
Ivabradine Lucinactant may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of Lucinactant.
Esmolol Esmolol may increase the bradycardic activities of Lucinactant.
Betaxolol Betaxolol may increase the bradycardic activities of Lucinactant.
Midodrine Midodrine may increase the bradycardic activities of Lucinactant.
Pregabalin Pregabalin may increase the bradycardic activities of Lucinactant.
Metoprolol Metoprolol may increase the bradycardic activities of Lucinactant.
Isradipine Isradipine may increase the bradycardic activities of Lucinactant.
Atenolol Atenolol may increase the bradycardic activities of Lucinactant.
Diltiazem Diltiazem may increase the bradycardic activities of Lucinactant.
Trimethadione Trimethadione may increase the bradycardic activities of Lucinactant.
Timolol Timolol may increase the bradycardic activities of Lucinactant.
Amlodipine Amlodipine may increase the bradycardic activities of Lucinactant.
Digoxin Digoxin may increase the bradycardic activities of Lucinactant.
Nimodipine Nimodipine may increase the bradycardic activities of Lucinactant.
Nisoldipine Nisoldipine may increase the bradycardic activities of Lucinactant.
Bendroflumethiazide Bendroflumethiazide may increase the bradycardic activities of Lucinactant.
Sotalol Sotalol may increase the bradycardic activities of Lucinactant.
Lercanidipine Lercanidipine may increase the bradycardic activities of Lucinactant.
Lamotrigine Lamotrigine may increase the bradycardic activities of Lucinactant.
Cinnarizine Cinnarizine may increase the bradycardic activities of Lucinactant.
Propranolol Propranolol may increase the bradycardic activities of Lucinactant.
Clonidine Clonidine may increase the bradycardic activities of Lucinactant.
Ethosuximide Ethosuximide may increase the bradycardic activities of Lucinactant.
Labetalol Labetalol may increase the bradycardic activities of Lucinactant.
Bisoprolol Bisoprolol may increase the bradycardic activities of Lucinactant.
Nicardipine Nicardipine may increase the bradycardic activities of Lucinactant.
Dexmedetomidine Dexmedetomidine may increase the bradycardic activities of Lucinactant.
Magnesium sulfate Magnesium sulfate may increase the bradycardic activities of Lucinactant.
Verapamil Verapamil may increase the bradycardic activities of Lucinactant.
Galantamine Galantamine may increase the bradycardic activities of Lucinactant.
Tizanidine Tizanidine may increase the bradycardic activities of Lucinactant.
Sufentanil Sufentanil may increase the bradycardic activities of Lucinactant.
Alfentanil Alfentanil may increase the bradycardic activities of Lucinactant.
Fentanyl Fentanyl may increase the bradycardic activities of Lucinactant.
Levomenthol Levomenthol may increase the bradycardic activities of Lucinactant.
Loperamide Loperamide may increase the bradycardic activities of Lucinactant.
Donepezil Donepezil may increase the bradycardic activities of Lucinactant.
Alprenolol Alprenolol may increase the bradycardic activities of Lucinactant.
Remifentanil Remifentanil may increase the bradycardic activities of Lucinactant.
Zonisamide Zonisamide may increase the bradycardic activities of Lucinactant.
Pindolol Pindolol may increase the bradycardic activities of Lucinactant.
Methyldopa Methyldopa may increase the bradycardic activities of Lucinactant.
Rivastigmine Rivastigmine may increase the bradycardic activities of Lucinactant.
Guanfacine Guanfacine may increase the bradycardic activities of Lucinactant.
Felodipine Felodipine may increase the bradycardic activities of Lucinactant.
Nitrendipine Nitrendipine may increase the bradycardic activities of Lucinactant.
Perhexiline Perhexiline may increase the bradycardic activities of Lucinactant.
Nifedipine Nifedipine may increase the bradycardic activities of Lucinactant.
Amiodarone Amiodarone may increase the bradycardic activities of Lucinactant.
Carvedilol Carvedilol may increase the bradycardic activities of Lucinactant.
Bretylium Bretylium may increase the bradycardic activities of Lucinactant.
Propafenone Propafenone may increase the bradycardic activities of Lucinactant.
Acebutolol Acebutolol may increase the bradycardic activities of Lucinactant.
Nadolol Nadolol may increase the bradycardic activities of Lucinactant.
Bepridil Bepridil may increase the bradycardic activities of Lucinactant.
Bevantolol Bevantolol may increase the bradycardic activities of Lucinactant.
Practolol Practolol may increase the bradycardic activities of Lucinactant.
Penbutolol Penbutolol may increase the bradycardic activities of Lucinactant.
Mibefradil Mibefradil may increase the bradycardic activities of Lucinactant.
Oxprenolol Oxprenolol may increase the bradycardic activities of Lucinactant.
Nimesulide Nimesulide may increase the bradycardic activities of Lucinactant.
Prenylamine Prenylamine may increase the bradycardic activities of Lucinactant.
Cyclandelate Cyclandelate may increase the bradycardic activities of Lucinactant.
Flunarizine Flunarizine may increase the bradycardic activities of Lucinactant.
Fluspirilene Fluspirilene may increase the bradycardic activities of Lucinactant.
Celiprolol Celiprolol may increase the bradycardic activities of Lucinactant.
Dronedarone Dronedarone may increase the bradycardic activities of Lucinactant.
Nebivolol Nebivolol may increase the bradycardic activities of Lucinactant.
Clevidipine Lucinactant may increase the bradycardic activities of Clevidipine.
Methsuximide Lucinactant may increase the bradycardic activities of Methsuximide.
Seletracetam Lucinactant may increase the bradycardic activities of Seletracetam.
Nylidrin Lucinactant may increase the bradycardic activities of Nylidrin.
Lacosamide The risk or severity of ventricular arrhythmias, bradycardia, and heart block can be increased when Lucinactant is combined with Lacosamide.
Calfactant Lucinactant may increase the bradycardic activities of Calfactant.
Dotarizine Lucinactant may increase the bradycardic activities of Dotarizine.
Pasireotide Lucinactant may increase the bradycardic activities of Pasireotide.
Nilvadipine Lucinactant may increase the bradycardic activities of Nilvadipine.
Bufuralol Lucinactant may increase the bradycardic activities of Bufuralol.
Beractant Lucinactant may increase the bradycardic activities of Beractant.
Lanreotide Lucinactant may increase the bradycardic activities of Lanreotide.
Tranilast Lucinactant may increase the bradycardic activities of Tranilast.
Bopindolol Lucinactant may increase the bradycardic activities of Bopindolol.
Bupranolol Lucinactant may increase the bradycardic activities of Bupranolol.
Agmatine Lucinactant may increase the bradycardic activities of Agmatine.
Crizotinib Crizotinib may increase the bradycardic activities of Lucinactant.
Fingolimod Lucinactant may increase the bradycardic activities of Fingolimod.
Tofacitinib Lucinactant may increase the bradycardic activities of Tofacitinib.
Regorafenib Lucinactant may increase the bradycardic activities of Regorafenib.
Indenolol Lucinactant may increase the bradycardic activities of Indenolol.
Fendiline Lucinactant may increase the bradycardic activities of Fendiline.
Eperisone Lucinactant may increase the bradycardic activities of Eperisone.
Trimebutine Lucinactant may increase the bradycardic activities of Trimebutine.
Pinaverium Lucinactant may increase the bradycardic activities of Pinaverium.
Poractant alfa Lucinactant may increase the bradycardic activities of Poractant alfa.
Arotinolol Lucinactant may increase the bradycardic activities of Arotinolol.
Tolfenamic acid Lucinactant may increase the bradycardic activities of Tolfenamic acid.
Barnidipine Lucinactant may increase the bradycardic activities of Barnidipine.
Aranidipine Lucinactant may increase the bradycardic activities of Aranidipine.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15805381
    Sinha SK, Lacaze-Masmonteil T, Valls i Soler A, Wiswell TE, Gadzinowski J, Hajdu J, Bernstein G, Sanchez-Luna M, Segal R, Schaber CJ, Massaro J, d'Agostino R: A multicenter, randomized, controlled trial of lucinactant versus poractant alfa among very premature infants at high risk for respiratory distress syndrome. Pediatrics. 2005 Apr;115(4):1030-8.
  • PMID: 17533176
    Moya F, Sinha S, Gadzinowski J, D'Agostino R, Segal R, Guardia C, Mazela J, Liu G: One-year follow-up of very preterm infants who received lucinactant for prevention of respiratory distress syndrome: results from 2 multicenter randomized, controlled trials. Pediatrics. 2007 Jun;119(6):e1361-70. Epub 2007 May 28.
  • PMID: 16740886
    Halliday HL, Speer CP: Lucinactant versus poractant-alpha in premature lambs. Pediatrics. 2006 Jun;117(6):2324-5; author reply 2325.
  • PMID: 16452346
    Gastiasoro-Cuesta E, Alvarez-Diaz FJ, Rey-Santano C, Arnaiz-Renedo A, Loureiro-Gonzalez B, Valls-i-Soler A: Acute and sustained effects of lucinactant versus poractant-alpha on pulmonary gas exchange and mechanics in premature lambs with respiratory distress syndrome. Pediatrics. 2006 Feb;117(2):295-303.
  • PMID: 15833063
    Donn SM: Lucinactant: a novel synthetic surfactant for the treatment of respiratory distress syndrome. Expert Opin Investig Drugs. 2005 Mar;14(3):329-34.
  • PMID: 15813666
    Moen MD, Perry CM, Wellington K: Lucinactant: in neonatal respiratory distress syndrome. Treat Respir Med. 2005;4(2):139-45; discussion 146-7.
  • PMID: 12802703
    Doyle I: Lucinactant (Discovery Laboratories). IDrugs. 2002 Jul;5(7):696-702.

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