Dapoxetine

DB04884

small molecule investigational

Deskripsi

Dapoxetine is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation. In a phase II proof-of-concept study conducted by PPD, dapoxetine demonstrated a statistically significant increase in ejaculatory latency when compared to placebo. Alza submitted a NDA to the FDA for dapoxetine for the treatment of premature ejaculation in December 2004. In October 2005, the company received a FDA Non-Approvable letter from the FDA, at which time they planned to work with regulators to address outstanding questions.

Struktur Molekul 2D

Berat 305.4134
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Initial half-life of 1-2 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1473 Data
Lomitapide The metabolism of Lomitapide can be decreased when combined with Dapoxetine.
Cyproheptadine The therapeutic efficacy of Dapoxetine can be decreased when used in combination with Cyproheptadine.
Desmopressin The risk or severity of hyponatremia can be increased when Dapoxetine is combined with Desmopressin.
Ioflupane I-123 Dapoxetine may decrease effectiveness of Ioflupane I-123 as a diagnostic agent.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Dapoxetine.
Metyrosine The risk or severity of extrapyramidal symptoms can be increased when Metyrosine is combined with Dapoxetine.
Pimozide The risk or severity of QTc prolongation can be increased when Dapoxetine is combined with Pimozide.
Ramipril Dapoxetine may increase the orthostatic hypotensive activities of Ramipril.
Fosinopril Dapoxetine may increase the orthostatic hypotensive activities of Fosinopril.
Trandolapril Dapoxetine may increase the orthostatic hypotensive activities of Trandolapril.
Benazepril Dapoxetine may increase the orthostatic hypotensive activities of Benazepril.
Enalapril Dapoxetine may increase the orthostatic hypotensive activities of Enalapril.
Moexipril Dapoxetine may increase the orthostatic hypotensive activities of Moexipril.
Lisinopril Dapoxetine may increase the orthostatic hypotensive activities of Lisinopril.
Perindopril Dapoxetine may increase the orthostatic hypotensive activities of Perindopril.
Quinapril Dapoxetine may increase the orthostatic hypotensive activities of Quinapril.
Omapatrilat Dapoxetine may increase the orthostatic hypotensive activities of Omapatrilat.
Rescinnamine Dapoxetine may increase the orthostatic hypotensive activities of Rescinnamine.
Captopril Dapoxetine may increase the orthostatic hypotensive activities of Captopril.
Cilazapril Dapoxetine may increase the orthostatic hypotensive activities of Cilazapril.
Spirapril Dapoxetine may increase the orthostatic hypotensive activities of Spirapril.
Temocapril Dapoxetine may increase the orthostatic hypotensive activities of Temocapril.
Enalaprilat Dapoxetine may increase the orthostatic hypotensive activities of Enalaprilat.
Imidapril Dapoxetine may increase the orthostatic hypotensive activities of Imidapril.
Zofenopril Dapoxetine may increase the orthostatic hypotensive activities of Zofenopril.
Delapril Dapoxetine may increase the orthostatic hypotensive activities of Delapril.
Benazeprilat Dapoxetine may increase the orthostatic hypotensive activities of Benazeprilat.
Fosinoprilat Dapoxetine may increase the orthostatic hypotensive activities of Fosinoprilat.
Ramiprilat Dapoxetine may increase the orthostatic hypotensive activities of Ramiprilat.
Trandolaprilat Dapoxetine may increase the orthostatic hypotensive activities of Trandolaprilat.
Moexiprilat Dapoxetine may increase the orthostatic hypotensive activities of Moexiprilat.
Perindoprilat Dapoxetine may increase the orthostatic hypotensive activities of Perindoprilat.
Quinaprilat Dapoxetine may increase the orthostatic hypotensive activities of Quinaprilat.
Cilazaprilat Dapoxetine may increase the orthostatic hypotensive activities of Cilazaprilat.
Buprenorphine Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Dapoxetine.
Dronabinol The serum concentration of Dronabinol can be increased when it is combined with Dapoxetine.
Hydrocodone Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Dapoxetine.
Magnesium sulfate The therapeutic efficacy of Dapoxetine can be increased when used in combination with Magnesium sulfate.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Dapoxetine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Dapoxetine.
Orphenadrine Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Dapoxetine.
Pramipexole Dapoxetine may increase the sedative activities of Pramipexole.
Ropinirole Dapoxetine may increase the sedative activities of Ropinirole.
Rotigotine Dapoxetine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Dapoxetine.
Sodium oxybate Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Dapoxetine.
Thalidomide Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Dapoxetine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Dapoxetine.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Dapoxetine.
Tadalafil The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Tadalafil.
Vardenafil The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Vardenafil.
Dipyridamole The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Dipyridamole.
Ibudilast The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Ibudilast.
Avanafil The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Avanafil.
Udenafil The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Udenafil.
Doxofylline The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Doxofylline.
Mirodenafil The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Mirodenafil.
Fostamatinib The risk or severity of orthostatic hypotension can be increased when Dapoxetine is combined with Fostamatinib.
Cilostazol The metabolism of Cilostazol can be decreased when combined with Dapoxetine.
Colchicine The metabolism of Colchicine can be decreased when combined with Dapoxetine.
Fentanyl The risk or severity of serotonin syndrome can be increased when Fentanyl is combined with Dapoxetine.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Dapoxetine.
Retapamulin The metabolism of Retapamulin can be decreased when combined with Dapoxetine.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with Dapoxetine.
Zopiclone The metabolism of Zopiclone can be decreased when combined with Dapoxetine.
Lovastatin The metabolism of Lovastatin can be decreased when combined with Dapoxetine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Dapoxetine.
Dihydroergotamine Dapoxetine may increase the orthostatic hypotensive activities of Dihydroergotamine.
Olanzapine Dapoxetine may increase the orthostatic hypotensive activities of Olanzapine.
Clozapine The serum concentration of Clozapine can be increased when it is combined with Dapoxetine.
Promazine Dapoxetine may increase the orthostatic hypotensive activities of Promazine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Dapoxetine.
Prazosin Dapoxetine may increase the orthostatic hypotensive activities of Prazosin.
Imipramine Dapoxetine may increase the orthostatic hypotensive activities of Imipramine.
Chlorpromazine Dapoxetine may increase the orthostatic hypotensive activities of Chlorpromazine.
Nortriptyline Dapoxetine may increase the orthostatic hypotensive activities of Nortriptyline.
Amoxapine Dapoxetine may increase the orthostatic hypotensive activities of Amoxapine.
Doxazosin Dapoxetine may increase the orthostatic hypotensive activities of Doxazosin.
Labetalol Dapoxetine may increase the orthostatic hypotensive activities of Labetalol.
Nicardipine Dapoxetine may increase the orthostatic hypotensive activities of Nicardipine.
Verapamil The metabolism of Dapoxetine can be decreased when combined with Verapamil.
Phentolamine Dapoxetine may increase the orthostatic hypotensive activities of Phentolamine.
Ergotamine Dapoxetine may increase the orthostatic hypotensive activities of Ergotamine.
Nicergoline Dapoxetine may increase the orthostatic hypotensive activities of Nicergoline.
Tamsulosin Dapoxetine may increase the orthostatic hypotensive activities of Tamsulosin.
Trimipramine Dapoxetine may increase the orthostatic hypotensive activities of Trimipramine.
Risperidone Dapoxetine may increase the orthostatic hypotensive activities of Risperidone.
Propiomazine Dapoxetine may increase the orthostatic hypotensive activities of Propiomazine.
Tolazoline Dapoxetine may increase the orthostatic hypotensive activities of Tolazoline.
Trifluoperazine Dapoxetine may increase the orthostatic hypotensive activities of Trifluoperazine.
Flupentixol Dapoxetine may increase the orthostatic hypotensive activities of Flupentixol.
Quinidine Dapoxetine may increase the orthostatic hypotensive activities of Quinidine.
Phenoxybenzamine Dapoxetine may increase the orthostatic hypotensive activities of Phenoxybenzamine.

Target Protein

5-hydroxytryptamine receptor 1A HTR1A
5-hydroxytryptamine receptor 1B HTR1B
5-hydroxytryptamine receptor 2C HTR2C

Referensi & Sumber

Artikel (PubMed)
  • PMID: 17625501
    Safarinejad MR: Safety and efficacy of dapoxetine in the treatment of premature ejaculation: a double-blind, placebo-controlled, fixed-dose, randomized study. Neuropsychopharmacology. 2008 May;33(6):1259-65. Epub 2007 Jul 11.
  • PMID: 17909314
    Cirillo-Penn K, Modi NB: Dapoxetine and paroxetine for the treatment of premature ejaculation. Clin Neuropharmacol. 2007 Sep-Oct;30(5):315.
  • PMID: 17909313
    McMahon C: Dapoxetine in the treatment of premature ejaculation. Clin Neuropharmacol. 2007 Sep-Oct;30(5):314-5.
  • PMID: 17624269
    Wang WF, Chang L, Minhas S, Ralph DJ: Selective serotonin reuptake inhibitors in the treatment of premature ejaculation. Chin Med J (Engl). 2007 Jun 5;120(11):1000-6.
  • PMID: 16962882
    Pryor JL, Althof SE, Steidle C, Rosen RC, Hellstrom WJ, Shabsigh R, Miloslavsky M, Kell S: Efficacy and tolerability of dapoxetine in treatment of premature ejaculation: an integrated analysis of two double-blind, randomised controlled trials. Lancet. 2006 Sep 9;368(9539):929-37.
  • PMID: 17052444
    Hellstrom WJ, Heintz JW: Treatment of premature ejaculation: new drugs and treatment strategies. Curr Urol Rep. 2006 Nov;7(6):473-8.
  • PMID: 17322143
    Modi NB, Dresser M, Desai D, Edgar C, Wesnes K: Dapoxetine has no pharmacokinetic or cognitive interactions with ethanol in healthy male volunteers. J Clin Pharmacol. 2007 Mar;47(3):315-22.
  • PMID: 17546831
    Payne RE, Sadovsky R: Identifying and treating premature ejaculation: importance of the sexual history. Cleve Clin J Med. 2007 May;74 Suppl 3:S47-53.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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