Enoximone

DB04880

small molecule approved investigational

Deskripsi

Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption. It is used in patients with congestive heart failure. Trials were halted in the U.S., but the drug is used in various countries.

Struktur Molekul 2D

Berat 248.301
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 4-10 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Bioavailabvility is 50% following oral administration.

Metabolisme

Hepatic oxidation

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

8 Data
Milrinone The risk or severity of congestive heart failure, bleeding, hypotension, and Tachycardia can be increased when Milrinone is combined with Enoximone.
Anagrelide The risk or severity of congestive heart failure, bleeding, hypotension, and Tachycardia can be increased when Anagrelide is combined with Enoximone.
Cilostazol The risk or severity of congestive heart failure, bleeding, hypotension, and Tachycardia can be increased when Cilostazol is combined with Enoximone.
Amrinone The risk or severity of congestive heart failure, bleeding, hypotension, and Tachycardia can be increased when Amrinone is combined with Enoximone.
Riociguat Enoximone may increase the hypotensive activities of Riociguat.
Patent Blue The therapeutic efficacy of Enoximone can be decreased when used in combination with Patent Blue.
Isosorbide mononitrate Enoximone may increase the vasodilatory activities of Isosorbide mononitrate.
Iloprost Iloprost may increase the hypotensive activities of Enoximone.

Target Protein

cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A PDE3A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16987374
    Sandroni C, Cavallaro F, Caricato A, Scapigliati A, Fenici P, Antonelli M: Enoximone in cardiac arrest caused by propranolol: two case reports. Acta Anaesthesiol Scand. 2006 Jul;50(6):759-61.
  • PMID: 17544886
    van der Maaten JM, de Vries AJ, Rietman GW, Gallandat Huet RC, De Hert SG: Effects of preemptive enoximone on left ventricular diastolic function after valve replacement for aortic stenosis. J Cardiothorac Vasc Anesth. 2007 Jun;21(3):357-66. Epub 2006 May 4.
  • PMID: 17696974
    Schauvliege S, Van den Eede A, Duchateau L, Gasthuys F: Cardiovascular effects of enoximone in isoflurane anaesthetized ponies. Vet Anaesth Analg. 2007 Nov;34(6):416-30. Epub 2007 Aug 13.
  • PMID: 17714066
    Boldt J, Suttner S: Combined use of ultra-short acting beta-blocker esmolol and intravenous phosphodiesterase 3 inhibitor enoximone. Expert Opin Pharmacother. 2007 Sep;8(13):2135-47.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Perfan

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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