Osanetant

DB04872

small molecule investigational

Deskripsi

Developed by Sanofi-Aventis (formerly Sanofi-Synthelabo), osanetant (SR-142801) is an NK3 receptor antagonist which was under development for the treatment of schizophrenia and other Central Nervous System (CNS) disorders. In a review of its R&D portfolio, the company announced in August 2005 that it would cease any further development of osanetant. This follows an earlier decision to discontinue development of eplivanserin for schizophrenia.

Struktur Molekul 2D

Berat 606.625
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

714 Data
Buprenorphine Osanetant may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Hydrocodone Osanetant may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Magnesium sulfate The therapeutic efficacy of Osanetant can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Osanetant may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Osanetant may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Mirtazapine Osanetant may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Orphenadrine Osanetant may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Osanetant may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Pramipexole Osanetant may increase the sedative activities of Pramipexole.
Ropinirole Osanetant may increase the sedative activities of Ropinirole.
Rotigotine Osanetant may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Osanetant.
Sodium oxybate Osanetant may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Osanetant may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Thalidomide Osanetant may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Osanetant may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Amisulpride Osanetant may increase the antipsychotic activities of Amisulpride.
Methylphenidate The risk or severity of adverse effects can be increased when Osanetant is combined with Methylphenidate.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Osanetant is combined with Dexmethylphenidate.
Metoclopramide The risk or severity of adverse effects can be increased when Metoclopramide is combined with Osanetant.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with Osanetant.
Sulpiride Osanetant may increase the antipsychotic activities of Sulpiride.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Osanetant.
Lithium citrate Lithium citrate may increase the neurotoxic activities of Osanetant.
Lithium hydroxide Lithium hydroxide may increase the neurotoxic activities of Osanetant.
Mequitazine Osanetant may increase the arrhythmogenic activities of Mequitazine.
Tetrabenazine The risk or severity of adverse effects can be increased when Osanetant is combined with Tetrabenazine.
Deutetrabenazine The risk or severity of adverse effects can be increased when Osanetant is combined with Deutetrabenazine.
Ethanol Osanetant may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Osanetant may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Osanetant.
Zimelidine The risk or severity of adverse effects can be increased when Osanetant is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Osanetant is combined with Dapoxetine.
Seproxetine The risk or severity of adverse effects can be increased when Osanetant is combined with Seproxetine.
Fluvoxamine The risk or severity of adverse effects can be increased when Osanetant is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Osanetant is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Osanetant is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Osanetant is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Osanetant is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Osanetant is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Osanetant is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Osanetant is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Osanetant is combined with Escitalopram.
Milnacipran The risk or severity of adverse effects can be increased when Osanetant is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Osanetant is combined with Desvenlafaxine.
Levomilnacipran The risk or severity of adverse effects can be increased when Levomilnacipran is combined with Osanetant.
Indalpine The risk or severity of adverse effects can be increased when Osanetant is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Osanetant is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Osanetant is combined with Alaproclate.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Osanetant.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Osanetant.
Zopiclone The risk or severity of adverse effects can be increased when Osanetant is combined with Zopiclone.
Eletriptan The risk or severity of adverse effects can be increased when Eletriptan is combined with Osanetant.
Cabergoline The risk or severity of adverse effects can be increased when Cabergoline is combined with Osanetant.
Zolmitriptan The risk or severity of adverse effects can be increased when Zolmitriptan is combined with Osanetant.
Dihydroergotamine The risk or severity of adverse effects can be increased when Dihydroergotamine is combined with Osanetant.
Meperidine The risk or severity of adverse effects can be increased when Meperidine is combined with Osanetant.
Dextromethorphan The risk or severity of adverse effects can be increased when Dextromethorphan is combined with Osanetant.
Mazindol The risk or severity of adverse effects can be increased when Mazindol is combined with Osanetant.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Osanetant.
Sumatriptan The risk or severity of adverse effects can be increased when Sumatriptan is combined with Osanetant.
Ergotamine The risk or severity of adverse effects can be increased when Ergotamine is combined with Osanetant.
Fentanyl The risk or severity of adverse effects can be increased when Fentanyl is combined with Osanetant.
Almotriptan The risk or severity of adverse effects can be increased when Almotriptan is combined with Osanetant.
Naratriptan The risk or severity of adverse effects can be increased when Naratriptan is combined with Osanetant.
Rizatriptan The risk or severity of adverse effects can be increased when Rizatriptan is combined with Osanetant.
Frovatriptan The risk or severity of adverse effects can be increased when Frovatriptan is combined with Osanetant.
Ergoloid mesylate The risk or severity of adverse effects can be increased when Ergoloid mesylate is combined with Osanetant.
Chlorpheniramine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Osanetant.
Procarbazine The risk or severity of adverse effects can be increased when Procarbazine is combined with Osanetant.
Bromocriptine The risk or severity of adverse effects can be increased when Bromocriptine is combined with Osanetant.
Ergometrine The risk or severity of adverse effects can be increased when Ergometrine is combined with Osanetant.
Rasagiline The risk or severity of adverse effects can be increased when Rasagiline is combined with Osanetant.
Lorcaserin The risk or severity of adverse effects can be increased when Lorcaserin is combined with Osanetant.
Etoperidone The risk or severity of adverse effects can be increased when Etoperidone is combined with Osanetant.
Lorpiprazole The risk or severity of adverse effects can be increased when Lorpiprazole is combined with Osanetant.
Amphetamine Osanetant may decrease the stimulatory activities of Amphetamine.
Phentermine Osanetant may decrease the stimulatory activities of Phentermine.
Pseudoephedrine Osanetant may decrease the stimulatory activities of Pseudoephedrine.
Benzphetamine Osanetant may decrease the stimulatory activities of Benzphetamine.
Diethylpropion Osanetant may decrease the stimulatory activities of Diethylpropion.
Lisdexamfetamine Osanetant may decrease the stimulatory activities of Lisdexamfetamine.
Mephentermine Osanetant may decrease the stimulatory activities of Mephentermine.
MMDA Osanetant may decrease the stimulatory activities of MMDA.
2,5-Dimethoxy-4-ethylamphetamine Osanetant may decrease the stimulatory activities of 2,5-Dimethoxy-4-ethylamphetamine.
Chlorphentermine Osanetant may decrease the stimulatory activities of Chlorphentermine.
Methylenedioxyethamphetamine Osanetant may decrease the stimulatory activities of Methylenedioxyethamphetamine.
Dextroamphetamine Osanetant may decrease the stimulatory activities of Dextroamphetamine.
Metamfetamine Osanetant may decrease the stimulatory activities of Metamfetamine.
Iofetamine I-123 Osanetant may decrease the stimulatory activities of Iofetamine I-123.
Ritobegron Osanetant may decrease the stimulatory activities of Ritobegron.
Mephedrone Osanetant may decrease the stimulatory activities of Mephedrone.

Target Protein

Neuromedin-K receptor TACR3

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15706463
    Kronenberg G, Berger P, Tauber RF, Bandelow B, Henkel V, Heuser I: Randomized, double-blind study of SR142801 (Osanetant). A novel neurokinin-3 (NK3) receptor antagonist in panic disorder with pre- and posttreatment cholecystokinin tetrapeptide (CCK-4) challenges. Pharmacopsychiatry. 2005 Jan;38(1):24-9.
  • PMID: 11757797
    Kamali F: Osanetant Sanofi-Synthelabo. Curr Opin Investig Drugs. 2001 Jul;2(7):950-6.

Contoh Produk & Brand

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Sekuens Gen/Protein (FASTA)

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