Halofuginone

DB04866

small molecule investigational vet_approved

Deskripsi

Halofuginone is a low molecular weight quinazolinone alkaloid, and a potent inhibitor of collagen alpha1(I) and matrix metalloproteinase 2 (MMP-2) gene expression. Halofuginone also effectively suppresses tumor progression and metastasis in mice. Collgard Biopharmaceuticals is developing halofuginone for the treatment of scleroderma and received orphan drug designation from the U.S. Food and Drug Administration in March, 2000.

Struktur Molekul 2D

Berat 414.681
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 23.8 to 72.1 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Readily bioavailable and rapidly absorbed following oral administration.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

48 Data
Pamidronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Pamidronic acid.
Zoledronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Zoledronic acid.
Alendronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Alendronic acid.
Ibandronate The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Ibandronate.
Clodronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Clodronic acid.
Risedronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Risedronic acid.
Etidronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Etidronic acid.
Tiludronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Tiludronic acid.
Incadronic acid The risk or severity of jaw osteonecrosis and anti-angiogenesis can be increased when Halofuginone is combined with Incadronic acid.
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Halofuginone.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Halofuginone.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Halofuginone.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Halofuginone.
Lidocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Quinisocaine.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Halofuginone.
Ambroxol The risk or severity of methemoglobinemia can be increased when Halofuginone is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Halofuginone is combined with Etrasimod.

Target Protein

Collagen alpha-1(I) chain COL1A1
72 kDa type IV collagenase MMP2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 11099465
    Elkin M, Miao HQ, Nagler A, Aingorn E, Reich R, Hemo I, Dou HL, Pines M, Vlodavsky I: Halofuginone: a potent inhibitor of critical steps in angiogenesis progression. FASEB J. 2000 Dec;14(15):2477-85.
  • PMID: 19498172
    Sundrud MS, Koralov SB, Feuerer M, Calado DP, Kozhaya AE, Rhule-Smith A, Lefebvre RE, Unutmaz D, Mazitschek R, Waldner H, Whitman M, Keller T, Rao A: Halofuginone inhibits TH17 cell differentiation by activating the amino acid starvation response. Science. 2009 Jun 5;324(5932):1334-8. doi: 10.1126/science.1172638.
  • PMID: 22327401
    Keller TL, Zocco D, Sundrud MS, Hendrick M, Edenius M, Yum J, Kim YJ, Lee HK, Cortese JF, Wirth DF, Dignam JD, Rao A, Yeo CY, Mazitschek R, Whitman M: Halofuginone and other febrifugine derivatives inhibit prolyl-tRNA synthetase. Nat Chem Biol. 2012 Feb 12;8(3):311-7. doi: 10.1038/nchembio.790.

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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