Peringatan Keamanan

Clinical signs of acute toxicity lead to decreased activity, ataxia, vomiting and tremors.

Posizolid

DB04850

small molecule investigational

Deskripsi

Posizolid (AZD2563) is an oxazolidinone antibiotic. In July 2002, after completion of phase I trials in December 2001, AstraZeneca announced that they were no longer pursuing the development of Posizolid, presumably due to negative trial results (though no results were reported).

Struktur Molekul 2D

Berat 465.41
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

58 Data
Eluxadoline The serum concentration of Eluxadoline can be increased when it is combined with Posizolid.
Pravastatin The excretion of Pravastatin can be decreased when combined with Posizolid.
Valsartan The excretion of Valsartan can be decreased when combined with Posizolid.
Erythromycin The excretion of Erythromycin can be decreased when combined with Posizolid.
Torasemide The excretion of Torasemide can be decreased when combined with Posizolid.
Liothyronine The excretion of Liothyronine can be decreased when combined with Posizolid.
Conjugated estrogens The excretion of Conjugated estrogens can be decreased when combined with Posizolid.
Digoxin The excretion of Digoxin can be decreased when combined with Posizolid.
Cerivastatin The excretion of Cerivastatin can be decreased when combined with Posizolid.
Raloxifene The excretion of Raloxifene can be decreased when combined with Posizolid.
Caspofungin The excretion of Caspofungin can be decreased when combined with Posizolid.
Bosentan The excretion of Bosentan can be decreased when combined with Posizolid.
Methotrexate The excretion of Methotrexate can be decreased when combined with Posizolid.
Enalapril The excretion of Enalapril can be decreased when combined with Posizolid.
Simvastatin The excretion of Simvastatin can be decreased when combined with Posizolid.
Sumatriptan The excretion of Sumatriptan can be decreased when combined with Posizolid.
Mycophenolate mofetil The excretion of Mycophenolate mofetil can be decreased when combined with Posizolid.
Penicillamine The excretion of Penicillamine can be decreased when combined with Posizolid.
Repaglinide The excretion of Repaglinide can be decreased when combined with Posizolid.
Dinoprostone The excretion of Dinoprostone can be decreased when combined with Posizolid.
Fexofenadine The excretion of Fexofenadine can be decreased when combined with Posizolid.
Ezetimibe The excretion of Ezetimibe can be decreased when combined with Posizolid.
Benzylpenicillin The excretion of Benzylpenicillin can be decreased when combined with Posizolid.
Atorvastatin The excretion of Atorvastatin can be decreased when combined with Posizolid.
Ouabain The excretion of Ouabain can be decreased when combined with Posizolid.
Fluvastatin The excretion of Fluvastatin can be decreased when combined with Posizolid.
Rosuvastatin The excretion of Rosuvastatin can be decreased when combined with Posizolid.
Liotrix The excretion of Liotrix can be decreased when combined with Posizolid.
Cholic Acid The excretion of Cholic Acid can be decreased when combined with Posizolid.
Taurocholic acid The excretion of Taurocholic acid can be decreased when combined with Posizolid.
Atrasentan The excretion of Atrasentan can be decreased when combined with Posizolid.
Simeprevir The excretion of Simeprevir can be decreased when combined with Posizolid.
Ambrisentan The excretion of Ambrisentan can be decreased when combined with Posizolid.
Axitinib The excretion of Axitinib can be decreased when combined with Posizolid.
Gimatecan The excretion of Gimatecan can be decreased when combined with Posizolid.
Temocapril The excretion of Temocapril can be decreased when combined with Posizolid.
Cholecystokinin The excretion of Cholecystokinin can be decreased when combined with Posizolid.
Gadoxetic acid The excretion of Gadoxetic acid can be decreased when combined with Posizolid.
Technetium Tc-99m mebrofenin The excretion of Technetium Tc-99m mebrofenin can be decreased when combined with Posizolid.
Fimasartan The excretion of Fimasartan can be decreased when combined with Posizolid.
Paritaprevir The excretion of Paritaprevir can be decreased when combined with Posizolid.
Tenofovir alafenamide The excretion of Tenofovir alafenamide can be decreased when combined with Posizolid.
Selexipag The excretion of Selexipag can be decreased when combined with Posizolid.
Grazoprevir The excretion of Grazoprevir can be decreased when combined with Posizolid.
Asunaprevir The excretion of Asunaprevir can be decreased when combined with Posizolid.
Elagolix The excretion of Elagolix can be decreased when combined with Posizolid.
Voxilaprevir The excretion of Voxilaprevir can be decreased when combined with Posizolid.
Letermovir The excretion of Letermovir can be decreased when combined with Posizolid.
Levosalbutamol The excretion of Levosalbutamol can be decreased when combined with Posizolid.
Glecaprevir The excretion of Glecaprevir can be decreased when combined with Posizolid.
Belantamab mafodotin The excretion of Belantamab mafodotin can be decreased when combined with Posizolid.
Revefenacin Posizolid may decrease the excretion rate of Revefenacin which could result in a higher serum level.
Brincidofovir The serum concentration of Brincidofovir can be increased when it is combined with Posizolid.
Atogepant The serum concentration of Atogepant can be increased when it is combined with Posizolid.
Mesalazine The excretion of Mesalazine can be decreased when combined with Posizolid.
Tezacaftor The excretion of Tezacaftor can be decreased when combined with Posizolid.
Momelotinib The serum concentration of Momelotinib can be increased when it is combined with Posizolid.
Resmetirom The serum concentration of Resmetirom can be increased when it is combined with Posizolid.

Target Protein

23S ribosomal RNA
Amine oxidase [flavin-containing] A MAOA

Referensi & Sumber

Artikel (PubMed)
  • PMID: 12096013
    Ednie LM, Jacobs MR, Appelbaum PC: Anti-anaerobic activity of AZD2563, a new oxazolidinone, compared with eight other agents. J Antimicrob Chemother. 2002 Jul;50(1):101-5.
  • PMID: 15008947
    Wookey A, Turner PJ, Greenhalgh JM, Eastwood M, Clarke J, Sefton C: AZD2563, a novel oxazolidinone: definition of antibacterial spectrum, assessment of bactericidal potential and the impact of miscellaneous factors on activity in vitro. Clin Microbiol Infect. 2004 Mar;10(3):247-54.
  • PMID: 14576139
    Howe RA, Wootton M, Noel AR, Bowker KE, Walsh TR, MacGowan AP: Activity of AZD2563, a novel oxazolidinone, against Staphylococcus aureus strains with reduced susceptibility to vancomycin or linezolid. Antimicrob Agents Chemother. 2003 Nov;47(11):3651-2.
  • PMID: 24189255
    Balasubramanian V, Solapure S, Iyer H, Ghosh A, Sharma S, Kaur P, Deepthi R, Subbulakshmi V, Ramya V, Ramachandran V, Balganesh M, Wright L, Melnick D, Butler SL, Sambandamurthy VK: Bactericidal activity and mechanism of action of AZD5847, a novel oxazolidinone for treatment of tuberculosis. Antimicrob Agents Chemother. 2014;58(1):495-502. doi: 10.1128/AAC.01903-13. Epub 2013 Nov 4.
Link

Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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