Cediranib

DB04849

small molecule investigational

Deskripsi

The novel indole-ether quinazoline Cediranib is a highly potent (IC50 < 1 nmol/L) ATP-competitive inhibitor of recombinant KDR tyrosine kinase in vitro. It is being developed clinically as a once-daily oral therapy for the treatment of cancer.

Struktur Molekul 2D

Berat 450.5053
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 12 to 35 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Available following oral administration.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

66 Data
Acetaminophen The serum concentration of Acetaminophen can be increased when it is combined with Cediranib.
Propacetamol The serum concentration of Propacetamol can be increased when it is combined with Cediranib.
Salmon calcitonin The therapeutic efficacy of Salmon calcitonin can be decreased when used in combination with Cediranib.
Thyrotropin alfa The therapeutic efficacy of Thyrotropin alfa can be decreased when used in combination with Cediranib.
Follitropin The therapeutic efficacy of Follitropin can be decreased when used in combination with Cediranib.
Liothyronine The therapeutic efficacy of Liothyronine can be decreased when used in combination with Cediranib.
Carbimazole The therapeutic efficacy of Carbimazole can be decreased when used in combination with Cediranib.
Levothyroxine The therapeutic efficacy of Levothyroxine can be decreased when used in combination with Cediranib.
Propylthiouracil The therapeutic efficacy of Propylthiouracil can be decreased when used in combination with Cediranib.
Methimazole The therapeutic efficacy of Methimazole can be decreased when used in combination with Cediranib.
Liotrix The therapeutic efficacy of Liotrix can be decreased when used in combination with Cediranib.
3,5-Diiodotyrosine The therapeutic efficacy of 3,5-Diiodotyrosine can be decreased when used in combination with Cediranib.
Tiratricol The therapeutic efficacy of Tiratricol can be decreased when used in combination with Cediranib.
Parathyroid hormone The therapeutic efficacy of Parathyroid hormone can be decreased when used in combination with Cediranib.
Teriparatide The therapeutic efficacy of Teriparatide can be decreased when used in combination with Cediranib.
Potassium Iodide The therapeutic efficacy of Potassium Iodide can be decreased when used in combination with Cediranib.
Dibromotyrosine The therapeutic efficacy of Dibromotyrosine can be decreased when used in combination with Cediranib.
Thyroid, porcine The therapeutic efficacy of Thyroid, porcine can be decreased when used in combination with Cediranib.
Potassium perchlorate The therapeutic efficacy of Potassium perchlorate can be decreased when used in combination with Cediranib.
Protirelin The therapeutic efficacy of Protirelin can be decreased when used in combination with Cediranib.
3,5-diiodothyropropionic acid The therapeutic efficacy of 3,5-diiodothyropropionic acid can be decreased when used in combination with Cediranib.
Methylthiouracil The therapeutic efficacy of Methylthiouracil can be decreased when used in combination with Cediranib.
Elcatonin The therapeutic efficacy of Elcatonin can be decreased when used in combination with Cediranib.
Benzylthiouracil The therapeutic efficacy of Benzylthiouracil can be decreased when used in combination with Cediranib.
Thyrotropin The therapeutic efficacy of Thyrotropin can be decreased when used in combination with Cediranib.
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Cediranib.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Cediranib.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Cediranib.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Cediranib.
Lidocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Quinisocaine.
Voriconazole The serum concentration of Cediranib can be increased when it is combined with Voriconazole.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Cediranib.
Ambroxol The risk or severity of methemoglobinemia can be increased when Cediranib is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Cediranib is combined with Etrasimod.
Palopegteriparatide The therapeutic efficacy of Palopegteriparatide can be decreased when used in combination with Cediranib.

Target Protein

Vascular endothelial growth factor receptor 2 KDR

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15899831
    Wedge SR, Kendrew J, Hennequin LF, Valentine PJ, Barry ST, Brave SR, Smith NR, James NH, Dukes M, Curwen JO, Chester R, Jackson JA, Boffey SJ, Kilburn LL, Barnett S, Richmond GH, Wadsworth PF, Walker M, Bigley AL, Taylor ST, Cooper L, Beck S, Jurgensmeier JM, Ogilvie DJ: AZD2171: a highly potent, orally bioavailable, vascular endothelial growth factor receptor-2 tyrosine kinase inhibitor for the treatment of cancer. Cancer Res. 2005 May 15;65(10):4389-400.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Recentin

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul