Ixabepilone

DB04845

small molecule approved investigational

Deskripsi

Ixabepilone is an epothilone B analog developed by Bristol-Myers Squibb as a cancer drug. It was FDA approved on October 16, 2007, for the treatment of unresponsive aggressive metastatic or locally advanced breast cancer. Ixabepilone is administered through injection, and will be marketed under the trade name Ixempra. Ixabepilone is a semisynthetic analogue of epothilone B. It has a lactone–lactam modification that minimizes susceptibility to esterase degradation.

Struktur Molekul 2D

Berat 506.7
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 52 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Mostly fecal and some renal.

Interaksi Makanan

2 Data
  • 1. Avoid grapefruit products. Grapefruit inhibits the CYP3A4 metabolism of ixabepilone, which may increase its serum concentration.
  • 2. Avoid St. John's Wort. This herb induces CYP3A metabolism and may reduce serum levels of ixabepilone.

Interaksi Obat

1030 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Ixabepilone.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Ixabepilone.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Ixabepilone.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Ixabepilone.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Ixabepilone.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Ixabepilone.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Ixabepilone.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Ixabepilone.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Ixabepilone.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Ixabepilone.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Ixabepilone.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Ixabepilone.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Ixabepilone.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Ixabepilone.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Ixabepilone.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Ixabepilone.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Ixabepilone.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Ixabepilone.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Ixabepilone.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Ixabepilone.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Ixabepilone.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Ixabepilone.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Ixabepilone.
Cladribine Ixabepilone may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Carmustine is combined with Ixabepilone.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Ixabepilone.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Ixabepilone.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Ixabepilone.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Ixabepilone.
Mitomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Ixabepilone.
Vindesine The risk or severity of adverse effects can be increased when Vindesine is combined with Ixabepilone.
Floxuridine The risk or severity of adverse effects can be increased when Floxuridine is combined with Ixabepilone.
Indomethacin The risk or severity of adverse effects can be increased when Indomethacin is combined with Ixabepilone.
Tioguanine The risk or severity of adverse effects can be increased when Tioguanine is combined with Ixabepilone.
Dexrazoxane The risk or severity of adverse effects can be increased when Dexrazoxane is combined with Ixabepilone.
Streptozocin The risk or severity of adverse effects can be increased when Streptozocin is combined with Ixabepilone.
Trifluridine The risk or severity of adverse effects can be increased when Trifluridine is combined with Ixabepilone.
Epirubicin The risk or severity of adverse effects can be increased when Epirubicin is combined with Ixabepilone.
Lenalidomide The risk or severity of adverse effects can be increased when Lenalidomide is combined with Ixabepilone.
Altretamine The risk or severity of adverse effects can be increased when Altretamine is combined with Ixabepilone.
Zidovudine The risk or severity of adverse effects can be increased when Zidovudine is combined with Ixabepilone.
Cisplatin The risk or severity of adverse effects can be increased when Cisplatin is combined with Ixabepilone.
Oxaliplatin The risk or severity of adverse effects can be increased when Oxaliplatin is combined with Ixabepilone.
Fluorouracil The risk or severity of adverse effects can be increased when Fluorouracil is combined with Ixabepilone.
Propylthiouracil The risk or severity of adverse effects can be increased when Propylthiouracil is combined with Ixabepilone.
Pentostatin The risk or severity of adverse effects can be increased when Pentostatin is combined with Ixabepilone.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Ixabepilone.
Clofarabine The risk or severity of adverse effects can be increased when Clofarabine is combined with Ixabepilone.
Pemetrexed The risk or severity of adverse effects can be increased when Pemetrexed is combined with Ixabepilone.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Mycophenolate mofetil is combined with Ixabepilone.
Irinotecan The risk or severity of adverse effects can be increased when Irinotecan is combined with Ixabepilone.
Sulfasalazine The risk or severity of adverse effects can be increased when Sulfasalazine is combined with Ixabepilone.
Dacarbazine The risk or severity of adverse effects can be increased when Dacarbazine is combined with Ixabepilone.
Temozolomide The risk or severity of adverse effects can be increased when Temozolomide is combined with Ixabepilone.
Penicillamine The risk or severity of adverse effects can be increased when Penicillamine is combined with Ixabepilone.
Mechlorethamine The risk or severity of adverse effects can be increased when Mechlorethamine is combined with Ixabepilone.
Azacitidine The risk or severity of adverse effects can be increased when Azacitidine is combined with Ixabepilone.
Carboplatin The risk or severity of adverse effects can be increased when Carboplatin is combined with Ixabepilone.
Azathioprine The risk or severity of adverse effects can be increased when Azathioprine is combined with Ixabepilone.
Hydroxyurea The risk or severity of adverse effects can be increased when Hydroxyurea is combined with Ixabepilone.
Mycophenolic acid The risk or severity of adverse effects can be increased when Mycophenolic acid is combined with Ixabepilone.
Mercaptopurine The risk or severity of adverse effects can be increased when Mercaptopurine is combined with Ixabepilone.
Thalidomide The metabolism of Ixabepilone can be increased when combined with Thalidomide.
Melphalan The risk or severity of adverse effects can be increased when Melphalan is combined with Ixabepilone.
Fludarabine The risk or severity of adverse effects can be increased when Fludarabine is combined with Ixabepilone.
Flucytosine The risk or severity of adverse effects can be increased when Flucytosine is combined with Ixabepilone.
Capecitabine The risk or severity of adverse effects can be increased when Capecitabine is combined with Ixabepilone.
Procarbazine The risk or severity of adverse effects can be increased when Procarbazine is combined with Ixabepilone.
Arsenic trioxide The risk or severity of adverse effects can be increased when Arsenic trioxide is combined with Ixabepilone.
Idarubicin The risk or severity of adverse effects can be increased when Idarubicin is combined with Ixabepilone.
Estramustine The risk or severity of adverse effects can be increased when Estramustine is combined with Ixabepilone.
Lomustine The risk or severity of adverse effects can be increased when Lomustine is combined with Ixabepilone.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Ixabepilone.
Decitabine The risk or severity of adverse effects can be increased when Decitabine is combined with Ixabepilone.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Ixabepilone.
Ciclesonide The risk or severity of adverse effects can be increased when Ciclesonide is combined with Ixabepilone.
Stepronin The risk or severity of adverse effects can be increased when Stepronin is combined with Ixabepilone.
Hydroxychloroquine The risk or severity of adverse effects can be increased when Hydroxychloroquine is combined with Ixabepilone.
Castanospermine The risk or severity of adverse effects can be increased when Castanospermine is combined with Ixabepilone.
Vorinostat The risk or severity of adverse effects can be increased when Vorinostat is combined with Ixabepilone.
2-Methoxyethanol The risk or severity of adverse effects can be increased when 2-Methoxyethanol is combined with Ixabepilone.
Brequinar The risk or severity of adverse effects can be increased when Brequinar is combined with Ixabepilone.
Pirfenidone The risk or severity of adverse effects can be increased when Ixabepilone is combined with Pirfenidone.
Belinostat The risk or severity of adverse effects can be increased when Ixabepilone is combined with Belinostat.
Interferon alfa The risk or severity of adverse effects can be increased when Ixabepilone is combined with Interferon alfa.
Glatiramer The risk or severity of adverse effects can be increased when Ixabepilone is combined with Glatiramer.
Briakinumab The risk or severity of adverse effects can be increased when Ixabepilone is combined with Briakinumab.
Human interferon omega-1 The risk or severity of adverse effects can be increased when Ixabepilone is combined with Human interferon omega-1.
Mepolizumab The risk or severity of adverse effects can be increased when Ixabepilone is combined with Mepolizumab.
Abetimus The risk or severity of adverse effects can be increased when Ixabepilone is combined with Abetimus.
Belatacept The risk or severity of adverse effects can be increased when Ixabepilone is combined with Belatacept.
Pralatrexate The risk or severity of adverse effects can be increased when Ixabepilone is combined with Pralatrexate.
Wortmannin The risk or severity of adverse effects can be increased when Ixabepilone is combined with Wortmannin.
Eribulin The risk or severity of adverse effects can be increased when Ixabepilone is combined with Eribulin.
Ruxolitinib The risk or severity of adverse effects can be increased when Ixabepilone is combined with Ruxolitinib.
Belimumab The risk or severity of adverse effects can be increased when Ixabepilone is combined with Belimumab.
Teriflunomide The risk or severity of adverse effects can be increased when Ixabepilone is combined with Teriflunomide.
Ponatinib The risk or severity of adverse effects can be increased when Ixabepilone is combined with Ponatinib.
Dimethyl fumarate The risk or severity of adverse effects can be increased when Ixabepilone is combined with Dimethyl fumarate.
Obinutuzumab The risk or severity of adverse effects can be increased when Ixabepilone is combined with Obinutuzumab.

Target Protein

Tubulin beta-3 chain TUBB3

Referensi & Sumber

Synthesis reference: Ismat Ullah, Gary Wiley, "Enteric coated bead comprising ixabepilone, and preparation and administration thereof." U.S. Patent US20060153917, issued July 13, 2006.

Contoh Produk & Brand

Produk: 4 • International brands: 0
Produk
  • Ixempra
    Kit • 15 mg/15mg • Intravenous • US • Approved
  • Ixempra
    Kit • 45 mg/45mg • Intravenous • US • Approved
  • Ixempra
    Injection, solution; Kit • 15 mg/15mg • Intravenous • US • Approved
  • Ixempra
    Kit • 45 mg/45mg • Intravenous • US • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul