Debrisoquine

DB04840

small molecule approved investigational

Deskripsi

An adrenergic neuron-blocking drug similar in effects to guanethidine. It is also noteworthy in being a substrate for a polymorphic cytochrome P-450 enzyme. Persons with certain isoforms of this enzyme are unable to properly metabolize this and many other clinically important drugs. They are commonly referred to as having a debrisoquin 4-hydroxylase polymorphism.

Struktur Molekul 2D

Berat 175.2303
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

871 Data
Alfuzosin Alfuzosin may increase the hypotensive activities of Debrisoquine.
Amifostine Debrisoquine may increase the hypotensive activities of Amifostine.
Diazoxide Diazoxide may increase the hypotensive activities of Debrisoquine.
Methylphenidate Methylphenidate may decrease the antihypertensive activities of Debrisoquine.
Dexmethylphenidate Dexmethylphenidate may decrease the antihypertensive activities of Debrisoquine.
Obinutuzumab Debrisoquine may increase the hypotensive activities of Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the hypotensive activities of Debrisoquine.
Rituximab Debrisoquine may increase the hypotensive activities of Rituximab.
Desmopressin Desmopressin may decrease the antihypertensive activities of Debrisoquine.
Phentermine Phentermine may decrease the antihypertensive activities of Debrisoquine.
Isoetharine Isoetharine may decrease the antihypertensive activities of Debrisoquine.
Methysergide Methysergide may decrease the antihypertensive activities of Debrisoquine.
Etomidate Etomidate may decrease the antihypertensive activities of Debrisoquine.
Zolmitriptan Zolmitriptan may decrease the antihypertensive activities of Debrisoquine.
Methylergometrine Methylergometrine may decrease the antihypertensive activities of Debrisoquine.
Norepinephrine Norepinephrine may decrease the antihypertensive activities of Debrisoquine.
Phenylephrine Phenylephrine may decrease the antihypertensive activities of Debrisoquine.
Phenylpropanolamine Phenylpropanolamine may decrease the antihypertensive activities of Debrisoquine.
Droperidol Droperidol may decrease the antihypertensive activities of Debrisoquine.
Doxapram Doxapram may decrease the antihypertensive activities of Debrisoquine.
Atropine Atropine may decrease the antihypertensive activities of Debrisoquine.
Metaraminol Metaraminol may decrease the antihypertensive activities of Debrisoquine.
Epinephrine Epinephrine may decrease the antihypertensive activities of Debrisoquine.
Methoxamine Methoxamine may decrease the antihypertensive activities of Debrisoquine.
Propiomazine Propiomazine may decrease the antihypertensive activities of Debrisoquine.
Orciprenaline Orciprenaline may decrease the antihypertensive activities of Debrisoquine.
Phenmetrazine Phenmetrazine may decrease the antihypertensive activities of Debrisoquine.
Dobutamine Dobutamine may decrease the antihypertensive activities of Debrisoquine.
Pseudoephedrine Pseudoephedrine may decrease the antihypertensive activities of Debrisoquine.
Benzphetamine Benzphetamine may decrease the antihypertensive activities of Debrisoquine.
Ritodrine Ritodrine may decrease the antihypertensive activities of Debrisoquine.
Terbutaline Terbutaline may decrease the antihypertensive activities of Debrisoquine.
Bitolterol Bitolterol may decrease the antihypertensive activities of Debrisoquine.
Diethylpropion Diethylpropion may decrease the antihypertensive activities of Debrisoquine.
Salmeterol Salmeterol may decrease the antihypertensive activities of Debrisoquine.
Naratriptan Naratriptan may decrease the antihypertensive activities of Debrisoquine.
Rizatriptan Rizatriptan may decrease the antihypertensive activities of Debrisoquine.
Dopamine Dopamine may decrease the antihypertensive activities of Debrisoquine.
Frovatriptan Frovatriptan may decrease the antihypertensive activities of Debrisoquine.
Albuterol Salbutamol may decrease the antihypertensive activities of Debrisoquine.
Ergoloid mesylate Ergoloid mesylate may decrease the antihypertensive activities of Debrisoquine.
Isoprenaline Isoprenaline may decrease the antihypertensive activities of Debrisoquine.
Arbutamine Arbutamine may decrease the antihypertensive activities of Debrisoquine.
Dutasteride Dutasteride may decrease the antihypertensive activities of Debrisoquine.
Finasteride Finasteride may decrease the antihypertensive activities of Debrisoquine.
Fenoterol Fenoterol may decrease the antihypertensive activities of Debrisoquine.
Pirbuterol Pirbuterol may decrease the antihypertensive activities of Debrisoquine.
Ephedra sinica root Ephedra sinica root may decrease the antihypertensive activities of Debrisoquine.
Ephedrine Ephedrine may decrease the antihypertensive activities of Debrisoquine.
Mephentermine Mephentermine may decrease the antihypertensive activities of Debrisoquine.
Procaterol Procaterol may decrease the antihypertensive activities of Debrisoquine.
Clenbuterol Clenbuterol may decrease the antihypertensive activities of Debrisoquine.
Bambuterol Bambuterol may decrease the antihypertensive activities of Debrisoquine.
MMDA MMDA may decrease the antihypertensive activities of Debrisoquine.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the antihypertensive activities of Debrisoquine.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the antihypertensive activities of Debrisoquine.
Tenamfetamine Tenamfetamine may decrease the antihypertensive activities of Debrisoquine.
Chlorphentermine Chlorphentermine may decrease the antihypertensive activities of Debrisoquine.
Dextroamphetamine Dextroamphetamine may decrease the antihypertensive activities of Debrisoquine.
Phendimetrazine Phendimetrazine may decrease the antihypertensive activities of Debrisoquine.
Solifenacin Solifenacin may decrease the antihypertensive activities of Debrisoquine.
Periciazine Periciazine may decrease the antihypertensive activities of Debrisoquine.
Acepromazine Acepromazine may decrease the antihypertensive activities of Debrisoquine.
Thioproperazine Thioproperazine may decrease the antihypertensive activities of Debrisoquine.
Epicaptopril Epicaptopril may decrease the antihypertensive activities of Debrisoquine.
1-benzylimidazole 1-benzylimidazole may decrease the antihypertensive activities of Debrisoquine.
Amineptine Amineptine may decrease the antihypertensive activities of Debrisoquine.
Amibegron Amibegron may decrease the antihypertensive activities of Debrisoquine.
Naluzotan Naluzotan may decrease the antihypertensive activities of Debrisoquine.
Nylidrin Nylidrin may decrease the antihypertensive activities of Debrisoquine.
Pizotifen Pizotifen may decrease the antihypertensive activities of Debrisoquine.
Solabegron Solabegron may decrease the antihypertensive activities of Debrisoquine.
Droxidopa Droxidopa may decrease the antihypertensive activities of Debrisoquine.
Nitrous oxide Nitrous oxide may decrease the antihypertensive activities of Debrisoquine.
Xylometazoline Xylometazoline may decrease the antihypertensive activities of Debrisoquine.
Isometheptene Isometheptene may decrease the antihypertensive activities of Debrisoquine.
Levonordefrin Levonordefrin may decrease the antihypertensive activities of Debrisoquine.
Naphazoline Naphazoline may decrease the antihypertensive activities of Debrisoquine.
Saralasin Saralasin may decrease the antihypertensive activities of Debrisoquine.
Tetryzoline Tetryzoline may decrease the antihypertensive activities of Debrisoquine.
Cinitapride Cinitapride may decrease the antihypertensive activities of Debrisoquine.
Lurasidone Lurasidone may decrease the antihypertensive activities of Debrisoquine.
Tyramine Tyramine may decrease the antihypertensive activities of Debrisoquine.
Adrafinil Adrafinil may decrease the antihypertensive activities of Debrisoquine.
Ifenprodil Ifenprodil may decrease the antihypertensive activities of Debrisoquine.
Hexoprenaline Hexoprenaline may decrease the antihypertensive activities of Debrisoquine.
Etilefrine Etilefrine may decrease the antihypertensive activities of Debrisoquine.
Dimetacrine Dimetacrine may decrease the antihypertensive activities of Debrisoquine.
Butriptyline Butriptyline may decrease the antihypertensive activities of Debrisoquine.
Olodaterol Olodaterol may decrease the antihypertensive activities of Debrisoquine.
Vilanterol Vilanterol may decrease the antihypertensive activities of Debrisoquine.
Cirazoline Cirazoline may decrease the antihypertensive activities of Debrisoquine.
Synephrine Synephrine may decrease the antihypertensive activities of Debrisoquine.
Moxisylyte Moxisylyte may decrease the antihypertensive activities of Debrisoquine.
Tianeptine Tianeptine may decrease the antihypertensive activities of Debrisoquine.
Oxaprotiline Oxaprotiline may decrease the antihypertensive activities of Debrisoquine.
Iofetamine I-123 Iofetamine I-123 may decrease the antihypertensive activities of Debrisoquine.
Racepinephrine Racepinephrine may decrease the antihypertensive activities of Debrisoquine.
Dihydroergocornine Dihydroergocornine may decrease the antihypertensive activities of Debrisoquine.
DL-Methylephedrine DL-Methylephedrine may decrease the antihypertensive activities of Debrisoquine.

Target Protein

Sodium-dependent noradrenaline transporter SLC6A2

Referensi & Sumber

Synthesis reference: Wenner,W.; U.S. Patent 3,157,573; November 17,1964; assigned to Hoffmann-LaRoche, Inc.

Contoh Produk & Brand

Produk: 0 • International brands: 3
International Brands
  • Bonipress — lkapharm
  • Declinax — Roche
  • Tendor — Chinoin

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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