Maraviroc

DB04835

small molecule approved investigational

Deskripsi

Maraviroc (brand-named Selzentry, or Celsentri outside the U.S.) is a chemokine receptor antagonist drug developed by the drug company Pfizer that is designed to act against HIV by interfering with the interaction between HIV and CCR5. It was originally labelled as UK-427857 during development but was assigned the Maraviroc name as it entered trials. It was approved for use by the FDA in August, 2007.

Struktur Molekul 2D

Berat 513.6655
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 14-18 hours
Volume Distribusi * 194 L
Klirens (Clearance) -

Absorpsi

The absolute oral bioavailability of a 100 mg dose is 23% and is predicted to be 33% at 300 mg. Coadministration of a 300mg tablet with a high fat breakfast reduced maraviroc Cmax and AUC by 33% in healthy volunteers.

Metabolisme

In vitro studies indicate that CYP3A is the major enzyme responsible for maraviroc metabolism.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid St. John's Wort. This herb induces CYP3A metabolism and may reduce serum levels of maraviroc.
  • 2. Take with or without food.

Interaksi Obat

126 Data
Efavirenz The serum concentration of Maraviroc can be decreased when it is combined with Efavirenz.
Pitolisant The serum concentration of Maraviroc can be decreased when it is combined with Pitolisant.
Metreleptin The metabolism of Maraviroc can be increased when combined with Metreleptin.
Rubella virus vaccine The therapeutic efficacy of Rubella virus vaccine can be decreased when used in combination with Maraviroc.
Bacillus calmette-guerin substrain tice live antigen The therapeutic efficacy of Bacillus calmette-guerin substrain tice live antigen can be decreased when used in combination with Maraviroc.
Bacillus calmette-guerin substrain connaught live antigen The therapeutic efficacy of Bacillus calmette-guerin substrain connaught live antigen can be decreased when used in combination with Maraviroc.
Yellow fever vaccine The therapeutic efficacy of Yellow fever vaccine can be decreased when used in combination with Maraviroc.
Anthrax vaccine The therapeutic efficacy of Anthrax vaccine can be decreased when used in combination with Maraviroc.
Typhoid Vaccine Live The therapeutic efficacy of Typhoid Vaccine Live can be decreased when used in combination with Maraviroc.
BCG vaccine The therapeutic efficacy of BCG vaccine can be decreased when used in combination with Maraviroc.
Human adenovirus e serotype 4 strain cl-68578 antigen The therapeutic efficacy of Human adenovirus e serotype 4 strain cl-68578 antigen can be decreased when used in combination with Maraviroc.
Vibrio cholerae CVD 103-HgR strain live antigen The therapeutic efficacy of Vibrio cholerae CVD 103-HgR strain live antigen can be decreased when used in combination with Maraviroc.
Adenovirus type 7 vaccine live The therapeutic efficacy of Adenovirus type 7 vaccine live can be decreased when used in combination with Maraviroc.
Varicella zoster vaccine (live/attenuated) The therapeutic efficacy of Varicella zoster vaccine (live/attenuated) can be decreased when used in combination with Maraviroc.
Bacillus calmette-guerin substrain russian BCG-I live antigen The therapeutic efficacy of Bacillus calmette-guerin substrain russian BCG-I live antigen can be decreased when used in combination with Maraviroc.
Pexidartinib Maraviroc may increase the hepatotoxic activities of Pexidartinib.
Cenobamate The serum concentration of Maraviroc can be decreased when it is combined with Cenobamate.
Darunavir The serum concentration of Maraviroc can be increased when it is combined with Darunavir.
Haloperidol The serum concentration of Haloperidol can be increased when it is combined with Maraviroc.
Tucatinib The metabolism of Tucatinib can be decreased when combined with Maraviroc.
Abametapir The serum concentration of Maraviroc can be increased when it is combined with Abametapir.
Satralizumab The serum concentration of Maraviroc can be decreased when it is combined with Satralizumab.
Sotorasib The serum concentration of Maraviroc can be decreased when it is combined with Sotorasib.
Ritonavir The metabolism of Maraviroc can be decreased when combined with Ritonavir.
Boceprevir The metabolism of Maraviroc can be decreased when combined with Boceprevir.
Voriconazole The metabolism of Maraviroc can be decreased when combined with Voriconazole.
Ditiocarb The metabolism of Maraviroc can be decreased when combined with Ditiocarb.
Stiripentol The metabolism of Maraviroc can be decreased when combined with Stiripentol.
Danoprevir The metabolism of Maraviroc can be decreased when combined with Danoprevir.
Methimazole The metabolism of Maraviroc can be decreased when combined with Methimazole.
Terfenadine The metabolism of Maraviroc can be decreased when combined with Terfenadine.
Ergotamine The metabolism of Maraviroc can be decreased when combined with Ergotamine.
Delavirdine The metabolism of Maraviroc can be decreased when combined with Delavirdine.
Conivaptan The metabolism of Maraviroc can be decreased when combined with Conivaptan.
Telithromycin The metabolism of Maraviroc can be decreased when combined with Telithromycin.
Ketoconazole The metabolism of Maraviroc can be decreased when combined with Ketoconazole.
Atazanavir The metabolism of Maraviroc can be decreased when combined with Atazanavir.
Nefazodone The metabolism of Maraviroc can be decreased when combined with Nefazodone.
Itraconazole The metabolism of Maraviroc can be decreased when combined with Itraconazole.
Clarithromycin The metabolism of Maraviroc can be decreased when combined with Clarithromycin.
Saquinavir The metabolism of Maraviroc can be decreased when combined with Saquinavir.
Posaconazole The metabolism of Maraviroc can be decreased when combined with Posaconazole.
Lopinavir The metabolism of Maraviroc can be decreased when combined with Lopinavir.
Nilotinib The metabolism of Maraviroc can be decreased when combined with Nilotinib.
Telaprevir The metabolism of Maraviroc can be decreased when combined with Telaprevir.
Midostaurin The metabolism of Maraviroc can be decreased when combined with Midostaurin.
Elvitegravir The metabolism of Maraviroc can be decreased when combined with Elvitegravir.
Ribociclib The metabolism of Maraviroc can be decreased when combined with Ribociclib.
Troleandomycin The metabolism of Maraviroc can be decreased when combined with Troleandomycin.
Lonafarnib The metabolism of Maraviroc can be decreased when combined with Lonafarnib.
Danazol The metabolism of Maraviroc can be decreased when combined with Danazol.
Nelfinavir The metabolism of Maraviroc can be decreased when combined with Nelfinavir.
Indinavir The metabolism of Maraviroc can be decreased when combined with Indinavir.
Amprenavir The metabolism of Maraviroc can be decreased when combined with Amprenavir.
Amiodarone The metabolism of Maraviroc can be decreased when combined with Amiodarone.
Cyclosporine The metabolism of Maraviroc can be decreased when combined with Cyclosporine.
Fluvoxamine The metabolism of Maraviroc can be decreased when combined with Fluvoxamine.
Fluconazole The metabolism of Maraviroc can be decreased when combined with Fluconazole.
Erythromycin The serum concentration of Maraviroc can be increased when it is combined with Erythromycin.
Ziprasidone The metabolism of Maraviroc can be decreased when combined with Ziprasidone.
Isradipine The metabolism of Maraviroc can be decreased when combined with Isradipine.
Diltiazem The metabolism of Maraviroc can be decreased when combined with Diltiazem.
Clozapine The metabolism of Maraviroc can be decreased when combined with Clozapine.
Ciprofloxacin The metabolism of Maraviroc can be decreased when combined with Ciprofloxacin.
Nicardipine The metabolism of Maraviroc can be decreased when combined with Nicardipine.
Verapamil The metabolism of Maraviroc can be decreased when combined with Verapamil.
Aprepitant The metabolism of Maraviroc can be decreased when combined with Aprepitant.
Isoniazid The metabolism of Maraviroc can be decreased when combined with Isoniazid.
Primaquine The metabolism of Maraviroc can be decreased when combined with Primaquine.
Miconazole The metabolism of Maraviroc can be decreased when combined with Miconazole.
Fusidic acid The metabolism of Maraviroc can be decreased when combined with Fusidic acid.
Zimelidine The metabolism of Maraviroc can be decreased when combined with Zimelidine.
Dronedarone The metabolism of Maraviroc can be decreased when combined with Dronedarone.
Milnacipran The metabolism of Maraviroc can be decreased when combined with Milnacipran.
Simeprevir The metabolism of Maraviroc can be decreased when combined with Simeprevir.
Isavuconazonium The metabolism of Maraviroc can be decreased when combined with Isavuconazonium.
Desvenlafaxine The metabolism of Maraviroc can be decreased when combined with Desvenlafaxine.
Nilvadipine The metabolism of Maraviroc can be decreased when combined with Nilvadipine.
Seproxetine The metabolism of Maraviroc can be decreased when combined with Seproxetine.
Linagliptin The metabolism of Maraviroc can be decreased when combined with Linagliptin.
Indalpine The metabolism of Maraviroc can be decreased when combined with Indalpine.
Netupitant The metabolism of Maraviroc can be decreased when combined with Netupitant.
Barnidipine The metabolism of Maraviroc can be decreased when combined with Barnidipine.
Benidipine The metabolism of Maraviroc can be decreased when combined with Benidipine.
Venetoclax The metabolism of Maraviroc can be decreased when combined with Venetoclax.
Isavuconazole The metabolism of Maraviroc can be decreased when combined with Isavuconazole.
Fosnetupitant The metabolism of Maraviroc can be decreased when combined with Fosnetupitant.
Berotralstat The metabolism of Maraviroc can be decreased when combined with Berotralstat.
Tipranavir The metabolism of Maraviroc can be decreased when combined with Tipranavir.
Phenytoin The metabolism of Maraviroc can be increased when combined with Phenytoin.
Pentobarbital The metabolism of Maraviroc can be increased when combined with Pentobarbital.
Carbamazepine The metabolism of Maraviroc can be increased when combined with Carbamazepine.
Mitotane The metabolism of Maraviroc can be increased when combined with Mitotane.
Primidone The metabolism of Maraviroc can be increased when combined with Primidone.
Rifampin The metabolism of Maraviroc can be increased when combined with Rifampicin.
Phenobarbital The metabolism of Maraviroc can be increased when combined with Phenobarbital.
Dexamethasone The metabolism of Maraviroc can be increased when combined with Dexamethasone.
Fosphenytoin The metabolism of Maraviroc can be increased when combined with Fosphenytoin.
St. John's Wort The metabolism of Maraviroc can be increased when combined with St. John's Wort.
Enzalutamide The metabolism of Maraviroc can be increased when combined with Enzalutamide.

Target Protein

C-C chemokine receptor type 5 CCR5

Contoh Produk & Brand

Produk: 40 • International brands: 0
Produk
  • Celsentri
    Tablet • 150 mg • Oral • Canada • Approved
  • Celsentri
    Tablet • 300 mg • Oral • Canada • Approved
  • Celsentri
    Tablet, film coated • 150 mg • Oral • EU • Approved
  • Celsentri
    Tablet, film coated • 150 mg • Oral • EU • Approved
  • Celsentri
    Tablet, film coated • 150 mg • Oral • EU • Approved
  • Celsentri
    Tablet, film coated • 150 mg • Oral • EU • Approved
  • Celsentri
    Tablet, film coated • 150 mg • Oral • EU • Approved
  • Celsentri
    Tablet, film coated • 300 mg • Oral • EU • Approved
Menampilkan 8 dari 40 produk.

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