Peringatan Keamanan

A likely cause of nomifensine toxicity is the aromatic amine group, as compounds containing this chemical substructure are notorious for producing toxic metabolites.

Nomifensine

DB04821

small molecule approved withdrawn

Deskripsi

Nomifensine, formerly marketed as Merital capsules, was associated with an increased incidence of hemolytic anemia. The approved application holder removed Merital capsules from the market on January 23, 1986. FDA published a notice of its determination that Merital capsules were removed from the market for safety reasons (see the Federal Register of June 17, 1986 (51 FR 21981)). Approval of the NDA for Merital capsules was withdrawn on March 20, 1992 (see the Federal Register of March 20, 1992 (57 FR 9729)). Also withdrawn from the Canadian and UK markets.

Struktur Molekul 2D

Berat 238.3275
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

676 Data
Buprenorphine Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Hydrocodone Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Magnesium sulfate The therapeutic efficacy of Nomifensine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Nomifensine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Mirtazapine Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Orphenadrine Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Pramipexole Nomifensine may increase the sedative activities of Pramipexole.
Ropinirole Nomifensine may increase the sedative activities of Ropinirole.
Rotigotine Nomifensine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Nomifensine.
Sodium oxybate Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Thalidomide Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Nomifensine.
Dicoumarol The risk or severity of adverse effects can be increased when Nomifensine is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Nomifensine is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when Nomifensine is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Nomifensine is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Nomifensine is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Nomifensine is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when Nomifensine is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Nomifensine is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Nomifensine is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Nomifensine is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Nomifensine is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Nomifensine is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when Nomifensine is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when Nomifensine is combined with (S)-Warfarin.
Ethanol Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Nomifensine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Fluvoxamine The risk or severity of adverse effects can be increased when Nomifensine is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Nomifensine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Nomifensine is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Nomifensine is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Nomifensine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Nomifensine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Nomifensine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Nomifensine is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Nomifensine is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Nomifensine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Nomifensine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Nomifensine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Nomifensine is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Nomifensine is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Nomifensine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Nomifensine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Nomifensine is combined with Alaproclate.
Zopiclone The risk or severity of adverse effects can be increased when Nomifensine is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Nomifensine.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Nomifensine.
Tryptophan The risk or severity of CNS depression can be increased when Tryptophan is combined with Nomifensine.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Nomifensine.
Lorazepam The risk or severity of CNS depression can be increased when Lorazepam is combined with Nomifensine.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Nomifensine.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Nomifensine.
Reserpine The risk or severity of CNS depression can be increased when Reserpine is combined with Nomifensine.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Nomifensine.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with Nomifensine.
Temazepam The risk or severity of CNS depression can be increased when Temazepam is combined with Nomifensine.
Reboxetine The risk or severity of CNS depression can be increased when Reboxetine is combined with Nomifensine.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with Nomifensine.
Butalbital The risk or severity of CNS depression can be increased when Butalbital is combined with Nomifensine.
Methysergide The risk or severity of CNS depression can be increased when Methysergide is combined with Nomifensine.
Cabergoline The risk or severity of CNS depression can be increased when Cabergoline is combined with Nomifensine.
Phenytoin The risk or severity of CNS depression can be increased when Phenytoin is combined with Nomifensine.
Topiramate The risk or severity of CNS depression can be increased when Topiramate is combined with Nomifensine.
Clemastine The risk or severity of CNS depression can be increased when Clemastine is combined with Nomifensine.
Venlafaxine The risk or severity of CNS depression can be increased when Venlafaxine is combined with Nomifensine.
Etomidate The risk or severity of CNS depression can be increased when Etomidate is combined with Nomifensine.
Morphine The risk or severity of CNS depression can be increased when Morphine is combined with Nomifensine.
Talbutal The risk or severity of CNS depression can be increased when Talbutal is combined with Nomifensine.
Pentobarbital The risk or severity of CNS depression can be increased when Pentobarbital is combined with Nomifensine.
Valproic acid The risk or severity of CNS depression can be increased when Valproic acid is combined with Nomifensine.
Zolmitriptan The risk or severity of CNS depression can be increased when Zolmitriptan is combined with Nomifensine.
Codeine The risk or severity of CNS depression can be increased when Codeine is combined with Nomifensine.
Dihydroergotamine The risk or severity of CNS depression can be increased when Dihydroergotamine is combined with Nomifensine.
Amitriptyline The risk or severity of CNS depression can be increased when Amitriptyline is combined with Nomifensine.
Tolcapone The risk or severity of CNS depression can be increased when Tolcapone is combined with Nomifensine.
Hydromorphone The risk or severity of CNS depression can be increased when Hydromorphone is combined with Nomifensine.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with Nomifensine.
Cetirizine The risk or severity of CNS depression can be increased when Cetirizine is combined with Nomifensine.
Protriptyline The risk or severity of CNS depression can be increased when Protriptyline is combined with Nomifensine.
Trimethadione The risk or severity of CNS depression can be increased when Trimethadione is combined with Nomifensine.
Clobazam The risk or severity of sedation, somnolence, and CNS depression can be increased when Clobazam is combined with Nomifensine.
Chlorzoxazone The risk or severity of CNS depression can be increased when Chlorzoxazone is combined with Nomifensine.
Clozapine The risk or severity of CNS depression can be increased when Clozapine is combined with Nomifensine.
Meprobamate The risk or severity of CNS depression can be increased when Meprobamate is combined with Nomifensine.
Thiethylperazine The risk or severity of CNS depression can be increased when Thiethylperazine is combined with Nomifensine.

Target Protein

D(2) dopamine receptor DRD2
Sodium-dependent noradrenaline transporter SLC6A2
Sodium-dependent dopamine transporter SLC6A3
Amine oxidase [flavin-containing] B MAOB
Amine oxidase [flavin-containing] A MAOA
Myeloperoxidase MPO
Sodium-dependent serotonin transporter SLC6A4
Synaptic vesicular amine transporter SLC18A2

Referensi & Sumber

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