Peringatan Keamanan

Oral TDLO (human): 1.429 mg/kg; Oral TDLO (woman): 2 mg/kg; Oral LD50 (rat): 200 mg/kg; Oral LD50 (mouse): 392 mg/kg

Nimesulide

DB04743

small molecule approved investigational withdrawn

Deskripsi

Nimesulide is a relatively COX-2 selective, non-steroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties. Its approved indications are the treatment of acute pain, the symptomatic treatment of osteoarthritis and primary dysmenorrhoea in adolescents and adults above 12 years old. Due to concerns about the risk of hepatotoxicity, nimesulide has been withdrawn from market in many countries.

Struktur Molekul 2D

Berat 308.31
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 1.8–4.7 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed following oral administration.

Metabolisme

Hepatic. Extensive biotransformation, mainly to 4-hydroxynimesulide (which also appears to be biologically active).

Rute Eliminasi

Renal (50%), fecal (29%)

Interaksi Obat

1831 Data
Apixaban The risk or severity of adverse effects can be increased when Nimesulide is combined with Apixaban.
Dasatinib Dasatinib may increase the anticoagulant activities of Nimesulide.
Ursodeoxycholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Ursodeoxycholic acid.
Glycochenodeoxycholic Acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Glycochenodeoxycholic Acid.
Cholic Acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Cholic Acid.
Glycocholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Glycocholic acid.
Deoxycholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Deoxycholic acid.
Taurocholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Taurocholic acid.
Obeticholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Obeticholic acid.
Chenodeoxycholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Chenodeoxycholic acid.
Taurochenodeoxycholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Taurochenodeoxycholic acid.
Tauroursodeoxycholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Tauroursodeoxycholic acid.
Bamet-UD2 The risk or severity of adverse effects can be increased when Nimesulide is combined with Bamet-UD2.
Dehydrocholic acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Dehydrocholic acid.
Hyodeoxycholic Acid The risk or severity of adverse effects can be increased when Nimesulide is combined with Hyodeoxycholic Acid.
Glucosamine Glucosamine may increase the antiplatelet activities of Nimesulide.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Nimesulide is combined with Ibritumomab tiuxetan.
Ibrutinib The risk or severity of adverse effects can be increased when Ibrutinib is combined with Nimesulide.
Obinutuzumab The risk or severity of adverse effects can be increased when Nimesulide is combined with Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the antiplatelet activities of Nimesulide.
Rivaroxaban Nimesulide may increase the anticoagulant activities of Rivaroxaban.
Tipranavir Tipranavir may increase the antiplatelet activities of Nimesulide.
Urokinase Nimesulide may increase the anticoagulant activities of Urokinase.
Vitamin E Vitamin E may increase the antiplatelet activities of Nimesulide.
Ceritinib Nimesulide may increase the bradycardic activities of Ceritinib.
Ivabradine Nimesulide may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of Nimesulide.
Isoetharine The risk or severity of hypertension can be increased when Isoetharine is combined with Nimesulide.
Zolmitriptan The risk or severity of hypertension can be increased when Zolmitriptan is combined with Nimesulide.
Norepinephrine The risk or severity of hypertension can be increased when Norepinephrine is combined with Nimesulide.
Phenylpropanolamine The risk or severity of hypertension can be increased when Phenylpropanolamine is combined with Nimesulide.
Doxapram The risk or severity of hypertension can be increased when Doxapram is combined with Nimesulide.
Metaraminol The risk or severity of hypertension can be increased when Metaraminol is combined with Nimesulide.
Methoxamine The risk or severity of hypertension can be increased when Methoxamine is combined with Nimesulide.
Isoflurane The risk or severity of hypertension can be increased when Isoflurane is combined with Nimesulide.
Orciprenaline The risk or severity of hypertension can be increased when Orciprenaline is combined with Nimesulide.
Propofol The risk or severity of hypertension can be increased when Propofol is combined with Nimesulide.
Phenmetrazine The risk or severity of hypertension can be increased when Phenmetrazine is combined with Nimesulide.
Pseudoephedrine The risk or severity of hypertension can be increased when Pseudoephedrine is combined with Nimesulide.
Ritodrine The risk or severity of hypertension can be increased when Ritodrine is combined with Nimesulide.
Bitolterol The risk or severity of hypertension can be increased when Bitolterol is combined with Nimesulide.
Oxymetazoline The risk or severity of hypertension can be increased when Oxymetazoline is combined with Nimesulide.
Diethylpropion The risk or severity of hypertension can be increased when Diethylpropion is combined with Nimesulide.
Naratriptan The risk or severity of hypertension can be increased when Naratriptan is combined with Nimesulide.
Formoterol The risk or severity of hypertension can be increased when Formoterol is combined with Nimesulide.
Frovatriptan The risk or severity of hypertension can be increased when Frovatriptan is combined with Nimesulide.
Isoprenaline The risk or severity of hypertension can be increased when Isoprenaline is combined with Nimesulide.
Arbutamine The risk or severity of hypertension can be increased when Arbutamine is combined with Nimesulide.
Desflurane The risk or severity of hypertension can be increased when Desflurane is combined with Nimesulide.
Lisdexamfetamine The risk or severity of hypertension can be increased when Lisdexamfetamine is combined with Nimesulide.
Fenoterol The risk or severity of hypertension can be increased when Fenoterol is combined with Nimesulide.
Pirbuterol The risk or severity of hypertension can be increased when Pirbuterol is combined with Nimesulide.
Ephedra sinica root The risk or severity of hypertension can be increased when Ephedra sinica root is combined with Nimesulide.
Ephedrine The risk or severity of hypertension can be increased when Ephedrine is combined with Nimesulide.
Mephentermine The risk or severity of hypertension can be increased when Mephentermine is combined with Nimesulide.
Procaterol The risk or severity of hypertension can be increased when Procaterol is combined with Nimesulide.
Clenbuterol The risk or severity of hypertension can be increased when Clenbuterol is combined with Nimesulide.
Bambuterol The risk or severity of hypertension can be increased when Bambuterol is combined with Nimesulide.
MMDA The risk or severity of hypertension can be increased when MMDA is combined with Nimesulide.
Midomafetamine The risk or severity of hypertension can be increased when Midomafetamine is combined with Nimesulide.
2,5-Dimethoxy-4-ethylamphetamine The risk or severity of hypertension can be increased when 2,5-Dimethoxy-4-ethylamphetamine is combined with Nimesulide.
4-Methoxyamphetamine The risk or severity of hypertension can be increased when 4-Methoxyamphetamine is combined with Nimesulide.
4-Bromo-2,5-dimethoxyamphetamine The risk or severity of hypertension can be increased when 4-Bromo-2,5-dimethoxyamphetamine is combined with Nimesulide.
Tenamfetamine The risk or severity of hypertension can be increased when Tenamfetamine is combined with Nimesulide.
Chlorphentermine The risk or severity of hypertension can be increased when Chlorphentermine is combined with Nimesulide.
Dextroamphetamine The risk or severity of hypertension can be increased when Dextroamphetamine is combined with Nimesulide.
Phendimetrazine The risk or severity of hypertension can be increased when Phendimetrazine is combined with Nimesulide.
Epicaptopril The risk or severity of hypertension can be increased when Epicaptopril is combined with Nimesulide.
1-benzylimidazole The risk or severity of hypertension can be increased when 1-benzylimidazole is combined with Nimesulide.
Amibegron The risk or severity of hypertension can be increased when Nimesulide is combined with Amibegron.
Naluzotan The risk or severity of hypertension can be increased when Nimesulide is combined with Naluzotan.
Solabegron The risk or severity of hypertension can be increased when Nimesulide is combined with Solabegron.
Esmirtazapine The risk or severity of hypertension can be increased when Nimesulide is combined with Esmirtazapine.
Nitrous oxide The risk or severity of hypertension can be increased when Nimesulide is combined with Nitrous oxide.
Dexmethylphenidate The risk or severity of hypertension can be increased when Nimesulide is combined with Dexmethylphenidate.
Isometheptene The risk or severity of hypertension can be increased when Nimesulide is combined with Isometheptene.
Levonordefrin The risk or severity of hypertension can be increased when Nimesulide is combined with Levonordefrin.
Naphazoline The risk or severity of hypertension can be increased when Nimesulide is combined with Naphazoline.
Tetryzoline The risk or severity of hypertension can be increased when Nimesulide is combined with Tetryzoline.
Cinitapride The risk or severity of hypertension can be increased when Nimesulide is combined with Cinitapride.
Tyramine The risk or severity of hypertension can be increased when Nimesulide is combined with Tyramine.
Adrafinil The risk or severity of hypertension can be increased when Nimesulide is combined with Adrafinil.
Isoxsuprine The risk or severity of hypertension can be increased when Nimesulide is combined with Isoxsuprine.
Ifenprodil The risk or severity of hypertension can be increased when Nimesulide is combined with Ifenprodil.
Hexoprenaline The risk or severity of hypertension can be increased when Nimesulide is combined with Hexoprenaline.
Etilefrine The risk or severity of hypertension can be increased when Nimesulide is combined with Etilefrine.
Olodaterol The risk or severity of hypertension can be increased when Nimesulide is combined with Olodaterol.
Cirazoline The risk or severity of hypertension can be increased when Nimesulide is combined with Cirazoline.
Synephrine The risk or severity of hypertension can be increased when Nimesulide is combined with Synephrine.
Doxofylline The risk or severity of hypertension can be increased when Nimesulide is combined with Doxofylline.
Iofetamine I-123 The risk or severity of hypertension can be increased when Nimesulide is combined with Iofetamine I-123.
Racepinephrine The risk or severity of hypertension can be increased when Nimesulide is combined with Racepinephrine.
Amitraz The risk or severity of hypertension can be increased when Nimesulide is combined with Amitraz.
Medetomidine The risk or severity of hypertension can be increased when Nimesulide is combined with Medetomidine.
Xylazine The risk or severity of hypertension can be increased when Nimesulide is combined with Xylazine.
Atipamezole The risk or severity of hypertension can be increased when Nimesulide is combined with Atipamezole.
Ractopamine The risk or severity of hypertension can be increased when Nimesulide is combined with Ractopamine.
Romifidine The risk or severity of hypertension can be increased when Nimesulide is combined with Romifidine.
Detomidine The risk or severity of hypertension can be increased when Nimesulide is combined with Detomidine.
Tetrahydrocannabivarin The risk or severity of hypertension can be increased when Nimesulide is combined with Tetrahydrocannabivarin.

Target Protein

Prostaglandin G/H synthase 2 PTGS2
Tumor necrosis factor ligand superfamily member 10 TNFSF10
Lactotransferrin LTF
Group IIE secretory phospholipase A2 PLA2G2E

Referensi & Sumber

Synthesis reference: Bernard Pirotte, Geraldine Piel, Philippe Neven, Isabelle Delneuville, Joszef Geczy, "Water-soluble nimesulide salt and its preparation, aqueous dolution containing it, nimesulide-based combinations and their uses." U.S. Patent US5756546, issued November, 1991.

Contoh Produk & Brand

Produk: 0 • International brands: 8
International Brands
  • Ainex
  • Aulin
  • Eskaflam
  • Mesulid
  • Nilsid
  • Nimalox
  • Nise
  • Sulide

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul